JP2011519360A5 - - Google Patents
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- Publication number
- JP2011519360A5 JP2011519360A5 JP2011504995A JP2011504995A JP2011519360A5 JP 2011519360 A5 JP2011519360 A5 JP 2011519360A5 JP 2011504995 A JP2011504995 A JP 2011504995A JP 2011504995 A JP2011504995 A JP 2011504995A JP 2011519360 A5 JP2011519360 A5 JP 2011519360A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- cycloalkyl
- alkylene
- heterocycloalkyl
- aryl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 C**(CC1)CN1C1=*C(*)=[U]C(N*C2CCC(*N*)CC2)=N1 Chemical compound C**(CC1)CN1C1=*C(*)=[U]C(N*C2CCC(*N*)CC2)=N1 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US4649608P | 2008-04-21 | 2008-04-21 | |
| US61/046,496 | 2008-04-21 | ||
| PCT/US2008/082202 WO2009131598A1 (en) | 2008-04-21 | 2008-11-03 | Heterocyclic compounds |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011519360A JP2011519360A (ja) | 2011-07-07 |
| JP2011519360A5 true JP2011519360A5 (https=) | 2012-01-19 |
| JP5661607B2 JP5661607B2 (ja) | 2015-01-28 |
Family
ID=41201620
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011504995A Active JP5661607B2 (ja) | 2008-04-21 | 2008-11-03 | 複素環化合物 |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US8372849B2 (https=) |
| EP (1) | EP2268635B1 (https=) |
| JP (1) | JP5661607B2 (https=) |
| KR (1) | KR101579999B1 (https=) |
| CN (1) | CN101565404B (https=) |
| AU (1) | AU2008355098B2 (https=) |
| CA (1) | CA2720229C (https=) |
| CY (1) | CY1116802T1 (https=) |
| DK (1) | DK2268635T3 (https=) |
| EA (1) | EA019289B1 (https=) |
| ES (1) | ES2545731T3 (https=) |
| HR (1) | HRP20150932T2 (https=) |
| HU (1) | HUE025179T2 (https=) |
| NZ (1) | NZ588989A (https=) |
| PL (1) | PL2268635T3 (https=) |
| PT (1) | PT2268635E (https=) |
| SI (1) | SI2268635T1 (https=) |
| TW (1) | TWI444188B (https=) |
| WO (1) | WO2009131598A1 (https=) |
| ZA (1) | ZA201008262B (https=) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9023834B2 (en) * | 2008-11-13 | 2015-05-05 | Taigen Biotechnology Co., Ltd. | Lyophilization formulation |
| CN103204816B (zh) * | 2012-01-16 | 2016-04-27 | 中国人民解放军军事医学科学院毒物药物研究所 | 哌嗪基嘧啶类衍生物及其制备方法和用途 |
| WO2013155347A1 (en) * | 2012-04-11 | 2013-10-17 | Izumi Raquel | Bruton's tyrosine kinase inhibitors for hematopoietic mobilization |
| ES2849998T3 (es) | 2014-09-22 | 2021-08-24 | National Health Res Inst | Compuestos heterocíclicos y su uso |
| US9375406B2 (en) * | 2014-09-30 | 2016-06-28 | Taigen Biotechnology Co., Ltd. | Substituted pyrimidines for mobilizing cells expressing a type 4 CXC chemokine receptor |
| TWI620748B (zh) | 2016-02-05 | 2018-04-11 | National Health Research Institutes | 氨基噻唑化合物及其用途 |
| RU2756055C2 (ru) * | 2017-01-10 | 2021-09-24 | Нэшнл Хелт Рисерч Инститьютс | Гетероциклические соединения и их применение |
| CN109553604B (zh) * | 2017-09-25 | 2021-08-27 | 盛世泰科生物医药技术(苏州)有限公司 | 4-氨基嘧啶衍生物作cxcr4抑制剂及其应用 |
| CN108794414B (zh) * | 2018-06-22 | 2021-01-01 | 浙江大学 | 芳酰胺基取代的均三嗪类化合物及制备和应用 |
