JP2023512206A5 - - Google Patents

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Publication number
JP2023512206A5
JP2023512206A5 JP2022545790A JP2022545790A JP2023512206A5 JP 2023512206 A5 JP2023512206 A5 JP 2023512206A5 JP 2022545790 A JP2022545790 A JP 2022545790A JP 2022545790 A JP2022545790 A JP 2022545790A JP 2023512206 A5 JP2023512206 A5 JP 2023512206A5
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JP
Japan
Prior art keywords
alkyl
alkanediyl
cycloalkyl
cancer
formula
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022545790A
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English (en)
Japanese (ja)
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JP2023512206A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/014980 external-priority patent/WO2021154666A1/en
Publication of JP2023512206A publication Critical patent/JP2023512206A/ja
Publication of JP2023512206A5 publication Critical patent/JP2023512206A5/ja
Pending legal-status Critical Current

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JP2022545790A 2020-01-27 2021-01-26 トール様受容体7(TLR7)アゴニストとしての1H-ピラゾロ[4,3-d]ピリミジン化合物 Pending JP2023512206A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202062966144P 2020-01-27 2020-01-27
US62/966,144 2020-01-27
US202063058230P 2020-07-29 2020-07-29
US63/058,230 2020-07-29
PCT/US2021/014980 WO2021154666A1 (en) 2020-01-27 2021-01-26 1H-PYRAZOLO[4,3-d]PYRIMIDINE COMPOUNDS AS TOLL-LIKE RECEPTOR 7 (TLR7) AGONISTS

Publications (2)

Publication Number Publication Date
JP2023512206A JP2023512206A (ja) 2023-03-24
JP2023512206A5 true JP2023512206A5 (https=) 2024-02-02

Family

ID=74595468

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022545790A Pending JP2023512206A (ja) 2020-01-27 2021-01-26 トール様受容体7(TLR7)アゴニストとしての1H-ピラゾロ[4,3-d]ピリミジン化合物

Country Status (6)

Country Link
US (1) US20230348468A1 (https=)
EP (1) EP4097100A1 (https=)
JP (1) JP2023512206A (https=)
KR (1) KR20220132593A (https=)
CN (1) CN115151548A (https=)
WO (1) WO2021154666A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021154661A1 (en) * 2020-01-27 2021-08-05 Bristol-Myers Squibb Company 1H-PYRAZOLO[4,3-d]PYRIMIDINE COMPOUNDS AS TOLL-LIKE RECEPTOR 7 (TLR7) AGONISTS
WO2021154662A1 (en) * 2020-01-27 2021-08-05 Bristol-Myers Squibb Company 1H-PYRAZOLO[4,3-d]PYRIMIDINE COMPOUNDS AS TOLL-LIKE RECEPTOR 7 (TLR7) AGONISTS
EP4097105A1 (en) * 2020-01-27 2022-12-07 Bristol-Myers Squibb Company 1h-pyrazolo[4,3-d]pyrimidine compounds as toll-like receptor 7 (tlr7) agonists
CN115279765B (zh) * 2020-01-27 2024-11-12 百时美施贵宝公司 作为Toll样受体7(TLR7)激动剂的1H-吡唑并[4,3-d]嘧啶化合物

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