JP2021098728A5 - - Google Patents
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- JP2021098728A5 JP2021098728A5 JP2021037000A JP2021037000A JP2021098728A5 JP 2021098728 A5 JP2021098728 A5 JP 2021098728A5 JP 2021037000 A JP2021037000 A JP 2021037000A JP 2021037000 A JP2021037000 A JP 2021037000A JP 2021098728 A5 JP2021098728 A5 JP 2021098728A5
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- Prior art keywords
- pharmaceutical composition
- pharmaceutically acceptable
- acceptable salt
- orally administered
- acceptable excipient
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- 239000008194 pharmaceutical composition Substances 0.000 claims 10
- 239000000546 pharmaceutical excipient Substances 0.000 claims 3
- 150000003839 salts Chemical class 0.000 claims 3
- 206010028980 Neoplasm Diseases 0.000 claims 2
- 201000011510 cancer Diseases 0.000 claims 2
- 239000002246 antineoplastic agent Substances 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 claims 1
- 229940127089 cytotoxic agent Drugs 0.000 claims 1
- 239000003814 drug Substances 0.000 claims 1
- 208000002154 non-small cell lung carcinoma Diseases 0.000 claims 1
- 229940124597 therapeutic agent Drugs 0.000 claims 1
- 230000001225 therapeutic effect Effects 0.000 claims 1
- 208000029729 tumor suppressor gene on chromosome 11 Diseases 0.000 claims 1
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2023032872A JP2023060145A (ja) | 2018-05-14 | 2023-03-03 | Ｍｃｌ－１阻害剤 |
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862671306P | 2018-05-14 | 2018-05-14 | |
| US62/671,306 | 2018-05-14 | ||
| US201862749918P | 2018-10-24 | 2018-10-24 | |
| US62/749,918 | 2018-10-24 | ||
| JP2020564228A JP6899975B2 (ja) | 2018-05-14 | 2019-05-13 | Ｍｃｌ−１阻害剤 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020564228A Division JP6899975B2 (ja) | 2018-05-14 | 2019-05-13 | Ｍｃｌ−１阻害剤 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023032872A Division JP2023060145A (ja) | 2018-05-14 | 2023-03-03 | Ｍｃｌ－１阻害剤 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021098728A JP2021098728A (ja) | 2021-07-01 |
| JP2021098728A5 true JP2021098728A5 (US20070167479A1-20070719-C00034.png) | 2022-10-12 |
| JP7240431B2 JP7240431B2 (ja) | 2023-03-15 |
Family
ID=66770559
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020564228A Active JP6899975B2 (ja) | 2018-05-14 | 2019-05-13 | Ｍｃｌ−１阻害剤 |
| JP2021037000A Active JP7240431B2 (ja) | 2018-05-14 | 2021-03-09 | Ｍｃｌ－１阻害剤 |
| JP2023032872A Pending JP2023060145A (ja) | 2018-05-14 | 2023-03-03 | Ｍｃｌ－１阻害剤 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020564228A Active JP6899975B2 (ja) | 2018-05-14 | 2019-05-13 | Ｍｃｌ−１阻害剤 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023032872A Pending JP2023060145A (ja) | 2018-05-14 | 2023-03-03 | Ｍｃｌ－１阻害剤 |
Country Status (29)
Families Citing this family (25)
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| CN118178645A (zh) | 2019-10-18 | 2024-06-14 | 四十七公司 | 用于治疗骨髓增生异常综合征和急性髓系白血病的联合疗法 |
| JP2022552748A (ja) | 2019-10-31 | 2022-12-19 | フォーティ セブン， インコーポレイテッド | 抗ｃｄ４７及び抗ｃｄ２０による血液癌の治療 |
| TWI778443B (zh) * | 2019-11-12 | 2022-09-21 | 美商基利科學股份有限公司 | Mcl1抑制劑 |
| CN114787139A (zh) * | 2019-11-26 | 2022-07-22 | 吉利德科学公司 | 用于制备mcl1抑制剂的方法和中间体 |
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| KR20230107848A (ko) * | 2020-11-19 | 2023-07-18 | 길리애드 사이언시즈, 인코포레이티드 | 거대고리형 mcl1 저해제를 제조하기 위한 방법 및 중간체 |
