JP2024511611A5 - - Google Patents

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Publication number
JP2024511611A5
JP2024511611A5 JP2023558350A JP2023558350A JP2024511611A5 JP 2024511611 A5 JP2024511611 A5 JP 2024511611A5 JP 2023558350 A JP2023558350 A JP 2023558350A JP 2023558350 A JP2023558350 A JP 2023558350A JP 2024511611 A5 JP2024511611 A5 JP 2024511611A5
Authority
JP
Japan
Prior art keywords
methyl
carbonyl
decane
azaspiro
piperidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023558350A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024511611A (ja
Filing date
Publication date
Priority claimed from GBGB2104097.7A external-priority patent/GB202104097D0/en
Application filed filed Critical
Publication of JP2024511611A publication Critical patent/JP2024511611A/ja
Publication of JP2024511611A5 publication Critical patent/JP2024511611A5/ja
Pending legal-status Critical Current

Links

JP2023558350A 2021-03-24 2022-03-24 ユビキチン特異的プロテアーゼ19阻害剤としての医薬化合物 Pending JP2024511611A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB2104097.7A GB202104097D0 (en) 2021-03-24 2021-03-24 Pharmaceutical compounds
GB2104097.7 2021-03-24
PCT/EP2022/057820 WO2022200523A1 (en) 2021-03-24 2022-03-24 Pharmaceuticals compounds as inhibitors of ubiquitin specific protease 19 (usp19)

Publications (2)

Publication Number Publication Date
JP2024511611A JP2024511611A (ja) 2024-03-14
JP2024511611A5 true JP2024511611A5 (https=) 2025-03-26

Family

ID=75689814

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023558350A Pending JP2024511611A (ja) 2021-03-24 2022-03-24 ユビキチン特異的プロテアーゼ19阻害剤としての医薬化合物

Country Status (12)

Country Link
US (1) US20240327382A1 (https=)
EP (1) EP4313295A1 (https=)
JP (1) JP2024511611A (https=)
KR (1) KR20230160901A (https=)
CN (1) CN117157285A (https=)
AU (1) AU2022244178A1 (https=)
BR (1) BR112023019323A2 (https=)
CA (1) CA3212236A1 (https=)
GB (1) GB202104097D0 (https=)
IL (1) IL307163A (https=)
MX (1) MX2023011012A (https=)
WO (1) WO2022200523A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN115656383A (zh) * 2022-11-11 2023-01-31 武汉海特生物创新医药研究有限公司 一种alpha-苯基哌啶-2-乙酰胺对映异构体的检测方法
GB202311227D0 (en) 2023-07-21 2023-09-06 Almac Discovery Ltd Pharmaceutical compounds

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2335701B1 (en) * 2003-12-15 2012-07-11 Schering Corporation Heterocyclic aspartyl protease inhibitors
US9938300B2 (en) * 2015-02-05 2018-04-10 Forma Therapeutics, Inc. Isothiazolopyrimidinones, pyrazolopyrimidinones, and pyrrolopyrimidinones as ubiquitin-specific protease 7 inhibitors
US9840491B2 (en) * 2015-02-05 2017-12-12 Forma Therapeutics, Inc. Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors
EP3253765A1 (en) * 2015-02-05 2017-12-13 Forma Therapeutics, Inc. Thienopyrimidinones as ubiquitin-specific protease 7 inhibitors
GB201612938D0 (en) 2016-07-26 2016-09-07 Almac Discovery Ltd Pharmaceutical compounds
JP7402792B2 (ja) * 2017-09-26 2023-12-21 デイナ ファーバー キャンサー インスティチュート,インコーポレイテッド 多発性骨髄腫を治療するための新規なusp7阻害剤
GB201801562D0 (en) * 2018-01-31 2018-03-14 Almac Diagnostics Ltd Pharmaceutical compounds
MX2021006542A (es) * 2018-12-06 2021-07-07 Almac Discovery Ltd Inhibidores de la usp19 para usarse en terapia.
CN113365696A (zh) * 2018-12-06 2021-09-07 阿尔麦克探索有限公司 药物化合物和其作为泛素特异性蛋白酶19(usp19)抑制剂的用途
EP3965749A4 (en) * 2019-05-06 2023-06-21 Valo Health, Inc. ESCAPEMENT OF USP19

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