JP2025508192A5 - - Google Patents

Info

Publication number
JP2025508192A5
JP2025508192A5 JP2024554912A JP2024554912A JP2025508192A5 JP 2025508192 A5 JP2025508192 A5 JP 2025508192A5 JP 2024554912 A JP2024554912 A JP 2024554912A JP 2024554912 A JP2024554912 A JP 2024554912A JP 2025508192 A5 JP2025508192 A5 JP 2025508192A5
Authority
JP
Japan
Prior art keywords
hydrocarbyl
membered
general formula
optionally substituted
halohydrocarbyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024554912A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025508192A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CN2023/080775 external-priority patent/WO2023174175A1/zh
Publication of JP2025508192A publication Critical patent/JP2025508192A/ja
Publication of JP2025508192A5 publication Critical patent/JP2025508192A5/ja
Pending legal-status Critical Current

Links

JP2024554912A 2022-03-17 2023-03-10 Kif18a阻害剤 Pending JP2025508192A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN202210266719.4 2022-03-17
CN202210266719 2022-03-17
PCT/CN2023/080775 WO2023174175A1 (zh) 2022-03-17 2023-03-10 Kif18a抑制剂

Publications (2)

Publication Number Publication Date
JP2025508192A JP2025508192A (ja) 2025-03-21
JP2025508192A5 true JP2025508192A5 (https=) 2026-03-18

Family

ID=88022235

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024554912A Pending JP2025508192A (ja) 2022-03-17 2023-03-10 Kif18a阻害剤

Country Status (7)

Country Link
US (1) US20250197382A1 (https=)
EP (1) EP4495113A4 (https=)
JP (1) JP2025508192A (https=)
CN (1) CN118613478A (https=)
AU (1) AU2023236101A1 (https=)
CA (1) CA3246028A1 (https=)
WO (1) WO2023174175A1 (https=)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20250027560A (ko) * 2022-06-30 2025-02-26 쑤저우 젠하우스 바이오 컴퍼니 리미티드 질소 함유 화합물 및 이의 용도
WO2024022508A1 (zh) * 2022-07-29 2024-02-01 武汉人福创新药物研发中心有限公司 Kif18a抑制剂及用途
TW202416973A (zh) 2022-08-18 2024-05-01 美商雅客森醫療公司 Kif18a抑制劑及其用途
KR20250044780A (ko) * 2022-09-08 2025-04-01 장춘 진사이언스 파마슈티컬 씨오., 엘티디. Kif18a 억제제 화합물, 약제학적 조성물 및 이의 제조 방법과 적용
CN119907796A (zh) * 2022-09-09 2025-04-29 海南先声再明医药股份有限公司 酰胺类化合物、其组合物及用途
CN119562952A (zh) * 2022-09-30 2025-03-04 山东轩竹医药科技有限公司 Kif18a抑制剂
WO2024083208A1 (zh) * 2022-10-21 2024-04-25 杭州邦顺制药有限公司 Kif18a蛋白抑制剂
JP2025538601A (ja) * 2022-11-24 2025-11-28 インベンティスバイオ カンパニー リミテッド 複素環化合物、その製造方法および用途
EP4628486A1 (en) * 2022-12-02 2025-10-08 Shenzhen Zhongge Biological Technology Co., Ltd. Amide or urea compound
CN120641408A (zh) * 2022-12-16 2025-09-12 抟相医药(上海)有限公司 含氮化合物、药物组合物及其用途
WO2024140799A1 (en) * 2022-12-28 2024-07-04 Insilico Medicine Ip Limited Inhibitors of kif18a and uses thereof
WO2024149189A1 (zh) * 2023-01-09 2024-07-18 浙江海正药业股份有限公司 芳香酰胺类衍生物及其制备方法和用途
JP2026509288A (ja) * 2023-03-10 2026-03-17 浙江海正薬業股▲ふん▼有限公司 芳香族アミド誘導体、その製造方法、およびその使用
WO2024217348A1 (zh) * 2023-04-18 2024-10-24 南京同诺康医药科技有限公司 Kif18a抑制剂及其制备方法和用途
WO2025167861A1 (zh) * 2024-02-06 2025-08-14 上海齐鲁制药研究中心有限公司 螺环kif18a抑制剂
WO2025190364A1 (zh) * 2024-03-14 2025-09-18 山东轩竹医药科技有限公司 Kif18a抑制剂及其用途
WO2025201531A1 (zh) * 2024-03-29 2025-10-02 深圳众格生物科技有限公司 三环类化合物及其用途
WO2025242166A1 (en) * 2024-05-22 2025-11-27 InventisBio Co., Ltd. Heterocyclic compounds, preparation methods and uses thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MA54543A (fr) * 2018-12-20 2022-03-30 Amgen Inc Inhibiteurs de kif18a
AU2019401495B2 (en) * 2018-12-20 2025-06-26 Amgen Inc. Heteroaryl amides useful as KIF18A inhibitors
JP7686559B2 (ja) * 2018-12-20 2025-06-02 アムジエン・インコーポレーテツド Kif18a阻害剤
EP4007638A1 (en) * 2019-08-02 2022-06-08 Amgen Inc. Pyridine derivatives as kif18a inhibitors
EP4007752B1 (en) * 2019-08-02 2025-09-24 Amgen Inc. Kif18a inhibitors
EP4007753B1 (en) * 2019-08-02 2025-09-24 Amgen Inc. Kif18a inhibitors
MX2022012992A (es) * 2020-04-14 2022-11-08 Amgen Inc Inhibidores de kif18a para el tratamiento de enfermedades neoplasicas.
TW202400582A (zh) * 2022-05-13 2024-01-01 大陸商上海湃隆生物科技有限公司 驅動蛋白kif18a抑制劑及其應用

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