| AU2021404501A1 (en) | 2020-12-17 | 2023-08-03 | Janssen Pharmaceutica Nv | Macrocyclic branched 3-fluoro-but-3-enamides as inhibitors of mcl-1 |
| TW202302145A (zh) | 2021-04-14 | 2023-01-16 | 美商基利科學股份有限公司 | ＣＤ４７／ＳＩＲＰα結合及ＮＥＤＤ８活化酶Ｅ１調節次單元之共抑制以用於治療癌症 |
| CN117295749A (zh) | 2021-04-26 | 2023-12-26 | 詹森药业有限公司 | 作为mcl-1抑制剂的大环2-烯丙基四氢呋喃 |
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2019
- 2019-05-13 CR CR20200544A patent/CR20200544A/es unknown
- 2019-05-13 CN CN201980032695.2A patent/CN112118845B/zh active Active
- 2019-05-13 LT LTEPPCT/US2019/032053T patent/LT3793565T/lt unknown
- 2019-05-13 CN CN202310897123.9A patent/CN117304130A/zh active Pending
- 2019-05-13 JP JP2020564228A patent/JP6899975B2/ja active Active
- 2019-05-13 US US16/410,457 patent/US10703733B2/en active Active
- 2019-05-13 AU AU2019269391A patent/AU2019269391B2/en active Active
- 2019-05-13 UA UAA202006695A patent/UA125163C2/uk unknown
- 2019-05-13 PT PT197287931T patent/PT3793565T/pt unknown
- 2019-05-13 BR BR112020021648-8A patent/BR112020021648A2/pt unknown
- 2019-05-13 PL PL19728793T patent/PL3793565T3/pl unknown
- 2019-05-13 IL IL291430A patent/IL291430B2/en unknown
- 2019-05-13 KR KR1020207035485A patent/KR102551319B1/ko active IP Right Grant
- 2019-05-13 PE PE2020001829A patent/PE20210004A1/es unknown
- 2019-05-13 EP EP19728793.1A patent/EP3793565B1/en active Active
- 2019-05-13 KR KR1020247015778A patent/KR20240074001A/ko active Search and Examination
- 2019-05-13 ES ES19728793T patent/ES2907923T3/es active Active
- 2019-05-13 EP EP21218221.6A patent/EP4029868A1/en active Pending
- 2019-05-13 SG SG11202010964VA patent/SG11202010964VA/en unknown
- 2019-05-13 HR HRP20220215TT patent/HRP20220215T1/hr unknown
- 2019-05-13 KR KR1020237022152A patent/KR102666717B1/ko active IP Right Grant
- 2019-05-13 CA CA3099152A patent/CA3099152C/en active Active
- 2019-05-13 DK DK19728793.1T patent/DK3793565T3/da active
- 2019-05-13 SI SI201930181T patent/SI3793565T1/sl unknown
- 2019-05-13 MX MX2020012137A patent/MX2020012137A/es unknown
- 2019-05-13 HU HUE19728793A patent/HUE057852T2/hu unknown
- 2019-05-13 WO PCT/US2019/032053 patent/WO2019222112A1/en unknown
- 2019-05-14 TW TW108116508A patent/TWI719478B/zh active
- 2019-05-14 TW TW110107128A patent/TWI813957B/zh active
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2020
- 2020-04-23 US US16/857,021 patent/US10988451B2/en active Active
- 2020-10-27 IL IL278336A patent/IL278336B/en unknown
- 2020-11-03 PH PH12020551881A patent/PH12020551881A1/en unknown
- 2020-11-10 CO CONC2020/0014009A patent/CO2020014009A2/es unknown
- 2020-11-10 CL CL2020002919A patent/CL2020002919A1/es unknown
- 2020-11-10 ZA ZA2020/07007A patent/ZA202007007B/en unknown
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2021
- 2021-02-09 US US17/171,201 patent/US11643400B2/en active Active
- 2021-03-09 JP JP2021037000A patent/JP7240431B2/ja active Active
- 2021-05-25 AU AU2021203373A patent/AU2021203373B2/en active Active
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2022
- 2022-03-16 CY CY20221100208T patent/CY1125065T1/el unknown
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2023
- 2023-03-03 JP JP2023032872A patent/JP2023060145A/ja active Pending
- 2023-03-09 US US18/181,336 patent/US20230312490A1/en active Pending
- 2023-11-24 AU AU2023270332A patent/AU2023270332A1/en active Pending
