JP2021501205A5 - - Google Patents
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- JP2021501205A5 JP2021501205A5 JP2020543266A JP2020543266A JP2021501205A5 JP 2021501205 A5 JP2021501205 A5 JP 2021501205A5 JP 2020543266 A JP2020543266 A JP 2020543266A JP 2020543266 A JP2020543266 A JP 2020543266A JP 2021501205 A5 JP2021501205 A5 JP 2021501205A5
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- JP
- Japan
- Prior art keywords
- optionally substituted
- formula
- compound
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- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 0 C*C(NC(CCC(CC(O*)=O)O*)S1OC(C)(C(C2)C(C)(C)C2C2)C2O1)=O Chemical compound C*C(NC(CCC(CC(O*)=O)O*)S1OC(C)(C(C2)C(C)(C)C2C2)C2O1)=O 0.000 description 2
- IFTRQJLVEBNKJK-UHFFFAOYSA-N CCC1CCCC1 Chemical compound CCC1CCCC1 IFTRQJLVEBNKJK-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762580343P | 2017-11-01 | 2017-11-01 | |
| US62/580,343 | 2017-11-01 | ||
| PCT/US2018/058143 WO2019089542A1 (en) | 2017-11-01 | 2018-10-30 | Synthesis of boronate ester derivatives and uses thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021501205A JP2021501205A (ja) | 2021-01-14 |
| JP2021501205A5 true JP2021501205A5 (https=) | 2021-12-09 |
| JP7480050B2 JP7480050B2 (ja) | 2024-05-09 |
Family
ID=66245250
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020543266A Active JP7480050B2 (ja) | 2017-11-01 | 2018-10-30 | ボロン酸エステル誘導体の合成およびその使用 |
Country Status (14)
| Country | Link |
|---|---|
| US (3) | US11999757B2 (https=) |
| EP (1) | EP3704130A4 (https=) |
| JP (1) | JP7480050B2 (https=) |
| KR (1) | KR20200076730A (https=) |
| CN (2) | CN111556872B (https=) |
| AU (1) | AU2018360502B2 (https=) |
| CA (1) | CA3080763A1 (https=) |
| CL (1) | CL2020001143A1 (https=) |
| CO (1) | CO2020006299A2 (https=) |
| JO (2) | JOP20200101B1 (https=) |
| MX (2) | MX2020004425A (https=) |
| PH (1) | PH12020550544A1 (https=) |
| SG (1) | SG11202003762VA (https=) |
| WO (1) | WO2019089542A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN111556872B (zh) | 2017-11-01 | 2024-05-10 | 梅琳塔治疗公司 | 硼酸酯衍生物的合成及其用途 |
| CN116789689B (zh) * | 2023-06-21 | 2026-03-20 | 清华大学 | 硼代萘系化合物及其制备方法和应用 |
Family Cites Families (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4783443A (en) | 1986-03-03 | 1988-11-08 | The University Of Chicago | Amino acyl cephalosporin derivatives |
| JP2852545B2 (ja) | 1989-11-14 | 1999-02-03 | チッソ株式会社 | 複数の不斉点を持つ光学活性化合物および製造法 |
| CA2165996C (en) | 1995-12-22 | 2002-01-29 | Murray Douglas Bailey | Stereoselective preparation of 2-substituted succinic derivatives |
| FR2745288B1 (fr) | 1996-02-27 | 1998-04-17 | Adir | Nouveaux derives de l'acide boronique, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| DE19917979A1 (de) | 1999-04-21 | 2000-10-26 | Clariant Gmbh | Verfahren zur Herstellung von substituierten Phenyl-boronsäuren |
| AU5104300A (en) | 1999-06-04 | 2000-12-28 | Kaneka Corporation | Processes for the preparation of 5-hydroxy-3-oxopentanoic acid derivatives |
| DE10032017A1 (de) | 2000-07-01 | 2002-01-10 | Clariant Gmbh | Verfahren zur Herstellung hochreiner Formylphenylboronsäuren |
| DE10112401A1 (de) * | 2001-03-13 | 2002-09-19 | Degussa | Alkohol-Dehydrogenase und deren Verwendung |
| DE10119274A1 (de) * | 2001-04-20 | 2002-10-31 | Juelich Enzyme Products Gmbh | Enzymatisches Verfahren zur enantioselektiven Reduktion von Ketoverbindungen |
