JP4563387B2 - 精神病の処置のためのグリシン取り込み阻害剤としての１−ベンゾイル−ピペラジン誘導体 - Google Patents

精神病の処置のためのグリシン取り込み阻害剤としての１−ベンゾイル−ピペラジン誘導体 Download PDF

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JP4563387B2
JP4563387B2 JP2006525700A JP2006525700A JP4563387B2 JP 4563387 B2 JP4563387 B2 JP 4563387B2 JP 2006525700 A JP2006525700 A JP 2006525700A JP 2006525700 A JP2006525700 A JP 2006525700A JP 4563387 B2 JP4563387 B2 JP 4563387B2
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phenyl
piperazine
fluoro
methanesulfonyl
piperazin
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JP2007505062A (ja
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アルベラティ−ジャンニ，ダニエーラ
ヨリドン，ジネーゼ
ナルキジアン，ロベール
ネッテコフェン，マサイアス・ハインリヒ
ノークロス，ロジャー・ディヴィッド
ピナール，エマニュエル
スタルダー，ヘンリ
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F Hoffmann La Roche AG
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    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/10—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms
    • C07D295/104—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms with the ring nitrogen atoms and the doubly bound oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
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JP2006525700A 2003-09-09 2004-08-31 精神病の処置のためのグリシン取り込み阻害剤としての１−ベンゾイル−ピペラジン誘導体 Active JP4563387B2 (ja)

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EP03019682 2003-09-09
PCT/EP2004/009699 WO2005023261A1 (en) 2003-09-09 2004-08-31 1-benzoyl-piperazine derivatives as glycine uptake inhibitors for the treatment of psychoses

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KR20060087550A (ko) 2006-08-02
CA2538135A1 (en) 2005-03-17
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AU2004269892A1 (en) 2005-03-17
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