JP2005538088A5 - - Google Patents
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- Publication number
- JP2005538088A5 JP2005538088A5 JP2004522603A JP2004522603A JP2005538088A5 JP 2005538088 A5 JP2005538088 A5 JP 2005538088A5 JP 2004522603 A JP2004522603 A JP 2004522603A JP 2004522603 A JP2004522603 A JP 2004522603A JP 2005538088 A5 JP2005538088 A5 JP 2005538088A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- defined above
- compound
- symbols
- prepared
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 description 10
- 238000000034 method Methods 0.000 description 6
- 125000005843 halogen group Chemical group 0.000 description 3
- 238000004519 manufacturing process Methods 0.000 description 3
- OAKJQQAXSVQMHS-UHFFFAOYSA-N Hydrazine Chemical compound NN OAKJQQAXSVQMHS-UHFFFAOYSA-N 0.000 description 2
- 0 CC(c1ccccc1)=* Chemical compound CC(c1ccccc1)=* 0.000 description 1
- 150000001540 azides Chemical class 0.000 description 1
- 150000002429 hydrazines Chemical class 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN548MA2002 | 2002-07-22 | ||
| IN548/MAS/2002 | 2002-07-22 | ||
| PCT/IB2003/002879 WO2004009560A1 (en) | 2002-07-22 | 2003-07-21 | Novel bio-active molecules |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005538088A JP2005538088A (ja) | 2005-12-15 |
| JP2005538088A5 true JP2005538088A5 (https=) | 2010-07-15 |
| JP4860151B2 JP4860151B2 (ja) | 2012-01-25 |
Family
ID=37775275
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004522603A Expired - Fee Related JP4860151B2 (ja) | 2002-07-22 | 2003-07-21 | 新規な生物活性分子 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US7317014B2 (https=) |
| EP (1) | EP1542978B1 (https=) |
| JP (1) | JP4860151B2 (https=) |
| AT (1) | ATE505462T1 (https=) |
| AU (1) | AU2003249484A1 (https=) |
| CA (1) | CA2492342C (https=) |
| DE (1) | DE60336735D1 (https=) |
| ES (1) | ES2365011T3 (https=) |
| WO (1) | WO2004009560A1 (https=) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2006510597A (ja) * | 2002-09-27 | 2006-03-30 | メルク エンド カムパニー インコーポレーテッド | 置換ピリミジン類 |
| TW200637556A (en) * | 2005-01-31 | 2006-11-01 | Basf Ag | Substituted 5-phenyl pyrimidines I in therapy |
| ES2600460T3 (es) | 2005-05-10 | 2017-02-09 | Intermune, Inc. | Derivados de piridona-2-ona como moduladores del sistema de proteína cinasa activada por estrés |
| US7452892B2 (en) | 2005-06-17 | 2008-11-18 | Bristol-Myers Squibb Company | Triazolopyrimidine cannabinoid receptor 1 antagonists |
| US8372851B2 (en) | 2005-10-21 | 2013-02-12 | Exelixis, Inc. | Pyrazolo pyrimidines as casein kinase II (CK2) modulators |
| PL1973884T3 (pl) * | 2006-01-19 | 2017-05-31 | Orchid Pharma Limited | Nowe związki heterocykliczne |
| US7863446B2 (en) * | 2006-01-19 | 2011-01-04 | Orchid Research Laboratories Limited | Heterocycles |
| DE102006054205A1 (de) * | 2006-11-15 | 2008-05-29 | Rheinische Friedrich-Wilhelms Universität | Verwendung von Cytohesin-Inhibitoren zur chemischen Induktion von Langlebigkeit |
| BRPI0912029A2 (pt) * | 2008-02-01 | 2020-06-30 | Orchid Research Laboratories Limited | novos heterociclos |
| WO2009128395A1 (ja) * | 2008-04-16 | 2009-10-22 | 株式会社林原生物化学研究所 | ２－アミノフェノール又はその誘導体を有効成分とする骨形成促進剤 |
| CN102099036B (zh) | 2008-06-03 | 2015-05-27 | 英特芒尼公司 | 用于治疗炎性疾患和纤维化疾患的化合物和方法 |
