JP2024522990A5 - - Google Patents
Info
- Publication number
- JP2024522990A5 JP2024522990A5 JP2023574150A JP2023574150A JP2024522990A5 JP 2024522990 A5 JP2024522990 A5 JP 2024522990A5 JP 2023574150 A JP2023574150 A JP 2023574150A JP 2023574150 A JP2023574150 A JP 2023574150A JP 2024522990 A5 JP2024522990 A5 JP 2024522990A5
- Authority
- JP
- Japan
- Prior art keywords
- mixtures
- tautomers
- item
- enantiomers
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202163195930P | 2021-06-02 | 2021-06-02 | |
| US63/195,930 | 2021-06-02 | ||
| US202163275113P | 2021-11-03 | 2021-11-03 | |
| US63/275,113 | 2021-11-03 | ||
| PCT/US2022/031815 WO2022256434A1 (en) | 2021-06-02 | 2022-06-01 | Protease inhibitors as antivirals |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024522990A JP2024522990A (ja) | 2024-06-25 |
| JP2024522990A5 true JP2024522990A5 (https=) | 2025-06-10 |
Family
ID=82321542
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023574150A Pending JP2024522990A (ja) | 2021-06-02 | 2022-06-01 | 抗ウイルス薬としてのプロテアーゼ阻害剤 |
Country Status (11)
| Country | Link |
|---|---|
| US (3) | US11753373B2 (https=) |
| EP (1) | EP4347034A1 (https=) |
| JP (1) | JP2024522990A (https=) |
| KR (1) | KR20240057384A (https=) |
| AU (1) | AU2022283816A1 (https=) |
| BR (1) | BR112023025358A2 (https=) |
| CA (1) | CA3220847A1 (https=) |
| IL (1) | IL308694A (https=) |
| MX (1) | MX2023014307A (https=) |
| TW (1) | TW202313567A (https=) |
| WO (1) | WO2022256434A1 (https=) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20220033383A1 (en) * | 2020-07-20 | 2022-02-03 | Enanta Pharmaceuticals, Inc. | Functionalized peptides as antiviral agents |
| KR20230124583A (ko) | 2020-11-23 | 2023-08-25 | 이난타 파마슈티칼스, 인코포레이티드 | 신규한 스피로피롤리딘 유래 항바이러스제 |
| US12540141B2 (en) | 2020-11-23 | 2026-02-03 | Enanta Pharmaceuticals, Inc. | Spiropyrrolidine derived antiviral agents |
| CA3200437A1 (en) * | 2020-12-01 | 2022-06-09 | Arun K. Ghosh | Compounds for the treatment of sars |
| US12398147B2 (en) | 2021-05-11 | 2025-08-26 | Enanta Pharmaceuticals, Inc. | Macrocyclic spiropyrrolidine derived antiviral agents |
| WO2022256434A1 (en) | 2021-06-02 | 2022-12-08 | ACEA Therapeutics, Inc. | Protease inhibitors as antivirals |
| US12479854B2 (en) | 2021-07-29 | 2025-11-25 | Enanta Pharmaceuticals, Inc. | Spiropyrrolidine derived antiviral agents |
| CN118302421A (zh) * | 2021-11-26 | 2024-07-05 | 海南先声药业有限公司 | 一种吡咯烷类抗病毒化合物 |
| US12145941B2 (en) | 2021-12-08 | 2024-11-19 | Enanta Pharmaceuticals, Inc. | Heterocyclic antiviral agents |
| TW202334123A (zh) * | 2021-12-31 | 2023-09-01 | 大陸商蘇州愛科百發生物醫藥技術有限公司 | 用於預防和治療冠狀病毒感染的化合物及其偶聯物和方法 |
| CN118451090A (zh) * | 2022-01-13 | 2024-08-06 | 海南先声药业有限公司 | 一种酰胺类抗病毒化合物 |
| WO2023196307A1 (en) | 2022-04-05 | 2023-10-12 | Enanta Pharmaceuticals, Inc. | Novel spiropyrrolidine derived antiviral agents |
| CN116535460A (zh) * | 2023-04-28 | 2023-08-04 | 中国人民解放军军事科学院军事医学研究院 | 一类含硫拟肽类化合物及其制备方法和用途 |
