JP2024509421A5 - - Google Patents
Info
- Publication number
- JP2024509421A5 JP2024509421A5 JP2023552539A JP2023552539A JP2024509421A5 JP 2024509421 A5 JP2024509421 A5 JP 2024509421A5 JP 2023552539 A JP2023552539 A JP 2023552539A JP 2023552539 A JP2023552539 A JP 2023552539A JP 2024509421 A5 JP2024509421 A5 JP 2024509421A5
- Authority
- JP
- Japan
- Prior art keywords
- triazole
- hydroxymethyl
- pyran
- methyl
- methoxytetrahydro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EPPCT/EP2021/055348 | 2021-03-03 | ||
| EP2021055348 | 2021-03-03 | ||
| PCT/EP2022/055224 WO2022184755A1 (en) | 2021-03-03 | 2022-03-02 | Triazolyl-methyl substituted alpha-d-galactopyranoside derivatives |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2024509421A JP2024509421A (ja) | 2024-03-01 |
| JP2024509421A5 true JP2024509421A5 (https=) | 2025-03-10 |
| JP7771205B2 JP7771205B2 (ja) | 2025-11-17 |
Family
ID=80682779
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023552539A Active JP7771205B2 (ja) | 2021-03-03 | 2022-03-02 | トリアゾリル-メチル置換アルファ-d-ガラクトピラノシド誘導体 |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US20240109930A1 (https=) |
| EP (1) | EP4301748B1 (https=) |
| JP (1) | JP7771205B2 (https=) |
| KR (1) | KR20230154221A (https=) |
| CN (1) | CN116888113A (https=) |
| AU (1) | AU2022228660A1 (https=) |
| BR (1) | BR112023017624A2 (https=) |
| CA (1) | CA3209917A1 (https=) |
| CL (1) | CL2023002578A1 (https=) |
| ES (1) | ES3033422T3 (https=) |
| HR (1) | HRP20250833T1 (https=) |
| HU (1) | HUE072194T2 (https=) |
| IL (1) | IL305581A (https=) |
| MA (1) | MA63589B1 (https=) |
| MX (1) | MX2023010241A (https=) |
| PL (1) | PL4301748T3 (https=) |
| RS (1) | RS67032B1 (https=) |
| TW (1) | TWI905393B (https=) |
| UA (1) | UA130562C2 (https=) |
| WO (1) | WO2022184755A1 (https=) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN114206893A (zh) | 2019-08-09 | 2022-03-18 | 爱杜西亚药品有限公司 | (杂)芳基-甲基-硫代-β-D-吡喃半乳糖苷衍生物 |
| WO2021028323A1 (en) | 2019-08-09 | 2021-02-18 | Idorsia Pharmaceuticals Ltd | (2-acetamidyl)thio-beta-d-galactopyranoside derivatives |
| MA56883B1 (fr) | 2019-08-15 | 2025-04-30 | Idorsia Pharmaceuticals Ltd | Dérivés de 2-hydroxycycloalcane-1-carbamoyle |
| CN114585619B (zh) | 2019-08-29 | 2024-09-27 | 爱杜西亚药品有限公司 | α-D-吡喃半乳糖苷衍生物 |
| US12312362B2 (en) | 2020-10-06 | 2025-05-27 | Idorsia Pharmaceuticals Ltd | Spiro derivatives of Alpha-D-galactopyranosides |
| EP4237419A1 (en) | 2020-11-02 | 2023-09-06 | Idorsia Pharmaceuticals Ltd | Galectin-3 inhibiting 2-hydroxycycloalkane-1 -carbamoyl derivatives |
| CN116806219A (zh) | 2021-02-09 | 2023-09-26 | 爱杜西亚药品有限公司 | 羟基杂环烷-氨甲酰基衍生物 |
Family Cites Families (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE0100172D0 (sv) | 2001-01-22 | 2001-01-22 | Ulf Nilsson | New inhibitors against galectins |
| SE0401300D0 (sv) | 2004-05-21 | 2004-05-21 | Forskarpatent I Syd Ab | Novel Galactoside Inhibitors of Galectins |
| SE0401301D0 (sv) | 2004-05-21 | 2004-05-21 | Forskarpatent I Syd Ab | Novel 3-triazolyl-galactoside inhibitors of galectins |
| DK2906227T3 (en) | 2012-10-10 | 2018-12-10 | Galectin Therapeutics Inc | GALACTOSE-CONTAINING CARBOHYDRATE COMPOUNDS FOR THE TREATMENT OF DIABETIC Nephropathy |
| CN104755088A (zh) | 2012-10-31 | 2015-07-01 | 格莱克特生物技术公司 | 半乳凝集素-3的半乳糖苷抑制剂及其用于治疗肺纤维化的应用 |
| EP2919802A4 (en) | 2012-11-15 | 2016-09-14 | Univ Tufts | METHOD, COMPOSITIONS AND KITS FOR TREATING, MODULATING OR PREVENTING ANGIOGENESIS OR FIBROSIS IN A PATIENT USING A GALECTINE PROTEIN HEMMER |
| CA2970062C (en) | 2015-01-30 | 2023-02-28 | Galecto Biotech Ab | Alpha-d-galactoside inhibitors of galectins |
| PL3456717T3 (pl) | 2015-07-06 | 2021-10-25 | Gilead Sciences, Inc. | Pochodna 4,6-diaminochinolino-3-karbonitrylu jako modulator cot (cancer osaka thyroid) do leczenia choroby zapalnej |
| EP3621973A4 (en) | 2017-05-12 | 2021-10-27 | Galectin Sciences, LLC | COMPOUNDS FOR THE PREVENTION AND TREATMENT OF DISEASES AND USES THEREOF |
