JP2020073474A5 - - Google Patents

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Publication number
JP2020073474A5
JP2020073474A5 JP2019183028A JP2019183028A JP2020073474A5 JP 2020073474 A5 JP2020073474 A5 JP 2020073474A5 JP 2019183028 A JP2019183028 A JP 2019183028A JP 2019183028 A JP2019183028 A JP 2019183028A JP 2020073474 A5 JP2020073474 A5 JP 2020073474A5
Authority
JP
Japan
Prior art keywords
compound
salt
trifluoromethanesulfonyloxy
toluenesulfonyloxy
methanesulfonyloxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP2019183028A
Other languages
English (en)
Japanese (ja)
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JP2020073474A (ja
Filing date
Publication date
Application filed filed Critical
Publication of JP2020073474A publication Critical patent/JP2020073474A/ja
Publication of JP2020073474A5 publication Critical patent/JP2020073474A5/ja
Ceased legal-status Critical Current

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JP2019183028A 2016-11-25 2019-10-03 トリアゾロピリジン化合物の製造方法 Ceased JP2020073474A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2016228897 2016-11-25
JP2016228897 2016-11-25

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2018552978A Division JP6600103B2 (ja) 2016-11-25 2017-11-24 トリアゾロピリジン化合物の製造方法

Publications (2)

Publication Number Publication Date
JP2020073474A JP2020073474A (ja) 2020-05-14
JP2020073474A5 true JP2020073474A5 (enExample) 2021-01-07

Family

ID=62195187

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2018552978A Active JP6600103B2 (ja) 2016-11-25 2017-11-24 トリアゾロピリジン化合物の製造方法
JP2019183028A Ceased JP2020073474A (ja) 2016-11-25 2019-10-03 トリアゾロピリジン化合物の製造方法

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2018552978A Active JP6600103B2 (ja) 2016-11-25 2017-11-24 トリアゾロピリジン化合物の製造方法

Country Status (11)

Country Link
US (1) US11434238B2 (enExample)
EP (1) EP3546459A4 (enExample)
JP (2) JP6600103B2 (enExample)
KR (1) KR102523786B1 (enExample)
CN (1) CN110214139B (enExample)
AU (1) AU2017364725B2 (enExample)
CA (1) CA3044654A1 (enExample)
IL (1) IL266858B (enExample)
MX (1) MX2019006083A (enExample)
RU (1) RU2752384C2 (enExample)
WO (1) WO2018097254A1 (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2752384C2 (ru) * 2016-11-25 2021-07-26 Джапан Тобакко Инк. Способ получения триазолопиридинового соединения
CN113387948B (zh) * 2021-02-06 2022-06-10 成都诺和晟泰生物科技有限公司 一种稠环杂芳基衍生物及其药物组合物和治疗方法及用途
CN114773333A (zh) * 2021-12-25 2022-07-22 上海泰坦科技股份有限公司 一种卤代三唑并吡啶的合成方法
CN117327066A (zh) * 2022-06-30 2024-01-02 上海济煜医药科技有限公司 一种新多晶型、其制备方法及其用于制备药物的用途
CN117486878A (zh) * 2023-10-27 2024-02-02 扬州市普林斯医药科技有限公司 一种恩那司他的制备方法
CN119039291A (zh) * 2024-09-09 2024-11-29 南京药坦生物科技有限公司 一种恩那度司他中间体及其制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT2455381E (pt) * 2009-07-17 2014-06-24 Japan Tobacco Inc Composto de triazolopiridina e sua acção como inibidor da prolil-hidroxilase e indutor da produção de eritropoietina
EP3305293A4 (en) * 2015-05-28 2019-01-16 Japan Tobacco Inc. METHOD FOR THE TREATMENT OR PREVENTION OF NEPHROPATHIA DIABETICA
ES2909122T3 (es) * 2015-11-09 2022-05-05 Forge Therapeutics Inc Compuestos a base de hidroxipiridinona e hidroxipirimidinona para el tratamiento de infecciones bacterianas
RU2752384C2 (ru) * 2016-11-25 2021-07-26 Джапан Тобакко Инк. Способ получения триазолопиридинового соединения

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