JP2670545B2 - 新規な方法及び中間体類 - Google Patents

新規な方法及び中間体類

Info

Publication number
JP2670545B2
JP2670545B2 JP1016543A JP1654389A JP2670545B2 JP 2670545 B2 JP2670545 B2 JP 2670545B2 JP 1016543 A JP1016543 A JP 1016543A JP 1654389 A JP1654389 A JP 1654389A JP 2670545 B2 JP2670545 B2 JP 2670545B2
Authority
JP
Japan
Prior art keywords
methyl
methoxy
reaction
reacting
product
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP1016543A
Other languages
English (en)
Japanese (ja)
Other versions
JPH021471A (ja
Inventor
コルブ ミッシェル
ヴァン ハイフティー ラック
Original Assignee
メレルダウファ―マス―ティカルズ インコーポレーテッド
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by メレルダウファ―マス―ティカルズ インコーポレーテッド filed Critical メレルダウファ―マス―ティカルズ インコーポレーテッド
Publication of JPH021471A publication Critical patent/JPH021471A/ja
Application granted granted Critical
Publication of JP2670545B2 publication Critical patent/JP2670545B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C43/00—Ethers; Compounds having groups, groups or groups
    • C07C43/02—Ethers
    • C07C43/03—Ethers having all ether-oxygen atoms bound to acyclic carbon atoms
    • C07C43/14—Unsaturated ethers
    • C07C43/178—Unsaturated ethers containing hydroxy or O-metal groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C405/00—Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C43/00—Ethers; Compounds having groups, groups or groups
    • C07C43/02—Ethers
    • C07C43/03—Ethers having all ether-oxygen atoms bound to acyclic carbon atoms
    • C07C43/14—Unsaturated ethers
    • C07C43/178—Unsaturated ethers containing hydroxy or O-metal groups
    • C07C43/1782—Unsaturated ethers containing hydroxy or O-metal groups containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/10—Oxygen atoms
    • C07D309/12—Oxygen atoms only hydrogen atoms and one oxygen atom directly attached to ring carbon atoms, e.g. tetrahydropyranyl ethers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F1/00—Compounds containing elements of Groups 1 or 11 of the Periodic Table
    • C07F1/02—Lithium compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F1/00—Compounds containing elements of Groups 1 or 11 of the Periodic Table
    • C07F1/08—Copper compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/22—Tin compounds
    • C07F7/2208—Compounds having tin linked only to carbon, hydrogen and/or halogen
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Materials Engineering (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrane Compounds (AREA)
JP1016543A 1988-01-28 1989-01-27 新規な方法及び中間体類 Expired - Lifetime JP2670545B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP88400199A EP0325869B1 (en) 1988-01-28 1988-01-28 Novel processes and intermediates
EP88400199,1 1988-01-28

Publications (2)

Publication Number Publication Date
JPH021471A JPH021471A (ja) 1990-01-05
JP2670545B2 true JP2670545B2 (ja) 1997-10-29

Family

ID=8200346

Family Applications (1)

Application Number Title Priority Date Filing Date
JP1016543A Expired - Lifetime JP2670545B2 (ja) 1988-01-28 1989-01-27 新規な方法及び中間体類

Country Status (13)

Country Link
US (1) US5055592A (enExample)
EP (1) EP0325869B1 (enExample)
JP (1) JP2670545B2 (enExample)
KR (1) KR0141104B1 (enExample)
AT (1) ATE82748T1 (enExample)
CA (1) CA1308100C (enExample)
DE (1) DE3876230T2 (enExample)
DK (1) DK36689A (enExample)
ES (1) ES2052750T3 (enExample)
GR (1) GR3006806T3 (enExample)
HU (2) HU203885B (enExample)
IL (1) IL89048A (enExample)
ZA (1) ZA89551B (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2917552B2 (ja) * 1991-02-26 1999-07-12 史衛 佐藤 α−メチレンシクロペンタノン誘導体の製造法
IT1402047B1 (it) * 2010-10-19 2013-08-28 Cross Pharma Sa Uso del mexiprostil nel trattamento delle malattie infiammatorie intestinali

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1162731B (it) * 1979-04-10 1987-04-01 Lepetit Spa 16-metil-16-metossi-5,6-diidro-prosta-glandine della serie e1 ad attivita'antisecretoria
DE3275542D1 (en) * 1981-11-13 1987-04-09 Teijin Ltd Process for prostaglandin e1, production and novel delta 7-prostaglandines e and 7-hydroxyprostaglandins e
EP0215949B1 (en) * 1985-01-29 1990-07-04 Teijin Limited Process for preparing 16-substituted prostaglandin e's

Also Published As

Publication number Publication date
KR0141104B1 (ko) 1998-07-01
DK36689A (da) 1989-07-29
ATE82748T1 (de) 1992-12-15
DE3876230D1 (de) 1993-01-07
HU200751B (en) 1990-08-28
KR890011839A (ko) 1989-08-22
ZA89551B (en) 1990-01-31
ES2052750T3 (es) 1994-07-16
DK36689D0 (da) 1989-01-27
IL89048A (en) 1993-06-10
US5055592A (en) 1991-10-08
HU902026D0 (en) 1990-08-28
DE3876230T2 (de) 1993-05-06
JPH021471A (ja) 1990-01-05
GR3006806T3 (enExample) 1993-06-30
EP0325869A1 (en) 1989-08-02
HUT49120A (en) 1989-08-28
CA1308100C (en) 1992-09-29
HU203885B (en) 1991-10-28
EP0325869B1 (en) 1992-11-25

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