JP2023542218A5 - - Google Patents

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Publication number
JP2023542218A5
JP2023542218A5 JP2023518426A JP2023518426A JP2023542218A5 JP 2023542218 A5 JP2023542218 A5 JP 2023542218A5 JP 2023518426 A JP2023518426 A JP 2023518426A JP 2023518426 A JP2023518426 A JP 2023518426A JP 2023542218 A5 JP2023542218 A5 JP 2023542218A5
Authority
JP
Japan
Prior art keywords
conjugate
salt
cancer
radionuclide
use according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2023518426A
Other languages
English (en)
Japanese (ja)
Other versions
JP7824281B2 (ja
JP2023542218A (ja
Filing date
Publication date
Priority claimed from EP20306109.8A external-priority patent/EP3973999A1/en
Application filed filed Critical
Publication of JP2023542218A publication Critical patent/JP2023542218A/ja
Publication of JP2023542218A5 publication Critical patent/JP2023542218A5/ja
Application granted granted Critical
Publication of JP7824281B2 publication Critical patent/JP7824281B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2023518426A 2020-09-28 2021-09-22 ガストリン放出ペプチド受容体アンタゴニストを含むコンジュゲートまたはその塩およびそれらの使用 Active JP7824281B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP20306109.8 2020-09-28
EP20306109.8A EP3973999A1 (en) 2020-09-28 2020-09-28 Conjugate or its salt comprising a gastrin-releasing peptide receptor antagonist and uses thereof
PCT/EP2021/076107 WO2022063850A1 (en) 2020-09-28 2021-09-22 Conjugate or its salt comprising a gastrin-releasing peptide receptor antagonist and uses thereof

Publications (3)

Publication Number Publication Date
JP2023542218A JP2023542218A (ja) 2023-10-05
JP2023542218A5 true JP2023542218A5 (enExample) 2024-07-09
JP7824281B2 JP7824281B2 (ja) 2026-03-04

Family

ID=74180915

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023518426A Active JP7824281B2 (ja) 2020-09-28 2021-09-22 ガストリン放出ペプチド受容体アンタゴニストを含むコンジュゲートまたはその塩およびそれらの使用

Country Status (21)

Country Link
US (1) US20230372552A1 (enExample)
EP (2) EP3973999A1 (enExample)
JP (1) JP7824281B2 (enExample)
KR (1) KR20230078690A (enExample)
CN (1) CN116322798A (enExample)
AU (1) AU2021348219A1 (enExample)
BR (1) BR112023003690A2 (enExample)
CA (1) CA3189680A1 (enExample)
DK (1) DK4188457T3 (enExample)
ES (1) ES2989009T3 (enExample)
FI (1) FI4188457T3 (enExample)
HR (1) HRP20241285T1 (enExample)
HU (1) HUE068360T2 (enExample)
IL (1) IL300486A (enExample)
LT (1) LT4188457T (enExample)
PL (1) PL4188457T3 (enExample)
PT (1) PT4188457T (enExample)
RS (1) RS65994B1 (enExample)
SI (1) SI4188457T1 (enExample)
SM (1) SMT202400392T1 (enExample)
WO (1) WO2022063850A1 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2025163082A1 (en) 2024-01-31 2025-08-07 Molecular Partners Ag Dll3-specific binding constructs and their use in radiotherapy
WO2026150109A1 (en) 2025-01-10 2026-07-16 Molecular Partners Ag Mesothelin-specific binding constructs and their use in radiotherapy

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2100900A1 (en) 2008-03-07 2009-09-16 Universitätsspital Basel Bombesin analog peptide antagonist conjugates
US20150217006A1 (en) * 2014-02-06 2015-08-06 Immunomedics, Inc. Al-f-18-labeled, al-f-19-labeled and ga-68-labeled gastrin-releasing peptide receptor (grpr)-antagonists for imaging of prostate cancer
CA3050094C (en) 2017-01-12 2024-01-02 Radiomedix Inc. Treatment of cancer cells overexpressing somatostatin receptors using ocreotide derivatives chelated to radioisotopes

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