| CN116120195B (zh) * | 2022-12-29 | 2025-02-25 | 长兴宜生药物科技有限公司 | 一种催化制备培哚普利中间体的方法 |
| PL247377B1 (pl) * | 2023-06-29 | 2025-06-23 | Politechnika Krakowska Im Tadeusza Kosciuszki | Nowa pochodna 1,3,5-triazyny i jej zastosowanie |
Family Cites Families (36)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6029A (en) * | 1849-01-16 | Method of directing the scoops in dredging machines | ||
| US3007A (en) * | 1843-03-21 | Improvement in salt-boilers | ||
| US5034560A (en) * | 1990-10-19 | 1991-07-23 | The Standard Oil Company | Synthesis of ethylamines |
| DK0594772T3 (https=) | 1991-07-04 | 1997-02-24 | Immunodex K S | |
| US5446090A (en) | 1993-11-12 | 1995-08-29 | Shearwater Polymers, Inc. | Isolatable, water soluble, and hydrolytically stable active sulfones of poly(ethylene glycol) and related polymers for modification of surfaces and molecules |
| IL112795A (en) | 1994-03-04 | 2001-01-28 | Astrazeneca Ab | Peptide derivatives as antithrombic agents their preparation and pharmaceutical compositions containing them |
| AU7692996A (en) | 1995-12-01 | 1997-06-27 | Ciba-Geigy Ag | Receptor antagonists |
| TW440563B (en) | 1996-05-23 | 2001-06-16 | Hoffmann La Roche | Aryl pyrimidine derivatives and a pharmaceutical composition thereof |
| AU3295297A (en) | 1996-06-04 | 1998-01-05 | Synaptic Pharmaceutical Corporation | Methods of modifying feeding behavior, compounds useful in such methods, and dna encoding a hypothalamic atypical neuropeptide y/peptide yy receptor (y5) |
| NO311614B1 (no) * | 1996-10-01 | 2001-12-17 | Janssen Pharmaceutica Nv | Substituerte diamino-1,3,5-triazinderivater |
| TW520362B (en) * | 1996-12-05 | 2003-02-11 | Amgen Inc | Substituted pyrimidine compounds and pharmaceutical composition comprising same |
| JP2003504301A (ja) | 1998-04-01 | 2003-02-04 | ブリストル−マイヤーズ スクイブ ファーマ カンパニー | インテグリンアンタゴニスト |
| US6420354B1 (en) * | 1998-06-08 | 2002-07-16 | Advanced Medicine, Inc. | Sodium channel drugs and uses |
| HUP0103622A3 (en) | 1998-08-20 | 2003-01-28 | Agouron Pharmaceuticals Inc La | Non-peptide gnrh agents, methods and intermediates for their preparation and medicaments containing them |
| GB9905075D0 (en) | 1999-03-06 | 1999-04-28 | Zeneca Ltd | Chemical compounds |
| US6274588B1 (en) | 1999-05-31 | 2001-08-14 | Hoffmann-La Roche Inc. | 4-phenyl-pyrimidine derivatives |
| EP1246823A1 (en) * | 1999-12-28 | 2002-10-09 | Pharmacopeia, Inc. | Pyrimidine and triazine kinase inhibitors |
| US6989385B2 (en) | 2000-12-21 | 2006-01-24 | Vertex Pharmaceuticals Incorporated | Pyrazole compounds useful as protein kinase inhibitors |
| CN101851173A (zh) * | 2001-09-14 | 2010-10-06 | 梅特希尔基因公司 | 组蛋白脱乙酰化酶抑制剂 |
| US6897220B2 (en) | 2001-09-14 | 2005-05-24 | Methylgene, Inc. | Inhibitors of histone deacetylase |
| WO2003026664A1 (en) | 2001-09-26 | 2003-04-03 | Bayer Corporation | 2-phenylamino-4- (5-pyrazolylamino) -pyramidine derivatives as kinase inhibitors, in particular, src kinase inhibitors |
