JP2025505521A5 - - Google Patents

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Publication number
JP2025505521A5
JP2025505521A5 JP2024543160A JP2024543160A JP2025505521A5 JP 2025505521 A5 JP2025505521 A5 JP 2025505521A5 JP 2024543160 A JP2024543160 A JP 2024543160A JP 2024543160 A JP2024543160 A JP 2024543160A JP 2025505521 A5 JP2025505521 A5 JP 2025505521A5
Authority
JP
Japan
Prior art keywords
formula
compound
fmoc
boc
adoc
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024543160A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025505521A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2023/053409 external-priority patent/WO2023152347A1/en
Publication of JP2025505521A publication Critical patent/JP2025505521A/ja
Publication of JP2025505521A5 publication Critical patent/JP2025505521A5/ja
Pending legal-status Critical Current

Links

JP2024543160A 2022-02-14 2023-02-13 大環状ペプチドを製造するための方法 Pending JP2025505521A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP22156480.0 2022-02-14
EP22156480 2022-02-14
PCT/EP2023/053409 WO2023152347A1 (en) 2022-02-14 2023-02-13 Process for manufacturing macrocyclic peptides

Publications (2)

Publication Number Publication Date
JP2025505521A JP2025505521A (ja) 2025-02-28
JP2025505521A5 true JP2025505521A5 (https=) 2026-02-09

Family

ID=80683163

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024543160A Pending JP2025505521A (ja) 2022-02-14 2023-02-13 大環状ペプチドを製造するための方法

Country Status (12)

Country Link
US (1) US20250109166A1 (https=)
EP (1) EP4479396A1 (https=)
JP (1) JP2025505521A (https=)
KR (1) KR20240144894A (https=)
CN (1) CN118660878A (https=)
AR (1) AR128501A1 (https=)
AU (1) AU2023217269A1 (https=)
CA (1) CA3237617A1 (https=)
IL (1) IL313664A (https=)
MX (1) MX2024009210A (https=)
TW (1) TW202342493A (https=)
WO (1) WO2023152347A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2026068674A1 (en) 2024-09-27 2026-04-02 F. Hoffmann-La Roche Ag Process for deprotection of aminoacid derivatives

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6136934B2 (ja) 2011-12-15 2017-05-31 味の素株式会社 Fmoc基の除去方法
US11819532B2 (en) 2018-04-23 2023-11-21 Hoffmann-La Roche Inc. Peptide macrocycles against Acinetobacter baumannii

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