JP2020518555A5 - - Google Patents
Info
- Publication number
- JP2020518555A5 JP2020518555A5 JP2019552993A JP2019552993A JP2020518555A5 JP 2020518555 A5 JP2020518555 A5 JP 2020518555A5 JP 2019552993 A JP2019552993 A JP 2019552993A JP 2019552993 A JP2019552993 A JP 2019552993A JP 2020518555 A5 JP2020518555 A5 JP 2020518555A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- oxadiazole
- dihydro
- fluorophenyl
- chloro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP17169277.5 | 2017-05-03 | ||
| EP17169277.5A EP3398941A1 (en) | 2017-05-03 | 2017-05-03 | Heterocyclic p2x7 antagonists |
| PCT/EP2018/061180 WO2018202694A1 (en) | 2017-05-03 | 2018-05-02 | Heterocyclic p2x7 antagonists |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2020518555A JP2020518555A (ja) | 2020-06-25 |
| JP2020518555A5 true JP2020518555A5 (enExample) | 2022-10-06 |
| JP7227916B2 JP7227916B2 (ja) | 2023-02-22 |
Family
ID=58668805
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019552993A Active JP7227916B2 (ja) | 2017-05-03 | 2018-05-02 | 複素環ｐ２ｘ７アンタゴニスト |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US11623919B2 (enExample) |
| EP (2) | EP3398941A1 (enExample) |
| JP (1) | JP7227916B2 (enExample) |
| CN (1) | CN110770214B (enExample) |
| CA (1) | CA3059525A1 (enExample) |
| DK (1) | DK3619200T3 (enExample) |
| ES (1) | ES2911049T3 (enExample) |
| IL (1) | IL270275B2 (enExample) |
| RU (1) | RU2768865C2 (enExample) |
| WO (1) | WO2018202694A1 (enExample) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN116782901A (zh) | 2020-11-30 | 2023-09-19 | 旭化成制药株式会社 | 用于使神经病理性疼痛缓和的药物 |
| US20240368092A1 (en) | 2021-09-03 | 2024-11-07 | Breye Therapeutics Aps | 2,4-Dihydro-3H-1,2,4-Triazol-3-One P2X7 Antagonists |
| WO2025057074A1 (en) | 2023-09-13 | 2025-03-20 | Suven Life Sciences Limited | N-aryl benzamide derivatives as p2x7 receptor antagonists |
| WO2026041663A1 (en) | 2024-08-22 | 2026-02-26 | Breye Therapeutics Aps | P2x7 receptor antagonists |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1529621A (fr) * | 1967-01-17 | 1968-06-21 | Dausse Lab | Nouvelles oxadiazolinones basiques et leur procédé de préparation |
| FR1529700A (fr) * | 1967-04-11 | 1968-06-21 | Dausse Sa Lab | Tertioaminoalcoyl oxadiazolinones et leur procédé de préparation |
| FR1575552A (enExample) * | 1967-12-07 | 1969-07-25 | ||
| GB1508210A (en) | 1975-12-22 | 1978-04-19 | Labaz | Benzofuran-derived amidoximes and process for preparing the same |
| JPS61106575A (ja) * | 1984-10-31 | 1986-05-24 | Nippon Soda Co Ltd | １，２，４−チアジアゾ−ル−５−オン誘導体及び製造方法 |
| US5066662A (en) * | 1990-05-21 | 1991-11-19 | Warner-Lambert Company | Substituted oxazolidin-2-ones and 1,2,4-oxadiazolin-5-ones and derivatives thereof acting at muscarinic receptors |
| ATE295832T1 (de) | 2000-03-24 | 2005-06-15 | Pharmacia Corp | Amidino-verbindung sowie salze davon verwendbar als hemmstoffe der stickstoffmonoxid-synthase |
| AR034120A1 (es) | 2000-04-13 | 2004-02-04 | Pharmacia Corp | Compuesto derivado halogenado del acido 2-amino-4,5 heptenoico, composicion farmaceutica que lo comprende y el uso de dicho compuesto y dicha composicion en la fabricacion de un medicamento para inhibir o modular la sintesis de acido nitrico |
| TWI290130B (en) | 2000-09-15 | 2007-11-21 | Pharmacia Corp | 2-Amino-2alkyl-5 heptenoic and heptynoic acid derivatives useful as nitric oxide synthase inhibitors |
| AR031129A1 (es) | 2000-09-15 | 2003-09-10 | Pharmacia Corp | Derivados de los acidos 2-amino-2-alquil-4-hexenoico y -hexinoico utiles como inhibidores de oxido nitrico sintetasa |
| ES2281801T3 (es) | 2003-05-12 | 2007-10-01 | Pfizer Products Inc. | Inhibidores benzamida del receptor p2x7. |
| GB0312609D0 (en) | 2003-06-02 | 2003-07-09 | Astrazeneca Ab | Novel compounds |
| EP2215086B1 (en) * | 2007-11-20 | 2011-08-24 | Sumitomo Chemical Company, Limited | Pyridine compound, pesticidal composition and method of controlling pest |
| KR100967889B1 (ko) * | 2008-02-01 | 2010-07-06 | 한국화학연구원 | 2-이미노벤조이미다졸 유도체를 포함하는 살균제 조성물 |
| WO2009108551A2 (en) | 2008-02-25 | 2009-09-03 | H. Lundbeck A/S | Heteroaryl amide analogues |
| KR101598397B1 (ko) | 2008-04-22 | 2016-02-29 | 얀센 파마슈티카 엔.브이. | 퀴놀린 또는 이소퀴놀린 치환된 피2엑스7 안타고니스트 |
| PL213249B1 (pl) * | 2009-12-08 | 2013-02-28 | Univ Medyczny W Lublinie | Zastosowanie pochodnych semikarbazydowych oraz 1,2,4-triazolino-5-onu posiadających układ 1-metylopirolu |
| JP2012041325A (ja) * | 2010-08-23 | 2012-03-01 | Bayer Cropscience Ag | オキサジアゾリノン誘導体およびその有害生物の防除用途 |
| US9988373B2 (en) | 2013-12-26 | 2018-06-05 | Shionogi & Co., Ltd. | Nitrogen-containing six-membered cyclic derivatives and pharmaceutical composition comprising the same |
| JP6285736B2 (ja) | 2014-02-04 | 2018-02-28 | 株式会社ソニー・インタラクティブエンタテインメント | 情報処理装置および入力デバイスの割当方法 |
-
2017
- 2017-05-03 EP EP17169277.5A patent/EP3398941A1/en not_active Withdrawn
-
2018
- 2018-05-02 JP JP2019552993A patent/JP7227916B2/ja active Active
- 2018-05-02 WO PCT/EP2018/061180 patent/WO2018202694A1/en not_active Ceased
- 2018-05-02 ES ES18724792T patent/ES2911049T3/es active Active
- 2018-05-02 RU RU2019134453A patent/RU2768865C2/ru active
- 2018-05-02 CA CA3059525A patent/CA3059525A1/en active Pending
- 2018-05-02 US US16/607,737 patent/US11623919B2/en active Active
- 2018-05-02 EP EP18724792.9A patent/EP3619200B1/en active Active
- 2018-05-02 DK DK18724792.9T patent/DK3619200T3/da active
- 2018-05-02 CN CN201880027662.4A patent/CN110770214B/zh active Active
-
2019
- 2019-10-29 IL IL270275A patent/IL270275B2/en unknown
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