| WO2011038204A1 (en) | 2009-09-25 | 2011-03-31 | N30 Pharmaceuticals, Llc | Novel dihydropyrimidin-2(1h)-one compounds as s-nitrosoglutathione reductase inhibitors |
| US8906933B2 (en) | 2010-09-24 | 2014-12-09 | N30 Pharmaceuticals, Inc. | Dihydropyrimidin-2(1H)-one compounds as neurokinin-3 receptor antagonists |
| CZ305457B6 (cs) * | 2011-02-28 | 2015-09-30 | Ústav organické chemie a biochemie, Akademie věd ČR v. v. i. | Pyrimidinové sloučeniny inhibující tvorbu oxidu dusnatého a prostaglandinu E2, způsob výroby a použití |
| AR092742A1 (es) | 2012-10-02 | 2015-04-29 | Intermune Inc | Piridinonas antifibroticas |
| MX382781B (es) | 2014-04-02 | 2025-03-13 | Intermune Inc | Piridinonas anti-fibroticas. |
| WO2019055832A1 (en) * | 2017-09-15 | 2019-03-21 | The Regents Of The University Of California | COMPOSITIONS AND METHODS FOR INHIBITING N-SMASE2 |
| TW202321229A (zh) | 2021-08-18 | 2023-06-01 | 美商富曼西公司 | 殺真菌的取代的雜環化合物 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2602794A (en) * | 1952-07-08 | Process for preparation of x-amino-s | ||
| BE759176A (fr) * | 1969-11-20 | 1971-05-19 | Sandoz Sa | Derives de la pyrimidine, leur preparation et medicaments contenant cesderives |
| DE2142317A1 (de) | 1971-08-24 | 1973-03-01 | Bayer Ag | Hypnotisches mittel |
| US4438117A (en) * | 1980-09-03 | 1984-03-20 | E. I. Du Pont De Nemours And Company | 2-Substituted thio-4,5-diarylpyrimidines |
| US4500533A (en) * | 1983-06-22 | 1985-02-19 | Eli Lilly And Company | 2,4,5-Triaryl pyrimidines and a method of treating pain, fever, thrombosis, inflammation and arthritis |
| DE3605002A1 (de) * | 1986-02-18 | 1987-08-20 | Bayer Ag | Phosphorsaeureester |
| GB8909560D0 (en) * | 1989-04-26 | 1989-06-14 | Smith Kline French Lab | Chemical compounds |
| WO1992002513A1 (en) | 1990-08-06 | 1992-02-20 | Fujisawa Pharmaceutical Co., Ltd. | Heterocyclic compounds |
| US5486534A (en) * | 1994-07-21 | 1996-01-23 | G. D. Searle & Co. | 3,4-substituted pyrazoles for the treatment of inflammation |
| US6096753A (en) * | 1996-12-05 | 2000-08-01 | Amgen Inc. | Substituted pyrimidinone and pyridone compounds and methods of use |
| US6410729B1 (en) * | 1996-12-05 | 2002-06-25 | Amgen Inc. | Substituted pyrimidine compounds and methods of use |
| WO2001062233A2 (en) * | 2000-02-25 | 2001-08-30 | F. Hoffmann La Roche Ag | Adenosine receptor modulators |
| JP4359146B2 (ja) * | 2002-02-13 | 2009-11-04 | エフ．ホフマン−ラ ロシュ アーゲー | 新規なピリジン−およびピリミジン−誘導体 |
| AU2003216585A1 (en) * | 2002-04-10 | 2003-10-20 | Orchid Chemicals And Pharmaceuticals Limited | Pyrimidinedione derivatives useful for the treatment of inflammation and immunological diseases |
-
2003
- 2003-07-21 JP JP2004522603A patent/JP4860151B2/ja not_active Expired - Fee Related
- 2003-07-21 AT AT03765232T patent/ATE505462T1/de active
- 2003-07-21 CA CA2492342A patent/CA2492342C/en not_active Expired - Fee Related
- 2003-07-21 EP EP03765232A patent/EP1542978B1/en not_active Expired - Lifetime
- 2003-07-21 AU AU2003249484A patent/AU2003249484A1/en not_active Abandoned
- 2003-07-21 US US10/469,647 patent/US7317014B2/en not_active Expired - Fee Related
- 2003-07-21 WO PCT/IB2003/002879 patent/WO2004009560A1/en not_active Ceased
- 2003-07-21 ES ES03765232T patent/ES2365011T3/es not_active Expired - Lifetime
- 2003-07-21 DE DE60336735T patent/DE60336735D1/de not_active Expired - Lifetime
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