JP2024536869A5 - - Google Patents

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Publication number
JP2024536869A5
JP2024536869A5 JP2024518884A JP2024518884A JP2024536869A5 JP 2024536869 A5 JP2024536869 A5 JP 2024536869A5 JP 2024518884 A JP2024518884 A JP 2024518884A JP 2024518884 A JP2024518884 A JP 2024518884A JP 2024536869 A5 JP2024536869 A5 JP 2024536869A5
Authority
JP
Japan
Prior art keywords
alkyl
cycloalkyl
pharmaceutically acceptable
unsubstituted
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024518884A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024536869A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/077001 external-priority patent/WO2023049887A1/en
Publication of JP2024536869A publication Critical patent/JP2024536869A/ja
Publication of JP2024536869A5 publication Critical patent/JP2024536869A5/ja
Pending legal-status Critical Current

Links

JP2024518884A 2021-09-27 2022-09-26 イミダゾピリダジンil-17阻害剤化合物 Pending JP2024536869A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US202163248566P 2021-09-27 2021-09-27
US63/248,566 2021-09-27
US202163273422P 2021-10-29 2021-10-29
US63/273,422 2021-10-29
US202263367546P 2022-07-01 2022-07-01
US63/367,546 2022-07-01
PCT/US2022/077001 WO2023049887A1 (en) 2021-09-27 2022-09-26 Imidazopyridazine il-17 inhibitor compounds

Publications (2)

Publication Number Publication Date
JP2024536869A JP2024536869A (ja) 2024-10-08
JP2024536869A5 true JP2024536869A5 (https=) 2025-09-19

Family

ID=83692741

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024518884A Pending JP2024536869A (ja) 2021-09-27 2022-09-26 イミダゾピリダジンil-17阻害剤化合物

Country Status (16)

Country Link
US (2) US12173007B2 (https=)
EP (1) EP4408847A1 (https=)
JP (1) JP2024536869A (https=)
KR (1) KR20240082369A (https=)
AU (1) AU2022349687A1 (https=)
CA (1) CA3233408A1 (https=)
CL (1) CL2024000867A1 (https=)
CO (1) CO2024003723A2 (https=)
DO (1) DOP2024000051A (https=)
IL (1) IL311751A (https=)
JO (1) JOP20240059A1 (https=)
MX (1) MX2024003772A (https=)
PE (1) PE20240935A1 (https=)
TW (1) TW202330530A (https=)
UY (1) UY39958A (https=)
WO (1) WO2023049887A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL311751A (en) 2021-09-27 2024-05-01 Janssen Pharmaceutica Nv IL-17 imidazopyridazine inhibitory compounds
CN118401519A (zh) 2021-10-25 2024-07-26 拓臻制药公司 作为glp-1r激动剂的化合物
TW202430165A (zh) 2022-12-02 2024-08-01 丹麥商理奧藥品公司 Il-17之小分子調節劑
CN120731202A (zh) * 2023-01-30 2025-09-30 戴斯阿尔法公司 基于苯并咪唑和氮杂-苯并咪唑的il-17a调节剂及其用途
CN121311483A (zh) * 2023-03-28 2026-01-09 詹森药业有限公司 含内酰胺的咪唑并哒嗪il-17抑制剂化合物
EP4568664B1 (en) 2023-04-07 2026-04-01 Terns Pharmaceuticals, Inc. Combination comprising a thr-beta agonist and a glp-1r agonist for use in treating obesity
WO2024215597A1 (en) * 2023-04-11 2024-10-17 Dice Alpha, Inc. Substituted 6-imidazopyridazine il-17a modulators and uses thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI752400B (zh) 2019-01-07 2022-01-11 美商美國禮來大藥廠 Il-17a抑制劑
GB201909190D0 (en) 2019-06-26 2019-08-07 Ucb Biopharma Sprl Therapeutic agents
PE20230469A1 (es) 2020-04-30 2023-03-14 Janssen Pharmaceutica Nv Imidazopiridazinas como moduladores de il-17
WO2023025783A1 (en) 2021-08-23 2023-03-02 Leo Pharma A/S Small molecule modulators of il-17
IL311751A (en) 2021-09-27 2024-05-01 Janssen Pharmaceutica Nv IL-17 imidazopyridazine inhibitory compounds
CN116143777A (zh) 2021-11-04 2023-05-23 四川海思科制药有限公司 一种可抑制il-17a的杂环化合物及其用途

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