| WO2024237816A1 (ru) * | 2023-05-12 | 2024-11-21 | Общество С Ограниченной Ответственностью "Промомед Рус" | Новые производные азабициклогексана |
| CN119306790A (zh) * | 2023-07-13 | 2025-01-14 | 深圳市塔吉瑞生物医药有限公司 | 酰胺衍生物及其组合物及用途 |
| EP4686470A1 (en) | 2024-08-01 | 2026-02-04 | Ospedale San Raffaele S.r.l. | Macrocyclic peptidomimetics as antiviral agents |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1704142A4 (en) * | 2003-12-31 | 2008-08-20 | Taigen Biotechnology Co Ltd | PROTEASE INHIBITORS |
| WO2005113580A1 (en) * | 2004-05-21 | 2005-12-01 | Pfizer Inc. | Anticoronviral compounds and compositions, their pharmaceutical uses and materials for their synthesis |
| WO2006061714A2 (en) * | 2004-12-09 | 2006-06-15 | Pfizer Inc. | Anticoronaviral compounds and compositions, their pharmaceutical uses and materials for their synthesis |
| CN110818691A (zh) | 2018-08-09 | 2020-02-21 | 中国科学院上海药物研究所 | 酮酰胺类化合物及其制备方法、药物组合物和用途 |
| CN113939267B (zh) | 2019-06-05 | 2025-11-11 | 法国特种经营公司 | 口腔护理组合物 |
| BR112021024310A2 (pt) | 2019-06-05 | 2022-02-15 | Univ Emory | Peptidomiméticos para o tratamento de infecções por coronavírus e picornavírus |
| WO2021205296A1 (en) | 2020-04-05 | 2021-10-14 | Pfizer Inc. | Method of treating covid-19 |
| AU2021254045A1 (en) * | 2020-04-10 | 2022-10-13 | Cocrystal Pharma, Inc. | Inhibitors of norovirus and coronavirus replication |
| US11124497B1 (en) * | 2020-04-17 | 2021-09-21 | Pardes Biosciences, Inc. | Inhibitors of cysteine proteases and methods of use thereof |
| BR112022021381A2 (pt) * | 2020-04-23 | 2022-12-06 | Purdue Research Foundation | Compostos para o tratamento de sars |
| BR112021023814A2 (pt) * | 2020-06-09 | 2022-12-20 | Pardes Biosciences Inc | Inibidores de proteases de cisteína e métodos de uso das mesmas |
| MX2023001756A (es) * | 2020-08-13 | 2023-05-04 | Enanta Pharm Inc | Peptidos funcionalizados como agentes antivirales. |
| US11351149B2 (en) * | 2020-09-03 | 2022-06-07 | Pfizer Inc. | Nitrile-containing antiviral compounds |
| WO2022256434A1 (en) | 2021-06-02 | 2022-12-08 | ACEA Therapeutics, Inc. | Protease inhibitors as antivirals |
-
2022
- 2022-06-01 WO PCT/US2022/031815 patent/WO2022256434A1/en not_active Ceased
- 2022-06-01 CA CA3220847A patent/CA3220847A1/en active Pending
- 2022-06-01 JP JP2023574150A patent/JP2024522990A/ja active Pending
- 2022-06-01 TW TW111120433A patent/TW202313567A/zh unknown
- 2022-06-01 US US17/830,185 patent/US11753373B2/en active Active
- 2022-06-01 BR BR112023025358A patent/BR112023025358A2/pt unknown
- 2022-06-01 IL IL308694A patent/IL308694A/en unknown
- 2022-06-01 EP EP22735725.8A patent/EP4347034A1/en active Pending
- 2022-06-01 KR KR1020237045446A patent/KR20240057384A/ko active Pending
- 2022-06-01 MX MX2023014307A patent/MX2023014307A/es unknown
- 2022-06-01 AU AU2022283816A patent/AU2022283816A1/en active Pending
-
2023
- 2023-06-15 US US18/210,555 patent/US11987554B2/en active Active
-
2024
- 2024-04-22 US US18/642,453 patent/US20250122153A1/en active Pending
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