JP2023528421A5 - - Google Patents

Info

Publication number
JP2023528421A5
JP2023528421A5 JP2022574229A JP2022574229A JP2023528421A5 JP 2023528421 A5 JP2023528421 A5 JP 2023528421A5 JP 2022574229 A JP2022574229 A JP 2022574229A JP 2022574229 A JP2022574229 A JP 2022574229A JP 2023528421 A5 JP2023528421 A5 JP 2023528421A5
Authority
JP
Japan
Prior art keywords
compound
membered
pharmaceutically acceptable
compound according
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022574229A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023528421A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/035509 external-priority patent/WO2021247748A1/en
Publication of JP2023528421A publication Critical patent/JP2023528421A/ja
Publication of JP2023528421A5 publication Critical patent/JP2023528421A5/ja
Priority to JP2025207773A priority Critical patent/JP2026048716A/ja
Pending legal-status Critical Current

Links

JP2022574229A 2020-06-02 2021-06-02 キナーゼ阻害剤 Pending JP2023528421A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025207773A JP2026048716A (ja) 2020-06-02 2025-11-28 キナーゼ阻害剤

Applications Claiming Priority (13)

Application Number Priority Date Filing Date Title
US202063033728P 2020-06-02 2020-06-02
US202063033724P 2020-06-02 2020-06-02
US202063033729P 2020-06-02 2020-06-02
US63/033,729 2020-06-02
US63/033,724 2020-06-02
US63/033,728 2020-06-02
US202163136587P 2021-01-12 2021-01-12
US202163136593P 2021-01-12 2021-01-12
US202163136577P 2021-01-12 2021-01-12
US63/136,587 2021-01-12
US63/136,593 2021-01-12
US63/136,577 2021-01-12
PCT/US2021/035509 WO2021247748A1 (en) 2020-06-02 2021-06-02 Kinase inhibitors

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025207773A Division JP2026048716A (ja) 2020-06-02 2025-11-28 キナーゼ阻害剤

Publications (2)

Publication Number Publication Date
JP2023528421A JP2023528421A (ja) 2023-07-04
JP2023528421A5 true JP2023528421A5 (https=) 2024-06-10

Family

ID=76601840

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022574229A Pending JP2023528421A (ja) 2020-06-02 2021-06-02 キナーゼ阻害剤
JP2025207773A Pending JP2026048716A (ja) 2020-06-02 2025-11-28 キナーゼ阻害剤

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025207773A Pending JP2026048716A (ja) 2020-06-02 2025-11-28 キナーゼ阻害剤

Country Status (7)

Country Link
US (1) US12448363B2 (https=)
EP (1) EP4157446A1 (https=)
JP (2) JP2023528421A (https=)
CN (1) CN115867346B (https=)
AU (1) AU2021283916A1 (https=)
CA (1) CA3179637A1 (https=)
WO (1) WO2021247748A1 (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2021398051A1 (en) 2020-12-10 2023-07-27 Principia Biopharma Inc. Crystal form of tolebrutinib, preparation method therefor and use thereof
US20240383871A1 (en) * 2021-08-30 2024-11-21 Bristol-Myers Squibb Company Compound useful for pet-imaging of bruton’s tyrosine kinase
WO2023227080A1 (zh) * 2022-05-25 2023-11-30 百极弘烨(南通)医药科技有限公司 一种protac化合物、含其的药物组合物及其制备方法和应用
CA3259743A1 (en) * 2022-06-22 2023-12-28 Principia Biopharma Inc. METHODS FOR MANUFACTURING MODIFIED BTK INHIBITORS
CN116284025B (zh) * 2023-02-20 2025-07-04 国科大杭州高等研究院 一种具有抗癌作用的螺杂环类化合物、药物组合物及其用途

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014210255A1 (en) * 2013-06-26 2014-12-31 Abbvie Inc. Primary carboxamides as btk inhibitors
RS59707B1 (sr) 2014-10-24 2020-01-31 Bristol Myers Squibb Co Derivati karbazola
PE20190710A1 (es) * 2014-10-24 2019-05-17 Bristol Myers Squibb Co Compuestos de indol carboxamida utiles como inhibidores de cinasas

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