JP2021530465A5 - - Google Patents

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Publication number
JP2021530465A5
JP2021530465A5 JP2020573467A JP2020573467A JP2021530465A5 JP 2021530465 A5 JP2021530465 A5 JP 2021530465A5 JP 2020573467 A JP2020573467 A JP 2020573467A JP 2020573467 A JP2020573467 A JP 2020573467A JP 2021530465 A5 JP2021530465 A5 JP 2021530465A5
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JP
Japan
Prior art keywords
optionally substituted
alkyl
clathrate
prodrug
solvate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020573467A
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English (en)
Japanese (ja)
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JP2021530465A (ja
JP7551087B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/039562 external-priority patent/WO2020006269A1/en
Publication of JP2021530465A publication Critical patent/JP2021530465A/ja
Publication of JP2021530465A5 publication Critical patent/JP2021530465A5/ja
Priority to JP2024076047A priority Critical patent/JP2024112835A/ja
Application granted granted Critical
Publication of JP7551087B2 publication Critical patent/JP7551087B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2020573467A 2018-06-27 2019-06-27 プロテアソーム活性増強化合物 Active JP7551087B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024076047A JP2024112835A (ja) 2018-06-27 2024-05-08 プロテアソーム活性増強化合物

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862690554P 2018-06-27 2018-06-27
US62/690,554 2018-06-27
PCT/US2019/039562 WO2020006269A1 (en) 2018-06-27 2019-06-27 Proteasome activity enhancing compounds

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024076047A Division JP2024112835A (ja) 2018-06-27 2024-05-08 プロテアソーム活性増強化合物

Publications (3)

Publication Number Publication Date
JP2021530465A JP2021530465A (ja) 2021-11-11
JP2021530465A5 true JP2021530465A5 (enExample) 2022-07-01
JP7551087B2 JP7551087B2 (ja) 2024-09-17

Family

ID=67297405

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2020573467A Active JP7551087B2 (ja) 2018-06-27 2019-06-27 プロテアソーム活性増強化合物
JP2024076047A Withdrawn JP2024112835A (ja) 2018-06-27 2024-05-08 プロテアソーム活性増強化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2024076047A Withdrawn JP2024112835A (ja) 2018-06-27 2024-05-08 プロテアソーム活性増強化合物

Country Status (5)

Country Link
US (2) US11746098B2 (enExample)
EP (1) EP3814336A1 (enExample)
JP (2) JP7551087B2 (enExample)
CN (1) CN112585130A (enExample)
WO (1) WO2020006269A1 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2020006269A1 (en) * 2018-06-27 2020-01-02 Proteostasis Therapeutics, Inc. Proteasome activity enhancing compounds
CN114699394B (zh) * 2022-05-24 2022-09-13 中山大学附属第一医院 用于肝癌放疗增敏的药物组合物及其应用

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