JP2023527961A - gpr39タンパク質のアンタゴニスト - Google Patents
gpr39タンパク質のアンタゴニスト Download PDFInfo
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- JP2023527961A JP2023527961A JP2022566301A JP2022566301A JP2023527961A JP 2023527961 A JP2023527961 A JP 2023527961A JP 2022566301 A JP2022566301 A JP 2022566301A JP 2022566301 A JP2022566301 A JP 2022566301A JP 2023527961 A JP2023527961 A JP 2023527961A
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| US202063018371P | 2020-04-30 | 2020-04-30 | |
| US63/018,371 | 2020-04-30 | ||
| PCT/US2021/030335 WO2021222858A1 (en) | 2020-04-30 | 2021-04-30 | Antagonists of gpr39 protein |
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| EP4486722A4 (en) * | 2022-03-02 | 2026-03-25 | Nico Therapeutics Inc | COMPOUNDS, COMPOSITIONS AND PROCESSES |
| CN117224684A (zh) * | 2023-09-27 | 2023-12-15 | 南京医科大学姑苏学院 | Gpr39抑制剂在制备预防或治疗高血压疾病的药物中的应用 |
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| JP2017509601A (ja) * | 2014-02-14 | 2017-04-06 | 武田薬品工業株式会社 | Gpr6のピラジンモジュレーター |
| WO2018124000A1 (ja) * | 2016-12-27 | 2018-07-05 | 第一三共株式会社 | ピリミジン誘導体 |
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| DE10164564B4 (de) * | 2001-12-14 | 2007-05-16 | Zentaris Gmbh | Tetrahydrocarbazolderivate als Liganden für G-Protein gekoppelte Rezeptoren (GPCR) |
| US20040071708A1 (en) | 2002-09-26 | 2004-04-15 | Immusol, Inc. | GPR 39 modulators that control cancerous cell growth |
| WO2004099782A2 (en) * | 2003-05-05 | 2004-11-18 | Bayer Healthcare Ag | Diagnostics and therapeutics for diseases associated with g-protein-coupled receptor gpr39 (gpr39) |
| US7459460B2 (en) * | 2003-05-28 | 2008-12-02 | Bristol-Myers Squibb Company | Trisubstituted heteroaromatic compounds as calcium sensing receptor modulators |
| US7767680B2 (en) * | 2004-11-03 | 2010-08-03 | Vertex Pharmaceuticals Incorporated | Ion channel modulators and methods of use |
| CN1850269A (zh) | 2005-04-22 | 2006-10-25 | 中国科学院上海生命科学研究院 | Gpr39基因在哺乳动物中枢神经系统的功能及其应用 |
| MX2008015670A (es) | 2006-06-08 | 2009-01-12 | Janssen Pharmaceutica Nv | Receptor 39 acoplado a proteina g (gpr39). |
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- 2021-04-30 WO PCT/US2021/030335 patent/WO2021222858A1/en not_active Ceased
- 2021-04-30 CN CN202180046666.9A patent/CN115996908B/zh active Active
- 2021-04-30 KR KR1020227041846A patent/KR20230017787A/ko active Pending
- 2021-04-30 EP EP21727055.2A patent/EP4143163A1/en active Pending
- 2021-04-30 JP JP2022566301A patent/JP2023527961A/ja active Pending
- 2021-04-30 US US17/997,533 patent/US20230174484A1/en active Pending
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| JP2017509601A (ja) * | 2014-02-14 | 2017-04-06 | 武田薬品工業株式会社 | Gpr6のピラジンモジュレーター |
| WO2018124000A1 (ja) * | 2016-12-27 | 2018-07-05 | 第一三共株式会社 | ピリミジン誘導体 |
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Also Published As
| Publication number | Publication date |
|---|---|
| CN115996908A (zh) | 2023-04-21 |
| CN115996908B (zh) | 2026-04-24 |
| EP4143163A1 (en) | 2023-03-08 |
| US20230174484A1 (en) | 2023-06-08 |
| WO2021222858A1 (en) | 2021-11-04 |
| KR20230017787A (ko) | 2023-02-06 |
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