JP2021515006A5 - - Google Patents

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Publication number
JP2021515006A5
JP2021515006A5 JP2020545547A JP2020545547A JP2021515006A5 JP 2021515006 A5 JP2021515006 A5 JP 2021515006A5 JP 2020545547 A JP2020545547 A JP 2020545547A JP 2020545547 A JP2020545547 A JP 2020545547A JP 2021515006 A5 JP2021515006 A5 JP 2021515006A5
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Japan
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pharmaceutical composition
composition according
pharmaceutical
alkyl
present
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JP2020545547A
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English (en)
Japanese (ja)
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JP7336450B2 (ja
JP2021515006A (ja
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Priority claimed from PCT/EP2019/055138 external-priority patent/WO2019166626A1/en
Publication of JP2021515006A publication Critical patent/JP2021515006A/ja
Publication of JP2021515006A5 publication Critical patent/JP2021515006A5/ja
Priority to JP2023133951A priority Critical patent/JP2023156480A/ja
Application granted granted Critical
Publication of JP7336450B2 publication Critical patent/JP7336450B2/ja
Priority to JP2025097679A priority patent/JP2025134766A/ja
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JP2020545547A 2018-03-01 2019-03-01 (2s)-n-{(1s)-1-シアノ-2-[4-(3-メチル-2-オキソ-2,3-ジヒドロ-1,3-ベンゾオキサゾール-5-イル)フェニル]エチル}-1,4-オキサゼパン-2-カルボキサミドを含む医薬組成物 Active JP7336450B2 (ja)

Priority Applications (2)

Application Number Priority Date Filing Date Title
JP2023133951A JP2023156480A (ja) 2018-03-01 2023-08-21 (2s)-n-{(1s)-1-シアノ-2-[4-(3-メチル-2-オキソ-2,3-ジヒドロ-1,3-ベンゾオキサゾール-5-イル)フェニル]エチル}-1,4-オキサゼパン-2-カルボキサミドを含む医薬組成物
JP2025097679A JP2025134766A (ja) 2018-03-01 2025-06-11 (2s)-n-{(1s)-1-シアノ-2-[4-(3-メチル-2-オキソ-2,3-ジヒドロ-1,3-ベンゾオキサゾール-5-イル)フェニル]エチル}-1,4-オキサゼパン-2-カルボキサミドを含む医薬組成物

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862636944P 2018-03-01 2018-03-01
US62/636,944 2018-03-01
PCT/EP2019/055138 WO2019166626A1 (en) 2018-03-01 2019-03-01 PHARMACEUTICAL COMPOSITIONS COMPRISING (2S)-N-{(1S)-1-CYANO-2-[4-(3-METHYL-2-OXO-2,3-DIHYDRO-1,3-BENZOXAZOL-5-yl)PHENYL]ETHYL}-1,4-OXAZEPANE-2-CARBOXAMIDE

Related Child Applications (1)

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JP2023133951A Division JP2023156480A (ja) 2018-03-01 2023-08-21 (2s)-n-{(1s)-1-シアノ-2-[4-(3-メチル-2-オキソ-2,3-ジヒドロ-1,3-ベンゾオキサゾール-5-イル)フェニル]エチル}-1,4-オキサゼパン-2-カルボキサミドを含む医薬組成物

Publications (3)

Publication Number Publication Date
JP2021515006A JP2021515006A (ja) 2021-06-17
JP2021515006A5 true JP2021515006A5 (enExample) 2022-03-02
JP7336450B2 JP7336450B2 (ja) 2023-08-31

