JP2022507795A5 - - Google Patents
Info
- Publication number
- JP2022507795A5 JP2022507795A5 JP2021527866A JP2021527866A JP2022507795A5 JP 2022507795 A5 JP2022507795 A5 JP 2022507795A5 JP 2021527866 A JP2021527866 A JP 2021527866A JP 2021527866 A JP2021527866 A JP 2021527866A JP 2022507795 A5 JP2022507795 A5 JP 2022507795A5
- Authority
- JP
- Japan
- Prior art keywords
- optionally substituted
- group
- alkyl
- alkylene
- pharmaceutically acceptable
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862769413P | 2018-11-19 | 2018-11-19 | |
| US62/769,413 | 2018-11-19 | ||
| PCT/US2019/062045 WO2020106636A1 (en) | 2018-11-19 | 2019-11-18 | C11-cyclic substituted 13-membered macrolides and uses thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2022507795A JP2022507795A (ja) | 2022-01-18 |
| JP2022507795A5 true JP2022507795A5 (https=) | 2022-11-29 |
Family
ID=68965978
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021527866A Pending JP2022507795A (ja) | 2018-11-19 | 2019-11-18 | C10環状置換13員マクロライド及びそれらの使用 |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20220177508A1 (https=) |
| EP (1) | EP3883945A1 (https=) |
| JP (1) | JP2022507795A (https=) |
| KR (1) | KR20210123288A (https=) |
| CN (1) | CN113646319A (https=) |
| AU (2) | AU2019385383B2 (https=) |
| BR (1) | BR112021009607A2 (https=) |
| CA (1) | CA3120235A1 (https=) |
| IL (2) | IL310280A (https=) |
| MX (1) | MX2021005421A (https=) |
| SG (1) | SG11202105228SA (https=) |
| WO (1) | WO2020106636A1 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW202313065A (zh) * | 2021-05-28 | 2023-04-01 | 美商季卡尼醫療公司 | 用於治療遺傳疾病之化合物 |
| WO2023235380A1 (en) * | 2022-06-01 | 2023-12-07 | Zikani Therapeutics, Inc. | Macrolides for treating genetic diseases |
| WO2023250513A1 (en) * | 2022-06-24 | 2023-12-28 | Zikani Therapeutics, Inc. | 13-membered macrolide compounds for treating diseases mediated by abnormal protein translation |
| KR20250048331A (ko) * | 2022-08-11 | 2025-04-08 | 지카니 테라퓨틱스, 인크. | 치료용 아자케톨라이드 제조용 합성 공정 및 중간체 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA70972C2 (uk) * | 1998-11-20 | 2004-11-15 | Пфайзер Продактс Інк. | 13-членні азаліди і їх застосування як антибіотиків |
| BRPI0017013B1 (pt) * | 2000-01-27 | 2015-07-14 | Zoetis P Llc | Composição de antibiótico azalídeo e método para sua obtenção |
| WO2003014136A1 (en) * | 2001-08-08 | 2003-02-20 | Taisho Pharmaceutical Co., Ltd. | 11a-AZALIDE COMPOUNDS AND PROCESS FOR PRODUCING THE SAME |
| WO2004108744A2 (en) * | 2003-05-19 | 2004-12-16 | Prasad K Deshpande | Azalides and azaketolides having antimicrobial activity |
| US8097708B2 (en) * | 2006-02-07 | 2012-01-17 | Taisho Pharmaceutical Co., Ltd. | 10a-Azalide compound |
| US20130102551A1 (en) * | 2010-07-01 | 2013-04-25 | Andreas Hotte | Antibiotic compositions |
| JP6437523B2 (ja) * | 2013-04-04 | 2018-12-12 | プレジデント アンド フェローズ オブ ハーバード カレッジ | マクロライドならびにそれらの調製および使用の方法 |
| CN106998685A (zh) * | 2014-10-08 | 2017-08-01 | 哈佛大学的校长及成员们 | 14‑元酮内酯及其制备和使用方法 |
| EP3273969A4 (en) * | 2015-03-25 | 2018-11-21 | President and Fellows of Harvard College | Macrolides with modified desosamine sugars and uses thereof |
-
2019
- 2019-11-18 MX MX2021005421A patent/MX2021005421A/es unknown
- 2019-11-18 IL IL310280A patent/IL310280A/en unknown
- 2019-11-18 WO PCT/US2019/062045 patent/WO2020106636A1/en not_active Ceased
- 2019-11-18 AU AU2019385383A patent/AU2019385383B2/en active Active
- 2019-11-18 IL IL283185A patent/IL283185B2/en unknown
- 2019-11-18 US US17/294,918 patent/US20220177508A1/en not_active Abandoned
- 2019-11-18 SG SG11202105228SA patent/SG11202105228SA/en unknown
- 2019-11-18 BR BR112021009607-8A patent/BR112021009607A2/pt not_active IP Right Cessation
- 2019-11-18 JP JP2021527866A patent/JP2022507795A/ja active Pending
- 2019-11-18 KR KR1020217018877A patent/KR20210123288A/ko not_active Ceased
- 2019-11-18 CA CA3120235A patent/CA3120235A1/en active Pending
- 2019-11-18 CN CN201980087585.6A patent/CN113646319A/zh active Pending
- 2019-11-18 EP EP19824030.1A patent/EP3883945A1/en not_active Withdrawn
-
2023
- 2023-09-13 AU AU2023229518A patent/AU2023229518A1/en not_active Abandoned
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