| KR20200015528A (ko) | 2017-05-12 | 2020-02-12 | 갈랙틴 사이언시즈, 엘엘씨 | 전신 인슐린 내성 질환의 치료용 화합물 및 그의 용도 |
| WO2019067702A1 (en) * | 2017-09-27 | 2019-04-04 | Bristol-Myers Squibb Company | INHIBITORS WITH SMALL MOLECULES OF GALECTIN-3 |
| US11072626B2 (en) | 2017-10-11 | 2021-07-27 | Bristol-Myers Squibb Company | Small molecule inhibitors of Galectin-3 |
| CA3080128A1 (en) | 2017-10-31 | 2019-05-09 | Galectin Sciences, Llc | Selenogalactoside compounds for the treatment of systemic insulin resistance disorders and the use thereof |
| WO2020104335A1 (en) | 2018-11-21 | 2020-05-28 | Galecto Biotech Ab | Alpha-d-galactoside inhibitors of galectins |
| US12269819B2 (en) * | 2019-04-10 | 2025-04-08 | Bristol-Myers Squibb Company | Small molecule inhibitors of Galectin-3 |
| JP7674276B2 (ja) | 2019-07-03 | 2025-05-09 | ガレクト バイオテック エービー | ガレクチンの新規なガラクトシド阻害剤 |
| WO2021004940A1 (en) | 2019-07-05 | 2021-01-14 | Galecto Biotech Ab | Novel galactoside inhibitor of galectins |
| WO2021028323A1 (en) | 2019-08-09 | 2021-02-18 | Idorsia Pharmaceuticals Ltd | (2-acetamidyl)thio-beta-d-galactopyranoside derivatives |
| CN114206893A (zh) | 2019-08-09 | 2022-03-18 | 爱杜西亚药品有限公司 | (杂)芳基-甲基-硫代-β-D-吡喃半乳糖苷衍生物 |
| MA56883B1 (fr) | 2019-08-15 | 2025-04-30 | Idorsia Pharmaceuticals Ltd | Dérivés de 2-hydroxycycloalcane-1-carbamoyle |
| CN114585619B (zh) | 2019-08-29 | 2024-09-27 | 爱杜西亚药品有限公司 | α-D-吡喃半乳糖苷衍生物 |
-
2022
- 2022-03-02 RS RS20250732A patent/RS67032B1/sr unknown
- 2022-03-02 PL PL22708569.3T patent/PL4301748T3/pl unknown
- 2022-03-02 WO PCT/EP2022/055224 patent/WO2022184755A1/en not_active Ceased
- 2022-03-02 AU AU2022228660A patent/AU2022228660A1/en active Pending
- 2022-03-02 HR HRP20250833TT patent/HRP20250833T1/hr unknown
- 2022-03-02 UA UAA202304634A patent/UA130562C2/uk unknown
- 2022-03-02 BR BR112023017624A patent/BR112023017624A2/pt unknown
- 2022-03-02 ES ES22708569T patent/ES3033422T3/es active Active
- 2022-03-02 KR KR1020237033375A patent/KR20230154221A/ko active Pending
- 2022-03-02 IL IL305581A patent/IL305581A/en unknown
- 2022-03-02 US US18/548,833 patent/US20240109930A1/en active Pending
- 2022-03-02 EP EP22708569.3A patent/EP4301748B1/en active Active
- 2022-03-02 CA CA3209917A patent/CA3209917A1/en active Pending
- 2022-03-02 MA MA63589A patent/MA63589B1/fr unknown
- 2022-03-02 TW TW111107565A patent/TWI905393B/zh active
- 2022-03-02 JP JP2023552539A patent/JP7771205B2/ja active Active
- 2022-03-02 MX MX2023010241A patent/MX2023010241A/es unknown
- 2022-03-02 HU HUE22708569A patent/HUE072194T2/hu unknown
- 2022-03-02 CN CN202280017484.3A patent/CN116888113A/zh active Pending
-
2023
- 2023-08-31 CL CL2023002578A patent/CL2023002578A1/es unknown
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2024509421A5 (https=) | ||
| HRP20250833T1 (hr) | Derivati alfa-d-galaktopiranozida supstituirani triazolil metilom | |
| JP2024506182A5 (https=) | ||
| US9079878B2 (en) | (4-phenylimidazol-2-yl) ethylamine derivatives useful as sodium channel modulators | |
| US8796253B2 (en) | Heteroaryl substituted pyrazole derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis | |
| JP2022544248A5 (https=) | ||
| JP2023547241A5 (https=) | ||
| JP2022546029A5 (https=) | ||
| JP7604457B2 (ja) | 2-ヒドロキシシクロアルカン-1-カルバモイル誘導体 | |
| JP2022554169A5 (https=) | ||
| IL276031B2 (en) | oxazine monoacylglycerol lipase (magl) inhibitors | |
| JP2021532124A5 (https=) | ||
| JP2022543859A5 (https=) | ||
| JP2019515931A5 (https=) | ||
| JP2023545046A5 (https=) | ||
| JP2022534261A5 (https=) | ||
| US20120142691A1 (en) | Picolinamide derivatives as ttx-s blockers | |
| JP2010508307A5 (https=) | ||
| JP2022543666A5 (https=) | ||
| JP2022530049A5 (https=) | ||
| US20130274243A1 (en) | Chemical Compounds | |
| EA032609B1 (ru) | Соединения аминопиримидинила в качестве ингибиторов jak | |
| NL2000284C2 (nl) | Pyrazine-derivaten. | |
| JP6208212B2 (ja) | 呼吸器疾患用薬 | |
| EA029280B1 (ru) | Новые ингибиторы cyp17/антиандрогены |