Family

ID=66102025

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2020545547A Active JP7336450B2 (ja) 2018-03-01 2019-03-01 (2s)-n-{(1s)-1-シアノ-2-[4-(3-メチル-2-オキソ-2,3-ジヒドロ-1,3-ベンゾオキサゾール-5-イル)フェニル]エチル}-1,4-オキサゼパン-2-カルボキサミドを含む医薬組成物
JP2023133951A Pending JP2023156480A (ja) 2018-03-01 2023-08-21 (2s)-n-{(1s)-1-シアノ-2-[4-(3-メチル-2-オキソ-2,3-ジヒドロ-1,3-ベンゾオキサゾール-5-イル)フェニル]エチル}-1,4-オキサゼパン-2-カルボキサミドを含む医薬組成物
JP2025097679A Pending JP2025134766A (ja) 2018-03-01 2025-06-11 (2s)-n-{(1s)-1-シアノ-2-[4-(3-メチル-2-オキソ-2,3-ジヒドロ-1,3-ベンゾオキサゾール-5-イル)フェニル]エチル}-1,4-オキサゼパン-2-カルボキサミドを含む医薬組成物

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2023133951A Pending JP2023156480A (ja) 2018-03-01 2023-08-21 (2s)-n-{(1s)-1-シアノ-2-[4-(3-メチル-2-オキソ-2,3-ジヒドロ-1,3-ベンゾオキサゾール-5-イル)フェニル]エチル}-1,4-オキサゼパン-2-カルボキサミドを含む医薬組成物
JP2025097679A Pending JP2025134766A (ja) 2018-03-01 2025-06-11 (2s)-n-{(1s)-1-シアノ-2-[4-(3-メチル-2-オキソ-2,3-ジヒドロ-1,3-ベンゾオキサゾール-5-イル)フェニル]エチル}-1,4-オキサゼパン-2-カルボキサミドを含む医薬組成物

Country Status (21)

Country Link
US (3) US12059424B2 (enExample)
EP (2) EP4516353A3 (enExample)
JP (3) JP7336450B2 (enExample)
KR (2) KR20250002710A (enExample)
CN (3) CN112055593B (enExample)
AU (3) AU2019228717C1 (enExample)
CA (1) CA3091707A1 (enExample)
DK (1) DK3758708T3 (enExample)
ES (1) ES3011730T3 (enExample)
FI (1) FI3758708T3 (enExample)
HR (1) HRP20250115T1 (enExample)
HU (1) HUE070049T2 (enExample)
LT (1) LT3758708T (enExample)
MA (1) MA52424B1 (enExample)
MD (1) MD3758708T2 (enExample)
PL (1) PL3758708T3 (enExample)
PT (1) PT3758708T (enExample)
RS (1) RS66494B1 (enExample)
SI (1) SI3758708T1 (enExample)
SM (1) SMT202500062T1 (enExample)
WO (1) WO2019166626A1 (enExample)

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HUE070049T2 (hu) 2018-03-01 2025-05-28 Astrazeneca Ab (2S)-{(1S)-1-ciano-2-[4-(3-metil-2-oxo-2,3-dihidro-1,3-benzoxazol-5-il)fenil]etil} -1,4-oxazepán-2-karboxamidot tartalmazó gyógyászati készítmények
WO2020018547A1 (en) 2018-07-17 2020-01-23 Insmed Incorporated Certain (2s)-n-[(1s)-1-cyano-2-phenylethyl]-1,4-oxazepane-2-carboxamides for treating lupus nephritis
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CN115925696A (zh) * 2021-10-29 2023-04-07 瑞石生物医药有限公司 一种1-氰基-2-苯基乙基甲酰胺衍生物及其用途
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JP2026503035A (ja) 2023-01-06 2026-01-27 インスメッド インコーポレイテッド 新規な可逆性dpp1阻害剤及びその用途
JP2026510407A (ja) * 2023-03-23 2026-04-02 ハイスコ ファーマスーティカル プライベート リミテッド ジペプチジルペプチダーゼ小分子阻害剤を含む医薬組成物

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WO2020018547A1 (en) 2018-07-17 2020-01-23 Insmed Incorporated Certain (2s)-n-[(1s)-1-cyano-2-phenylethyl]-1,4-oxazepane-2-carboxamides for treating lupus nephritis
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