JP2022536183A5 - - Google Patents
Info
- Publication number
- JP2022536183A5 JP2022536183A5 JP2021574193A JP2021574193A JP2022536183A5 JP 2022536183 A5 JP2022536183 A5 JP 2022536183A5 JP 2021574193 A JP2021574193 A JP 2021574193A JP 2021574193 A JP2021574193 A JP 2021574193A JP 2022536183 A5 JP2022536183 A5 JP 2022536183A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- group
- independently selected
- aryl
- carboxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2025119759A JP2025165966A (ja) | 2019-06-14 | 2025-07-16 | アスタシンプロテイナーゼのヘテロ芳香族インヒビター |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP19180240.4 | 2019-06-14 | ||
| EP19180240.4A EP3750878B1 (en) | 2019-06-14 | 2019-06-14 | Heteroaromatic inhibitors of astacin proteinases |
| PCT/EP2020/066352 WO2020249760A1 (en) | 2019-06-14 | 2020-06-12 | Heteroaromatic inhibitors of astacin proteinases |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025119759A Division JP2025165966A (ja) | 2019-06-14 | 2025-07-16 | アスタシンプロテイナーゼのヘテロ芳香族インヒビター |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022536183A JP2022536183A (ja) | 2022-08-12 |
| JP2022536183A5 true JP2022536183A5 (https=) | 2023-05-25 |
| JP7773377B2 JP7773377B2 (ja) | 2025-11-19 |
Family
ID=67105691
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021574193A Active JP7773377B2 (ja) | 2019-06-14 | 2020-06-12 | アスタシンプロテイナーゼのヘテロ芳香族インヒビター |
| JP2025119759A Pending JP2025165966A (ja) | 2019-06-14 | 2025-07-16 | アスタシンプロテイナーゼのヘテロ芳香族インヒビター |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025119759A Pending JP2025165966A (ja) | 2019-06-14 | 2025-07-16 | アスタシンプロテイナーゼのヘテロ芳香族インヒビター |
Country Status (13)
| Country | Link |
|---|---|
| US (2) | US20230122243A1 (https=) |
| EP (2) | EP3750878B1 (https=) |
| JP (2) | JP7773377B2 (https=) |
| KR (2) | KR20260036022A (https=) |
| CN (1) | CN114585608B (https=) |
| AU (1) | AU2020291114B2 (https=) |
| BR (1) | BR112021024327A2 (https=) |
| CA (2) | CA3300715A1 (https=) |
| IL (2) | IL288851B2 (https=) |
| MX (2) | MX2021015324A (https=) |
| SG (1) | SG11202112905UA (https=) |
| WO (1) | WO2020249760A1 (https=) |
| ZA (1) | ZA202109419B (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US12448391B2 (en) | 2019-06-07 | 2025-10-21 | Elanco Tiergesundheit Ag | Bicyclic derivatives for treating endoparasites |
| WO2022180269A1 (en) | 2021-02-26 | 2022-09-01 | Sun Chemical Corporation | Photoinitiator resins with dibenzoylmethane substructure |
| CN113698349B (zh) * | 2021-09-02 | 2023-08-01 | 河南师范大学 | 一种2-(2-苯基-2h-吲唑-3-基)乙酸酯类化合物的水相光催化制备方法 |
| CN114262296B (zh) * | 2021-12-21 | 2023-07-18 | 南京工业大学 | 一种利用微通道反应装置合成咪唑类化合物的方法 |
| US12264120B2 (en) | 2021-12-24 | 2025-04-01 | Sun Chemical Corporation | Amine synergists with UV—a absorption |
| CN119101046A (zh) * | 2024-08-30 | 2024-12-10 | 沈阳药科大学 | 3-萘基噻吩类衍生物及其制备方法和应用 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1036004B (it) * | 1968-05-21 | 1979-10-30 | Abc Ist Biolog Chem Spa | Acidt 3 indolil adetoidrossamici |
| US4146721A (en) * | 1969-09-12 | 1979-03-27 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Pyrazol-4-acetic acid compounds |
| US4021448A (en) * | 1975-10-21 | 1977-05-03 | Sterling Drug Inc. | 2-Substituted-indole-1-lower-alkanecarboxamides |
| KR100432928B1 (ko) * | 2001-04-26 | 2004-05-28 | 주식회사 코오롱 | 신규한 하이드록스아믹산 유도체, 신규한 그의 중간체화합물 및 그들의 제조방법 |
| EP1812451A4 (en) * | 2004-11-01 | 2009-10-21 | Nuada Llc | COMPOUNDS AND METHODS OF USE THEREOF |
| DE102005019181A1 (de) * | 2005-04-25 | 2006-10-26 | Novartis Ag | Peptid-Deformylase (PDF) Inhibitoren 1 |
| BRPI0811651A2 (pt) | 2007-05-18 | 2014-11-11 | Inhibox Ltd | Composto, composição farmacêutica, métodos para preparar uma composição farmacêutica, para tratar uma doença, distúrbio ou condição, para inibir a tace em uma célula, in vitro ou in vivo, e de regular (por exemplo, inibir) a liberação da citocina (por exemplo, a liberação da tnf-alfa) em uma célula, in vitro ou in vivo, uso de um composto, e, kit |
| PL3445744T3 (pl) | 2016-04-18 | 2022-02-07 | Vivoryon Therapeutics Ag | Nowe inhibitory mepryny alfa i beta |
-
2019
- 2019-06-14 EP EP19180240.4A patent/EP3750878B1/en active Active
-
2020
- 2020-06-12 IL IL288851A patent/IL288851B2/en unknown
- 2020-06-12 US US17/618,964 patent/US20230122243A1/en not_active Abandoned
- 2020-06-12 BR BR112021024327A patent/BR112021024327A2/pt unknown
- 2020-06-12 CA CA3300715A patent/CA3300715A1/en active Pending
- 2020-06-12 CN CN202080057197.6A patent/CN114585608B/zh active Active
- 2020-06-12 EP EP20733712.2A patent/EP3986868A1/en active Pending
- 2020-06-12 SG SG11202112905UA patent/SG11202112905UA/en unknown
- 2020-06-12 JP JP2021574193A patent/JP7773377B2/ja active Active
- 2020-06-12 KR KR1020267005267A patent/KR20260036022A/ko active Pending
- 2020-06-12 CA CA3142992A patent/CA3142992A1/en active Pending
- 2020-06-12 KR KR1020217043341A patent/KR102930913B1/ko active Active
- 2020-06-12 AU AU2020291114A patent/AU2020291114B2/en active Active
- 2020-06-12 WO PCT/EP2020/066352 patent/WO2020249760A1/en not_active Ceased
- 2020-06-12 MX MX2021015324A patent/MX2021015324A/es unknown
-
2021
- 2021-11-23 ZA ZA2021/09419A patent/ZA202109419B/en unknown
- 2021-12-10 MX MX2025005324A patent/MX2025005324A/es unknown
-
2025
- 2025-07-16 JP JP2025119759A patent/JP2025165966A/ja active Pending
- 2025-09-02 US US19/316,605 patent/US20250388544A1/en active Pending
- 2025-09-14 IL IL323353A patent/IL323353A/en unknown
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