| JP4824874B2 (ja) * | 2001-07-19 | 2011-11-30 | 高砂香料工業株式会社 | 光学活性γ−ブチロラクトンの製造方法 |
| ES2544579T3 (es) * | 2002-07-30 | 2015-09-01 | Takasago International Corporation | Procedimiento de producción de un beta-aminoácido ópticamente activo |
| TWI372725B (en) | 2004-01-30 | 2012-09-21 | Semequip Inc | Methods of synthesis of isotopically enriched borohydride and methods of synthesis of isotopically enriched boranes |
| DE102004022397A1 (de) * | 2004-05-06 | 2005-12-01 | Consortium für elektrochemische Industrie GmbH | Chirale C2-symmetrische Biphenyle, deren Herstellung sowie Metallkomplexe enthaltend diese Liganden und deren Verwendung als Katalysatoren in chirogenen Synthesen |
| WO2007034909A1 (ja) * | 2005-09-22 | 2007-03-29 | Kaneka Corporation | （３ｒ，５ｒ）－７－アミノ－３，５－ジヒドロキシヘプタン酸誘導体の製造法 |
| GB2474687A (en) | 2009-10-23 | 2011-04-27 | Phoenix Chemicals Ltd | A continuous process for the production of (R)-6-cyano-5-hydroxy-3-oxo-hexanoic acid tert-butyl ester (and derivatives) |
| CA2807546C (en) | 2010-08-10 | 2022-08-23 | Rempex Pharmaceuticals, Inc. | Cyclic boronic acid ester derivatives and therapeutic uses thereof |
| WO2013056163A1 (en) | 2011-10-14 | 2013-04-18 | The Regents Of The University Of California | Beta-lactamase inhibitors |
| EP2814483A2 (en) * | 2012-02-15 | 2014-12-24 | Rempex Pharmaceuticals, Inc. | Methods of treating bacterial infections |
| CN104395326B (zh) | 2012-08-20 | 2017-04-05 | 玛耐科股份有限公司 | 二取代硼酸衍生物的制造方法和新型二取代硼酸衍生物 |
| CN102965403A (zh) | 2012-11-19 | 2013-03-13 | 苏州汉酶生物技术有限公司 | (3r,5s)-6-氯-3,5-二羟基己酸叔丁酯的生物制备方法 |
| AU2013355110B2 (en) * | 2012-12-07 | 2017-11-09 | VenatoRx Pharmaceuticals, Inc. | Beta-lactamase inhibitors |
| PT3369724T (pt) | 2013-11-05 | 2021-02-10 | Bracco Imaging Spa | Processo para a preparação de iopamidol |
| ES2750805T3 (es) * | 2014-05-05 | 2020-03-27 | Rempex Pharmaceuticals Inc | Síntesis de sales de boronato y usos de las mismas |
| CN111556872B (zh) | 2017-11-01 | 2024-05-10 | 梅琳塔治疗公司 | 硼酸酯衍生物的合成及其用途 |
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2018
- 2018-10-30 CN CN201880079247.3A patent/CN111556872B/zh active Active
- 2018-10-30 CA CA3080763A patent/CA3080763A1/en active Pending
- 2018-10-30 AU AU2018360502A patent/AU2018360502B2/en active Active
- 2018-10-30 WO PCT/US2018/058143 patent/WO2019089542A1/en not_active Ceased
- 2018-10-30 US US16/760,369 patent/US11999757B2/en active Active
- 2018-10-30 MX MX2020004425A patent/MX2020004425A/es unknown
- 2018-10-30 EP EP18874877.6A patent/EP3704130A4/en active Pending
- 2018-10-30 CN CN202410485244.7A patent/CN118388347A/zh active Pending
- 2018-10-30 KR KR1020207015638A patent/KR20200076730A/ko not_active Ceased
- 2018-10-30 SG SG11202003762VA patent/SG11202003762VA/en unknown
- 2018-10-30 JP JP2020543266A patent/JP7480050B2/ja active Active
- 2018-10-31 US US16/176,302 patent/US20190127396A1/en not_active Abandoned
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2020
- 2020-04-30 CL CL2020001143A patent/CL2020001143A1/es unknown
- 2020-05-01 PH PH12020550544A patent/PH12020550544A1/en unknown
- 2020-05-06 JO JOJO/P/2020/0101A patent/JOP20200101B1/ar active
- 2020-05-26 CO CONC2020/0006299A patent/CO2020006299A2/es unknown
- 2020-07-13 MX MX2023000529A patent/MX2023000529A/es unknown
-
2024
- 2024-04-04 US US18/627,105 patent/US20240279248A1/en active Pending
- 2024-10-20 JO JOJO/P/2024/0234A patent/JOP20240234A1/ar unknown