JP2024537564A5 - - Google Patents

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Publication number
JP2024537564A5
JP2024537564A5 JP2024513882A JP2024513882A JP2024537564A5 JP 2024537564 A5 JP2024537564 A5 JP 2024537564A5 JP 2024513882 A JP2024513882 A JP 2024513882A JP 2024513882 A JP2024513882 A JP 2024513882A JP 2024537564 A5 JP2024537564 A5 JP 2024537564A5
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Japan
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compound
formula
crystal form
crystalline form
free acid
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JP2024513882A
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English (en)
Japanese (ja)
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JP2024537564A (ja
JP7819298B2 (ja
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Priority claimed from PCT/CN2022/116768 external-priority patent/WO2023030492A1/zh
Publication of JP2024537564A publication Critical patent/JP2024537564A/ja
Publication of JP2024537564A5 publication Critical patent/JP2024537564A5/ja
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JP2024513882A 2021-09-03 2022-09-02 Ep4拮抗剤化合物及びその塩、結晶多形並びに使用 Active JP7819298B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN202111034159.1 2021-09-03
CN202111034159 2021-09-03
PCT/CN2022/116768 WO2023030492A1 (zh) 2021-09-03 2022-09-02 一种ep4拮抗剂化合物及其盐、多晶型和用途

Publications (3)

Publication Number Publication Date
JP2024537564A JP2024537564A (ja) 2024-10-11
JP2024537564A5 true JP2024537564A5 (https=) 2024-11-14
JP7819298B2 JP7819298B2 (ja) 2026-02-24

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ID=85349540

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Application Number Title Priority Date Filing Date
JP2024513882A Active JP7819298B2 (ja) 2021-09-03 2022-09-02 Ep4拮抗剤化合物及びその塩、結晶多形並びに使用

Country Status (7)

Country Link
US (1) US20240368088A1 (https=)
EP (1) EP4397654A4 (https=)
JP (1) JP7819298B2 (https=)
CN (1) CN115745892A (https=)
CA (1) CA3230557A1 (https=)
TW (1) TW202328073A (https=)
WO (1) WO2023030492A1 (https=)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2011260332B2 (en) 2010-06-03 2014-10-02 Bayer Cropscience Ag N-[(het)arylethyl)] pyrazole(thio)carboxamides and their heterosubstituted analogues
PE20131343A1 (es) * 2010-09-21 2013-11-18 Eisai Randd Man Co Ltd Derivados de acido benzoico
AU2015264102C1 (en) * 2014-05-23 2020-10-08 Eisai R&D Management Co., Ltd. Combination therapies for the treatment of cancer
KR102796877B1 (ko) * 2020-03-04 2025-04-15 우한 휴먼웰 이노베이티브 드러그 리서치 앤드 디벨롭먼트 센터 리미티드 컴퍼니 신규 ep4 길항제의 합성 및 암과 염증에서의 이의 용도
TWI877433B (zh) * 2020-11-30 2025-03-21 大陸商杭州阿諾生物醫藥科技有限公司 用於治療pik3ca突變癌症的組合療法
CN114790176A (zh) * 2021-01-25 2022-07-26 武汉人福创新药物研发中心有限公司 咪唑类化合物及其制备方法和用途
WO2022161418A1 (zh) * 2021-01-28 2022-08-04 深圳晶泰科技有限公司 吡唑酰胺衍生物及其制备方法和应用

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