JP2023119042A5 - - Google Patents

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Publication number
JP2023119042A5
JP2023119042A5 JP2023113057A JP2023113057A JP2023119042A5 JP 2023119042 A5 JP2023119042 A5 JP 2023119042A5 JP 2023113057 A JP2023113057 A JP 2023113057A JP 2023113057 A JP2023113057 A JP 2023113057A JP 2023119042 A5 JP2023119042 A5 JP 2023119042A5
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Japan
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alkyl
compound
item
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JP2023113057A
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Japanese (ja)
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JP7689160B2 (ja
JP2023119042A (ja
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Priority claimed from PCT/US2018/067306 external-priority patent/WO2019126761A1/en
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Priority to JP2025034943A priority Critical patent/JP2025078783A/ja
Publication of JP2023119042A5 publication Critical patent/JP2023119042A5/ja
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JP2023113057A 2017-12-22 2023-07-10 Ｃｎｓ障害の処置のための組成物および方法 Active JP7689160B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025034943A JP2025078783A (ja) 2017-12-22 2025-03-05 Ｃｎｓ障害の処置のための組成物および方法

Applications Claiming Priority (20)

Application Number Priority Date Filing Date Title
US201762610067P 2017-12-22 2017-12-22
US62/610,067 2017-12-22
US201762612067P 2017-12-29 2017-12-29
US201762612070P 2017-12-29 2017-12-29
US201762611977P 2017-12-29 2017-12-29
US201762612164P 2017-12-29 2017-12-29
US62/611,977 2017-12-29
US62/612,164 2017-12-29
US62/612,067 2017-12-29
US62/612,070 2017-12-29
US201862765164P 2018-08-17 2018-08-17
US62/765,164 2018-08-17
US201862728499P 2018-09-07 2018-09-07
US62/728,499 2018-09-07
US201862737559P 2018-09-27 2018-09-27
US62/737,559 2018-09-27
US201862754977P 2018-11-02 2018-11-02
US62/754,977 2018-11-02
PCT/US2018/067306 WO2019126761A1 (en) 2017-12-22 2018-12-21 Compositions and methods for treating cns disorders
JP2020534302A JP2021506904A (ja) 2017-12-22 2018-12-21 Ｃｎｓ障害の処置のための組成物および方法

Related Parent Applications (1)

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JP2020534302A Division JP2021506904A (ja) 2017-12-22 2018-12-21 Ｃｎｓ障害の処置のための組成物および方法

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025034943A Division JP2025078783A (ja) 2017-12-22 2025-03-05 Ｃｎｓ障害の処置のための組成物および方法

Publications (3)

Publication Number Publication Date
JP2023119042A JP2023119042A (ja) 2023-08-25
JP2023119042A5 true JP2023119042A5 (enExample) 2025-03-14
JP7689160B2 JP7689160B2 (ja) 2025-06-05

Family

ID=65234664

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2020534302A Withdrawn JP2021506904A (ja) 2017-12-22 2018-12-21 Ｃｎｓ障害の処置のための組成物および方法
JP2023113057A Active JP7689160B2 (ja) 2017-12-22 2023-07-10 Ｃｎｓ障害の処置のための組成物および方法
JP2025034943A Pending JP2025078783A (ja) 2017-12-22 2025-03-05 Ｃｎｓ障害の処置のための組成物および方法

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2020534302A Withdrawn JP2021506904A (ja) 2017-12-22 2018-12-21 Ｃｎｓ障害の処置のための組成物および方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025034943A Pending JP2025078783A (ja) 2017-12-22 2025-03-05 Ｃｎｓ障害の処置のための組成物および方法

Country Status (13)

