JP2023533855A5 - - Google Patents

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Publication number
JP2023533855A5
JP2023533855A5 JP2023502881A JP2023502881A JP2023533855A5 JP 2023533855 A5 JP2023533855 A5 JP 2023533855A5 JP 2023502881 A JP2023502881 A JP 2023502881A JP 2023502881 A JP2023502881 A JP 2023502881A JP 2023533855 A5 JP2023533855 A5 JP 2023533855A5
Authority
JP
Japan
Prior art keywords
compound
pharmaceutically acceptable
formula
acceptable salt
solvate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023502881A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023533855A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/034599 external-priority patent/WO2022015423A1/en
Publication of JP2023533855A publication Critical patent/JP2023533855A/ja
Publication of JP2023533855A5 publication Critical patent/JP2023533855A5/ja
Pending legal-status Critical Current

Links

JP2023502881A 2020-07-16 2021-05-27 イソキノリン化合物およびそのAhR不均衡の治療への使用 Pending JP2023533855A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202063052574P 2020-07-16 2020-07-16
US202063052561P 2020-07-16 2020-07-16
US63/052,574 2020-07-16
US63/052,561 2020-07-16
PCT/US2021/034599 WO2022015423A1 (en) 2020-07-16 2021-05-27 ISOQUINOLINE COMPOUNDS AND THEIR USE IN TREATING AhR IMBALANCE

Publications (2)

Publication Number Publication Date
JP2023533855A JP2023533855A (ja) 2023-08-04
JP2023533855A5 true JP2023533855A5 (https=) 2025-09-12

Family

ID=79293345

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023502881A Pending JP2023533855A (ja) 2020-07-16 2021-05-27 イソキノリン化合物およびそのAhR不均衡の治療への使用

Country Status (10)

Country Link
US (5) US11267788B2 (https=)
EP (1) EP4185566A4 (https=)
JP (1) JP2023533855A (https=)
KR (1) KR20230041021A (https=)
CN (1) CN116157387A (https=)
AU (1) AU2021308209A1 (https=)
CA (1) CA3185793A1 (https=)
IL (1) IL299756A (https=)
MX (1) MX2023000263A (https=)
WO (1) WO2022015423A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2023533855A (ja) 2020-07-16 2023-08-04 ダーマヴァント サイエンシーズ ゲーエムベーハー イソキノリン化合物およびそのAhR不均衡の治療への使用
WO2024020170A1 (en) * 2022-07-21 2024-01-25 Allianthera (Suzhou) Biopharmaceutical Co., Ltd. Aryl hydrocarbon receptor agonist prodrugs and methods of use thereof
US20260069585A1 (en) * 2022-08-30 2026-03-12 Dermavant Sciences GmbH ISOQUINOLINE COMPOUNDS AND THEIR USE IN TREATING AhR MEDIATED DISEASES
WO2024152993A1 (zh) * 2023-01-17 2024-07-25 上海泽德曼医药科技有限公司 稠环类化合物、其制备方法及其在医药上的应用
CN117447402A (zh) * 2023-10-18 2024-01-26 德明药泰生物技术(深圳)有限公司 芳香烃受体调节剂类化合物及其制备方法和应用
CN117229208B (zh) * 2023-11-13 2024-02-23 上海泽德曼医药科技有限公司 稠环类化合物、其制备方法及其在医药上的应用
WO2026083733A1 (ja) * 2024-10-18 2026-04-23 株式会社ヤクルト本社 試験方法、ゲル状組成物、及び試験装置

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WO1992018123A2 (en) 1991-04-10 1992-10-29 Octamer, Inc. A method for inhibition of retroviral replication
US5919970A (en) 1997-04-24 1999-07-06 Allergan Sales, Inc. Substituted diaryl or diheteroaryl methanes, ethers and amines having retinoid agonist, antagonist or inverse agonist type biological activity
ATE404539T1 (de) * 1997-10-02 2008-08-15 Eisai R&D Man Co Ltd Kondensierte pyridinderivate
HRP20040102A2 (en) 2001-07-09 2004-10-31 Combinatorx Combinations for the treatment of inflammatory disorders
WO2003053359A2 (en) * 2001-12-19 2003-07-03 Atherogenics, Inc. 1,3-bis-(substituted-phenyl)-2-propyn-1-ones and their use to treat disorders
IL162533A0 (en) * 2001-12-19 2005-11-20 Atherogenics Inc Chalcone derivatives and their use to treat diseases
JPWO2005063222A1 (ja) 2003-12-26 2007-07-19 協和醗酵工業株式会社 Hsp90ファミリー蛋白質阻害剤
WO2006058201A2 (en) 2004-11-23 2006-06-01 Reddy Us Therapeutics, Inc. Heterocyclic and bicyclic compounds, compositions and methods
GB0704718D0 (en) 2007-03-12 2007-04-18 Prendergast Patrick T Compounds and methods for preventing and treating mucositis
EP2014651A1 (en) 2007-07-12 2009-01-14 Exonhit Therapeutics SA Compounds and methods for modulating Rho GTPases
JP5439127B2 (ja) 2009-11-13 2014-03-12 株式会社さいわいメディカル 乾癬又はアトピー性皮膚炎治療剤
WO2011156626A1 (en) 2010-06-09 2011-12-15 Rutgers, The State University Of New Jersey Antimicrobial agents
GB201216017D0 (en) * 2012-09-07 2012-10-24 Cancer Rec Tech Ltd Inhibitor compounds
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JP7138654B2 (ja) * 2017-03-29 2022-09-16 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツング 金属錯体
US11548867B2 (en) * 2017-07-19 2023-01-10 Idea Ya Biosciences, Inc. Amido compounds as AhR modulators
EP3752512B1 (de) * 2018-02-13 2023-03-01 Merck Patent GmbH Metallkomplexe
TWI828664B (zh) 2018-03-19 2024-01-11 愛爾蘭商Udc愛爾蘭責任有限公司 金屬錯合物
JP2023533855A (ja) 2020-07-16 2023-08-04 ダーマヴァント サイエンシーズ ゲーエムベーハー イソキノリン化合物およびそのAhR不均衡の治療への使用
WO2023020512A1 (zh) * 2021-08-16 2023-02-23 成都奥睿药业有限公司 取代的吡啶类似物、其制备方法及作为ahr调节剂的用途
CN116947799B (zh) * 2023-03-08 2024-05-03 上海泽德曼医药科技有限公司 酚类化合物、其制备方法及其在医药上的应用

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