| EP1432693A2 (en) | 2001-10-01 | 2004-06-30 | Taisho Pharmaceutical Co. Ltd. | Mch receptor antagonists |
| EP1518855B1 (en) | 2002-06-28 | 2011-10-26 | Astellas Pharma Inc. | Diaminopyrimidinecarboxa mide derivative |
| EP1571146A4 (en) * | 2002-12-10 | 2010-09-01 | Ono Pharmaceutical Co | NITROGENIC HETEROCYCLIC COMPOUNDS AND THEIR MEDICAL USE |
| US20040242613A1 (en) * | 2003-01-30 | 2004-12-02 | Boehringer Ingelheim Pharmaceuticals, Inc. | Pyrimidine derivatives useful as inhibitors of PKC-theta |
| JP4339890B2 (ja) | 2003-09-22 | 2009-10-07 | エフ．ホフマン−ラ ロシュ アーゲー | アミノアルキルアミド置換シクロヘキシル誘導体 |
| MXPA06010900A (es) * | 2004-03-26 | 2007-02-21 | Methylgene Inc | Inhibidores de histona desacetilasa. |
| EP3461813A1 (en) | 2004-05-23 | 2019-04-03 | Gerard M. Housey | Theramutein modulators |
| JP2006124387A (ja) * | 2004-09-30 | 2006-05-18 | Taisho Pharmaceut Co Ltd | 新規なキノリン、テトラヒドロキナゾリン、及びピリミジン誘導体と、これらを使用することに関連した治療方法 |
| NZ564222A (en) * | 2005-06-14 | 2011-10-28 | Taigen Biotechnology Co Ltd | Pyrimidine compounds |
| EP1928847A4 (en) | 2005-08-29 | 2011-08-10 | Gerard M Housey | THERAMUTEINE MODULATORS |
| KR101415426B1 (ko) | 2005-09-27 | 2014-07-04 | 아이알엠 엘엘씨 | 디아릴아민-함유 화합물 및 조성물, 및 ｃ-ｋｉｔ 수용체의조절제로서의 그의 용도 |
| CN103789389B (zh) | 2005-11-23 | 2017-01-04 | 杰勒德·M·豪斯 | 鉴定、合成、优化和表征蛋白调节剂的化合物和方法 |
| CN101563336A (zh) | 2006-03-16 | 2009-10-21 | 诺瓦提斯公司 | 用于治疗特别是黑素瘤的杂环有机化合物 |
| WO2007129195A2 (en) | 2006-05-04 | 2007-11-15 | Pfizer Products Inc. | 4-pyrimidine-5-amino-pyrazole compounds |
| EP2043651A2 (en) * | 2006-07-05 | 2009-04-08 | Exelixis, Inc. | Methods of using igf1r and abl kinase modulators |
-
2008
- 2008-11-03 DK DK08874003.0T patent/DK2268635T3/en active
- 2008-11-03 KR KR1020107025309A patent/KR101579999B1/ko active Active
- 2008-11-03 ES ES08874003.0T patent/ES2545731T3/es active Active
- 2008-11-03 PT PT88740030T patent/PT2268635E/pt unknown
- 2008-11-03 EP EP08874003.0A patent/EP2268635B1/en active Active
- 2008-11-03 NZ NZ588989A patent/NZ588989A/en unknown
- 2008-11-03 AU AU2008355098A patent/AU2008355098B2/en active Active
- 2008-11-03 CA CA2720229A patent/CA2720229C/en active Active
- 2008-11-03 JP JP2011504995A patent/JP5661607B2/ja active Active
- 2008-11-03 HR HRP20150932TT patent/HRP20150932T2/hr unknown
- 2008-11-03 SI SI200831498T patent/SI2268635T1/sl unknown
- 2008-11-03 PL PL08874003T patent/PL2268635T3/pl unknown
- 2008-11-03 HU HUE08874003A patent/HUE025179T2/en unknown
- 2008-11-03 EA EA201071221A patent/EA019289B1/ru unknown
- 2008-11-03 US US12/263,671 patent/US8372849B2/en active Active
- 2008-11-03 WO PCT/US2008/082202 patent/WO2009131598A1/en not_active Ceased
- 2008-11-05 TW TW097142682A patent/TWI444188B/zh active
- 2008-12-01 CN CN2008101796944A patent/CN101565404B/zh active Active
-
2010
- 2010-11-18 ZA ZA2010/08262A patent/ZA201008262B/en unknown
-
2015
- 2015-09-07 CY CY20151100774T patent/CY1116802T1/el unknown
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