Country Link
US (2) US20220315621A1 (enExample)
EP (1) EP3728285A1 (enExample)
JP (3) JP2021506904A (enExample)
KR (1) KR20200104349A (enExample)
CN (3) CN118085004A (enExample)
AR (1) AR114044A1 (enExample)
AU (2) AU2018392093B2 (enExample)
BR (1) BR112020012761A2 (enExample)
CA (1) CA3086189A1 (enExample)
IL (1) IL275506A (enExample)
MA (1) MA51316A (enExample)
MX (3) MX2020006608A (enExample)
WO (1) WO2019126761A1 (enExample)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ773177A (en) 2012-01-23 2022-09-30 Sage Therapeutics Inc Neuroactive steroid formulations and methods of treating cns disorders
IL275725B (en) 2012-08-21 2022-08-01 Sage Therapeutics Inc Treatment methods for epilepsy and status epilepticus
AU2014256229B2 (en) 2013-04-17 2018-10-04 Sage Therapeutics, Inc. 19-nor C3,3-disubstituted C21-N-pyrazolyl steroids and methods of use thereof
US10246482B2 (en) 2014-06-18 2019-04-02 Sage Therapeutics, Inc. Neuroactive steroids, compositions, and uses thereof
JOP20200195A1 (ar) 2014-09-08 2017-06-16 Sage Therapeutics Inc سترويدات وتركيبات نشطة عصبياً، واستخداماتها
US10774108B2 (en) 2014-11-27 2020-09-15 Sage Therapeutics, Inc. Compositions and methods for treating CNS disorders
NZ791594A (en) 2016-08-23 2025-08-29 Sage Therapeutics Inc A crystalline 19-nor C3, 3-disubstituted C21-N-pyrazolyl steroid
WO2019113494A1 (en) 2017-12-08 2019-06-13 Sage Therapeutics, Inc. Deuterated 21 -[4-cyano-pyrazol-1 -yl]-19-nor-pregan-3. alpha-ol-20-one derivatives for treating cns disorders
AR114044A1 (es) 2017-12-22 2020-07-15 Sage Therapeutics Inc Composiciones y métodos para el tratamiento de trastornos en el sistema nervioso central
EP3737687B1 (en) 2018-01-12 2025-10-22 Sage Therapeutics, Inc. Aza-, oxa and thia-pregnan-20-one-3.alpha.-ol compounds for use in treating cns disorders
ES3018614T3 (es) * 2018-02-11 2025-05-16 Jiangsu Hansoh Pharmaceutical Group Co Ltd Reguladores derivados de esteroides, método para prepararlos y usos de los mismos
US11634453B2 (en) 2018-10-12 2023-04-25 Sage Therapeutics, Inc. Neuroactive steroids substituted in position 10 with a cyclic group for use in the treatment of CNS disorders
TWI874337B (zh) 2018-12-05 2025-03-01 美商賽吉醫療公司 神經活性類固醇及其使用方法
EP3909967A4 (en) * 2019-01-08 2022-11-09 Chengdu Kanghong Pharmaceutical Co., Ltd. STEROID COMPOUND AND USE THEREOF AND METHOD OF MANUFACTURE THEREOF
CR20240234A (es) 2019-05-31 2024-07-09 Sage Therapeutics Inc ESTEROIDES NEUROACTIVOS Y COMPOSICIONES DE ESTOS (Divisional 2021-629)
CA3143545A1 (en) 2019-06-27 2020-12-30 Sage Therapeutics, Inc. Compounds for treating cns disorders
TWI896547B (zh) * 2019-06-27 2025-09-11 美商賽吉醫療公司 用於治療cns病症之組合物及方法
KR20220038681A (ko) * 2019-06-27 2022-03-29 세이지 테라퓨틱스, 인크. Cns 장애를 치료하기 위한 조성물 및 방법
US10857163B1 (en) 2019-09-30 2020-12-08 Athenen Therapeutics, Inc. Compositions that preferentially potentiate subtypes of GABAA receptors and methods of use thereof
WO2022246634A1 (en) * 2021-05-25 2022-12-01 Zhejiang Jiachi Development Pharmaceuticals Ltd. Compositions for treating insomnia and uses thereof
CN119306783A (zh) * 2023-07-14 2025-01-14 成都康弘药业集团股份有限公司 一种甾体类化合物的晶型及其用途
CN119529013B (zh) * 2024-11-25 2025-11-07 湖南新合新生物医药有限公司 一种祖拉诺龙中间体的合成方法

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WO1998005337A1 (en) * 1996-08-01 1998-02-12 Cocensys, Inc. Use of gaba and nmda receptor ligands for the treatment of migraine headache
WO2002026762A1 (en) 2000-09-29 2002-04-04 Regents Of The University Of Minnesota Triterpenes having antibacterial activity
AU2014256229B2 (en) * 2013-04-17 2018-10-04 Sage Therapeutics, Inc. 19-nor C3,3-disubstituted C21-N-pyrazolyl steroids and methods of use thereof
WO2016061527A1 (en) * 2014-10-16 2016-04-21 Sage Therapeutics, Inc. Compositions and methods for treating cns disorders
AR114044A1 (es) 2017-12-22 2020-07-15 Sage Therapeutics Inc Composiciones y métodos para el tratamiento de trastornos en el sistema nervioso central
EP3909967A4 (en) * 2019-01-08 2022-11-09 Chengdu Kanghong Pharmaceutical Co., Ltd. STEROID COMPOUND AND USE THEREOF AND METHOD OF MANUFACTURE THEREOF
KR20220038681A (ko) 2019-06-27 2022-03-29 세이지 테라퓨틱스, 인크. Cns 장애를 치료하기 위한 조성물 및 방법

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