JP2023546742A5 - - Google Patents

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Publication number
JP2023546742A5
JP2023546742A5 JP2023548994A JP2023548994A JP2023546742A5 JP 2023546742 A5 JP2023546742 A5 JP 2023546742A5 JP 2023548994 A JP2023548994 A JP 2023548994A JP 2023548994 A JP2023548994 A JP 2023548994A JP 2023546742 A5 JP2023546742 A5 JP 2023546742A5
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JP
Japan
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independently selected
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appropriately substituted
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Pending
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JP2023548994A
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English (en)
Japanese (ja)
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JP2023546742A (ja
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Priority claimed from PCT/CN2021/125409 external-priority patent/WO2022083703A1/en
Publication of JP2023546742A publication Critical patent/JP2023546742A/ja
Publication of JP2023546742A5 publication Critical patent/JP2023546742A5/ja
Pending legal-status Critical Current

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JP2023548994A 2020-10-22 2021-10-21 Lpa受容体活性に付随する症状を治療するための化合物および組成物 Pending JP2023546742A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
CNPCT/CN2020/122794 2020-10-22
CN2020122794 2020-10-22
CN2021113042 2021-08-17
CNPCT/CN2021/113042 2021-08-17
CN2021122851 2021-10-09
CNPCT/CN2021/122851 2021-10-09
PCT/CN2021/125409 WO2022083703A1 (en) 2020-10-22 2021-10-21 Compounds and compositions for treating conditions associated with lpa receptor activity

Publications (2)

Publication Number Publication Date
JP2023546742A JP2023546742A (ja) 2023-11-07
JP2023546742A5 true JP2023546742A5 (https=) 2024-10-29

Family

ID=78516438

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023548994A Pending JP2023546742A (ja) 2020-10-22 2021-10-21 Lpa受容体活性に付随する症状を治療するための化合物および組成物

Country Status (7)

Country Link
US (1) US20240018102A1 (https=)
EP (2) EP4232431B1 (https=)
JP (1) JP2023546742A (https=)
CN (1) CN116583501A (https=)
ES (1) ES3049795T3 (https=)
TW (1) TW202233575A (https=)
WO (1) WO2022083703A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4419509A4 (en) * 2021-10-21 2025-10-15 Lhotse Bio Inc COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH LPA RECEPTOR ACTIVITY
TW202342017A (zh) 2022-02-25 2023-11-01 美商洛子峰生物有限公司 用於治療與lpa受體活性相關的病狀的化合物及組合物
WO2026002179A1 (en) * 2024-06-28 2026-01-02 Rezubio Pharmaceuticals Co., Ltd Compounds and compositions

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7820682B2 (en) * 2002-10-03 2010-10-26 Ono Pharmaceutical Co., Ltd. LPA receptor antagonist
ATE528276T1 (de) * 2003-12-19 2011-10-15 Ono Pharmaceutical Co Lysophosphatidylsäurerezeptor-antagonistische verbindungen und ihre anwendungen
CN101119714A (zh) * 2005-02-14 2008-02-06 弗吉尼亚大学专利基金会 含有由氨基和苯基取代的环烷基和5元杂环的1-磷酸鞘氨醇激动剂
JP2014525932A (ja) * 2011-08-15 2014-10-02 インターミューン, インコーポレイテッド リゾホスファチド酸レセプターアンタゴニスト
AR108838A1 (es) * 2016-06-21 2018-10-03 Bristol Myers Squibb Co Ácidos de carbamoiloximetil triazol ciclohexilo como antagonistas de lpa
CN111712492B (zh) * 2017-12-19 2024-05-31 百时美施贵宝公司 作为lpa拮抗剂的环己基酸三唑唑类
US11447475B2 (en) * 2017-12-19 2022-09-20 Bristol-Myers Squibb Company Isoxazole N-linked carbamoyl cyclohexyl acids as LPA antagonists

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