JP2022536183A5 - - Google Patents

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Publication number
JP2022536183A5
JP2022536183A5 JP2021574193A JP2021574193A JP2022536183A5 JP 2022536183 A5 JP2022536183 A5 JP 2022536183A5 JP 2021574193 A JP2021574193 A JP 2021574193A JP 2021574193 A JP2021574193 A JP 2021574193A JP 2022536183 A5 JP2022536183 A5 JP 2022536183A5
Authority
JP
Japan
Application number
JP2021574193A
Other languages
Japanese (ja)
Other versions
JPWO2020249760A5 (https=
JP7773377B2 (ja
JP2022536183A (ja
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Publication date
Priority claimed from EP19180240.4A external-priority patent/EP3750878B1/en
Application filed filed Critical
Publication of JP2022536183A publication Critical patent/JP2022536183A/ja
Publication of JPWO2020249760A5 publication Critical patent/JPWO2020249760A5/ja
Publication of JP2022536183A5 publication Critical patent/JP2022536183A5/ja
Priority to JP2025119759A priority Critical patent/JP2025165966A/ja
Application granted granted Critical
Publication of JP7773377B2 publication Critical patent/JP7773377B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2021574193A 2019-06-14 2020-06-12 アスタシンプロテイナーゼのヘテロ芳香族インヒビター Active JP7773377B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025119759A JP2025165966A (ja) 2019-06-14 2025-07-16 アスタシンプロテイナーゼのヘテロ芳香族インヒビター

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP19180240.4 2019-06-14
EP19180240.4A EP3750878B1 (en) 2019-06-14 2019-06-14 Heteroaromatic inhibitors of astacin proteinases
PCT/EP2020/066352 WO2020249760A1 (en) 2019-06-14 2020-06-12 Heteroaromatic inhibitors of astacin proteinases

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025119759A Division JP2025165966A (ja) 2019-06-14 2025-07-16 アスタシンプロテイナーゼのヘテロ芳香族インヒビター

Publications (4)

Publication Number Publication Date
JP2022536183A JP2022536183A (ja) 2022-08-12
JPWO2020249760A5 JPWO2020249760A5 (https=) 2023-05-25
JP2022536183A5 true JP2022536183A5 (https=) 2023-05-25
JP7773377B2 JP7773377B2 (ja) 2025-11-19

Family

ID=67105691

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021574193A Active JP7773377B2 (ja) 2019-06-14 2020-06-12 アスタシンプロテイナーゼのヘテロ芳香族インヒビター
JP2025119759A Pending JP2025165966A (ja) 2019-06-14 2025-07-16 アスタシンプロテイナーゼのヘテロ芳香族インヒビター

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025119759A Pending JP2025165966A (ja) 2019-06-14 2025-07-16 アスタシンプロテイナーゼのヘテロ芳香族インヒビター

Country Status (13)

Country Link
US (2) US20230122243A1 (https=)
EP (2) EP3750878B1 (https=)
JP (2) JP7773377B2 (https=)
KR (2) KR20260036022A (https=)
CN (1) CN114585608B (https=)
AU (1) AU2020291114B2 (https=)
BR (1) BR112021024327A2 (https=)
CA (2) CA3142992A1 (https=)
IL (2) IL288851B2 (https=)
MX (2) MX2021015324A (https=)
SG (1) SG11202112905UA (https=)
WO (1) WO2020249760A1 (https=)
ZA (1) ZA202109419B (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112021024726A2 (pt) 2019-06-07 2022-01-18 Elanco Tiergesundheit Ag Novos derivados bicíclicos
EP4244281B1 (en) 2021-02-26 2024-04-03 Sun Chemical B.V. Photoinitiator resins with dibenzoylmethane substructure
CN113698349B (zh) * 2021-09-02 2023-08-01 河南师范大学 一种2-(2-苯基-2h-吲唑-3-基)乙酸酯类化合物的水相光催化制备方法
CN114262296B (zh) * 2021-12-21 2023-07-18 南京工业大学 一种利用微通道反应装置合成咪唑类化合物的方法
WO2023118482A1 (en) 2021-12-24 2023-06-29 Sun Chemical Corporation Amine synergists with uv-a absorption
CN119101046A (zh) * 2024-08-30 2024-12-10 沈阳药科大学 3-萘基噻吩类衍生物及其制备方法和应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1036004B (it) * 1968-05-21 1979-10-30 Abc Ist Biolog Chem Spa Acidt 3 indolil adetoidrossamici
US4146721A (en) * 1969-09-12 1979-03-27 Byk Gulden Lomberg Chemische Fabrik Gmbh Pyrazol-4-acetic acid compounds
US4021448A (en) * 1975-10-21 1977-05-03 Sterling Drug Inc. 2-Substituted-indole-1-lower-alkanecarboxamides
KR100432928B1 (ko) * 2001-04-26 2004-05-28 주식회사 코오롱 신규한 하이드록스아믹산 유도체, 신규한 그의 중간체화합물 및 그들의 제조방법
US20090005344A1 (en) 2004-11-01 2009-01-01 Nkuada, Llc Compounds and Methods of Use Thereof
DE102005019181A1 (de) * 2005-04-25 2006-10-26 Novartis Ag Peptid-Deformylase (PDF) Inhibitoren 1
AU2008252628A1 (en) 2007-05-18 2008-11-27 Inhibox Ltd. Bicyclosulfonyl acid (BCSA) compounds and their use as therapeutic agents
KR102410199B1 (ko) 2016-04-18 2022-06-17 프라운호퍼-게젤샤프트 츄어 푀르더룽 데어 안게반텐 포르슝에.파우. 새로운 메프린 알파 및 베타 저해제

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