JP2025165966A5 - - Google Patents

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Publication number
JP2025165966A5
JP2025165966A5 JP2025119759A JP2025119759A JP2025165966A5 JP 2025165966 A5 JP2025165966 A5 JP 2025165966A5 JP 2025119759 A JP2025119759 A JP 2025119759A JP 2025119759 A JP2025119759 A JP 2025119759A JP 2025165966 A5 JP2025165966 A5 JP 2025165966A5
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JP
Japan
Prior art keywords
alkyl
methyl
independently selected
carboxy
aryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2025119759A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025165966A (ja
Filing date
Publication date
Priority claimed from EP19180240.4A external-priority patent/EP3750878B1/en
Application filed filed Critical
Publication of JP2025165966A publication Critical patent/JP2025165966A/ja
Publication of JP2025165966A5 publication Critical patent/JP2025165966A5/ja
Pending legal-status Critical Current

Links

JP2025119759A 2019-06-14 2025-07-16 アスタシンプロテイナーゼのヘテロ芳香族インヒビター Pending JP2025165966A (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP19180240.4 2019-06-14
EP19180240.4A EP3750878B1 (en) 2019-06-14 2019-06-14 Heteroaromatic inhibitors of astacin proteinases
JP2021574193A JP7773377B2 (ja) 2019-06-14 2020-06-12 アスタシンプロテイナーゼのヘテロ芳香族インヒビター
PCT/EP2020/066352 WO2020249760A1 (en) 2019-06-14 2020-06-12 Heteroaromatic inhibitors of astacin proteinases

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2021574193A Division JP7773377B2 (ja) 2019-06-14 2020-06-12 アスタシンプロテイナーゼのヘテロ芳香族インヒビター

Publications (2)

Publication Number Publication Date
JP2025165966A JP2025165966A (ja) 2025-11-05
JP2025165966A5 true JP2025165966A5 (https=) 2026-02-02

Family

ID=67105691

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021574193A Active JP7773377B2 (ja) 2019-06-14 2020-06-12 アスタシンプロテイナーゼのヘテロ芳香族インヒビター
JP2025119759A Pending JP2025165966A (ja) 2019-06-14 2025-07-16 アスタシンプロテイナーゼのヘテロ芳香族インヒビター

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2021574193A Active JP7773377B2 (ja) 2019-06-14 2020-06-12 アスタシンプロテイナーゼのヘテロ芳香族インヒビター

Country Status (13)

Country Link
US (2) US20230122243A1 (https=)
EP (2) EP3750878B1 (https=)
JP (2) JP7773377B2 (https=)
KR (2) KR20260036022A (https=)
CN (1) CN114585608B (https=)
AU (1) AU2020291114B2 (https=)
BR (1) BR112021024327A2 (https=)
CA (2) CA3142992A1 (https=)
IL (2) IL288851B2 (https=)
MX (2) MX2021015324A (https=)
SG (1) SG11202112905UA (https=)
WO (1) WO2020249760A1 (https=)
ZA (1) ZA202109419B (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112021024726A2 (pt) 2019-06-07 2022-01-18 Elanco Tiergesundheit Ag Novos derivados bicíclicos
EP4244281B1 (en) 2021-02-26 2024-04-03 Sun Chemical B.V. Photoinitiator resins with dibenzoylmethane substructure
CN113698349B (zh) * 2021-09-02 2023-08-01 河南师范大学 一种2-(2-苯基-2h-吲唑-3-基)乙酸酯类化合物的水相光催化制备方法
CN114262296B (zh) * 2021-12-21 2023-07-18 南京工业大学 一种利用微通道反应装置合成咪唑类化合物的方法
WO2023118482A1 (en) 2021-12-24 2023-06-29 Sun Chemical Corporation Amine synergists with uv-a absorption
CN119101046A (zh) * 2024-08-30 2024-12-10 沈阳药科大学 3-萘基噻吩类衍生物及其制备方法和应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1036004B (it) * 1968-05-21 1979-10-30 Abc Ist Biolog Chem Spa Acidt 3 indolil adetoidrossamici
US4146721A (en) * 1969-09-12 1979-03-27 Byk Gulden Lomberg Chemische Fabrik Gmbh Pyrazol-4-acetic acid compounds
US4021448A (en) * 1975-10-21 1977-05-03 Sterling Drug Inc. 2-Substituted-indole-1-lower-alkanecarboxamides
KR100432928B1 (ko) * 2001-04-26 2004-05-28 주식회사 코오롱 신규한 하이드록스아믹산 유도체, 신규한 그의 중간체화합물 및 그들의 제조방법
US20090005344A1 (en) 2004-11-01 2009-01-01 Nkuada, Llc Compounds and Methods of Use Thereof
DE102005019181A1 (de) * 2005-04-25 2006-10-26 Novartis Ag Peptid-Deformylase (PDF) Inhibitoren 1
AU2008252628A1 (en) 2007-05-18 2008-11-27 Inhibox Ltd. Bicyclosulfonyl acid (BCSA) compounds and their use as therapeutic agents
KR102410199B1 (ko) 2016-04-18 2022-06-17 프라운호퍼-게젤샤프트 츄어 푀르더룽 데어 안게반텐 포르슝에.파우. 새로운 메프린 알파 및 베타 저해제

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