JP3126775B2 - 環状アミンの光学分割法と該方法によって得られた光学活性体 - Google Patents

環状アミンの光学分割法と該方法によって得られた光学活性体

Info

Publication number
JP3126775B2
JP3126775B2 JP03321290A JP32129091A JP3126775B2 JP 3126775 B2 JP3126775 B2 JP 3126775B2 JP 03321290 A JP03321290 A JP 03321290A JP 32129091 A JP32129091 A JP 32129091A JP 3126775 B2 JP3126775 B2 JP 3126775B2
Authority
JP
Japan
Prior art keywords
optical resolution
compound
methylamino
formula
methylenepyrrolidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
JP03321290A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0532621A (ja
Inventor
哲夫 岡田
忠彦 津島
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Shionogi and Co Ltd
Original Assignee
Shionogi and Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi and Co Ltd filed Critical Shionogi and Co Ltd
Publication of JPH0532621A publication Critical patent/JPH0532621A/ja
Application granted granted Critical
Publication of JP3126775B2 publication Critical patent/JP3126775B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP03321290A 1990-11-21 1991-11-08 環状アミンの光学分割法と該方法によって得られた光学活性体 Expired - Fee Related JP3126775B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2-319107 1990-11-21
JP31910790 1990-11-21

Publications (2)

Publication Number Publication Date
JPH0532621A JPH0532621A (ja) 1993-02-09
JP3126775B2 true JP3126775B2 (ja) 2001-01-22

Family

ID=18106542

Family Applications (1)

Application Number Title Priority Date Filing Date
JP03321290A Expired - Fee Related JP3126775B2 (ja) 1990-11-21 1991-11-08 環状アミンの光学分割法と該方法によって得られた光学活性体

Country Status (5)

Country Link
EP (1) EP0487030A3 (enExample)
JP (1) JP3126775B2 (enExample)
KR (1) KR920009790A (enExample)
DK (1) DK0487030T3 (enExample)
TW (1) TW230770B (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7902227B2 (en) * 2007-07-27 2011-03-08 Janssen Pharmaceutica Nv. C-7 isoxazolinyl quinolone / naphthyridine derivatives useful as antibacterial agents

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4111951A (en) * 1977-01-17 1978-09-05 Hoffmann-La Roche Inc. Process for L-3,4-dehydroproline
CA1332605C (en) * 1988-10-03 1994-10-18 Yasuhiro Nishitani Pyridonecarboxylic acids

Also Published As

Publication number Publication date
DK0487030T3 (da) 1992-11-19
JPH0532621A (ja) 1993-02-09
KR920009790A (ko) 1992-06-25
EP0487030A2 (en) 1992-05-27
TW230770B (enExample) 1994-09-21
EP0487030A3 (en) 1992-11-19

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Legal Events

Date Code Title Description
LAPS Cancellation because of no payment of annual fees