JP2023512227A5 - - Google Patents

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Publication number
JP2023512227A5
JP2023512227A5 JP2022545915A JP2022545915A JP2023512227A5 JP 2023512227 A5 JP2023512227 A5 JP 2023512227A5 JP 2022545915 A JP2022545915 A JP 2022545915A JP 2022545915 A JP2022545915 A JP 2022545915A JP 2023512227 A5 JP2023512227 A5 JP 2023512227A5
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JP
Japan
Prior art keywords
alkanediyl
alkyl
cycloalkyl
compound according
cancer
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JP2022545915A
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English (en)
Japanese (ja)
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JP2023512227A (ja
JP7698653B2 (ja
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Priority claimed from PCT/US2021/014977 external-priority patent/WO2021154663A1/en
Publication of JP2023512227A publication Critical patent/JP2023512227A/ja
Publication of JP2023512227A5 publication Critical patent/JP2023512227A5/ja
Application granted granted Critical
Publication of JP7698653B2 publication Critical patent/JP7698653B2/ja
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JP2022545915A 2020-01-27 2021-01-26 トール様受容体7(TLR7)アゴニストとしての1H-ピラゾロ[4,3-d]ピリミジン化合物 Active JP7698653B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062966111P 2020-01-27 2020-01-27
US62/966,111 2020-01-27
PCT/US2021/014977 WO2021154663A1 (en) 2020-01-27 2021-01-26 1H-PYRAZOLO[4,3-d]PYRIMIDINE COMPOUNDS AS TOLL-LIKE RECEPTOR 7 (TLR7) AGONISTS

Publications (3)

Publication Number Publication Date
JP2023512227A JP2023512227A (ja) 2023-03-24
JP2023512227A5 true JP2023512227A5 (https=) 2024-02-02
JP7698653B2 JP7698653B2 (ja) 2025-06-25

Family

ID=74661498

Family Applications (1)

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JP2022545915A Active JP7698653B2 (ja) 2020-01-27 2021-01-26 トール様受容体7(TLR7)アゴニストとしての1H-ピラゾロ[4,3-d]ピリミジン化合物

Country Status (6)

Country Link
US (1) US20230122249A1 (https=)
EP (1) EP4097104A1 (https=)
JP (1) JP7698653B2 (https=)
KR (1) KR20220132591A (https=)
CN (1) CN115210235A (https=)
WO (1) WO2021154663A1 (https=)

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WO2021154661A1 (en) * 2020-01-27 2021-08-05 Bristol-Myers Squibb Company 1H-PYRAZOLO[4,3-d]PYRIMIDINE COMPOUNDS AS TOLL-LIKE RECEPTOR 7 (TLR7) AGONISTS
WO2021154662A1 (en) * 2020-01-27 2021-08-05 Bristol-Myers Squibb Company 1H-PYRAZOLO[4,3-d]PYRIMIDINE COMPOUNDS AS TOLL-LIKE RECEPTOR 7 (TLR7) AGONISTS
EP4097105A1 (en) * 2020-01-27 2022-12-07 Bristol-Myers Squibb Company 1h-pyrazolo[4,3-d]pyrimidine compounds as toll-like receptor 7 (tlr7) agonists
AR122043A1 (es) * 2020-05-12 2022-08-03 Bristol Myers Squibb Co Dosificación y administración del anticuerpo anti-ctla-4 activable

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WO2021154662A1 (en) * 2020-01-27 2021-08-05 Bristol-Myers Squibb Company 1H-PYRAZOLO[4,3-d]PYRIMIDINE COMPOUNDS AS TOLL-LIKE RECEPTOR 7 (TLR7) AGONISTS
KR20220132601A (ko) * 2020-01-27 2022-09-30 브리스톨-마이어스 스큅 컴퍼니 톨-유사 수용체 7 (TLR7) 효능제로서의 1H-피라졸로[4,3-d]피리미딘 화합물

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