JP2020073474A5 - - Google Patents
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- Publication number
- JP2020073474A5 JP2020073474A5 JP2019183028A JP2019183028A JP2020073474A5 JP 2020073474 A5 JP2020073474 A5 JP 2020073474A5 JP 2019183028 A JP2019183028 A JP 2019183028A JP 2019183028 A JP2019183028 A JP 2019183028A JP 2020073474 A5 JP2020073474 A5 JP 2020073474A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- salt
- trifluoromethanesulfonyloxy
- toluenesulfonyloxy
- methanesulfonyloxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
- 150000003839 salts Chemical class 0.000 claims 21
- 150000001875 compounds Chemical class 0.000 claims 17
- -1 p-toluenesulfonyloxy, methanesulfonyloxy Chemical group 0.000 claims 10
- 238000004519 manufacturing process Methods 0.000 claims 8
- NMJQBLVCTWZTJG-UHFFFAOYSA-M 1,2-dimethyl-1-[3-(2-methylphenoxy)-3-phenylpropyl]piperidin-1-ium;bromide Chemical compound [Br-].CC1CCCC[N+]1(C)CCC(C=1C=CC=CC=1)OC1=CC=CC=C1C NMJQBLVCTWZTJG-UHFFFAOYSA-M 0.000 claims 4
- 125000000217 alkyl group Chemical group 0.000 claims 4
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 claims 4
- 229910052736 halogen Inorganic materials 0.000 claims 4
- 150000002367 halogens Chemical class 0.000 claims 4
- 125000005951 trifluoromethanesulfonyloxy group Chemical group 0.000 claims 4
- MEKOFIRRDATTAG-UHFFFAOYSA-N 2,2,5,8-tetramethyl-3,4-dihydrochromen-6-ol Chemical compound C1CC(C)(C)OC2=C1C(C)=C(O)C=C2C MEKOFIRRDATTAG-UHFFFAOYSA-N 0.000 claims 3
- DTQVDTLACAAQTR-UHFFFAOYSA-N Trifluoroacetic acid Chemical group OC(=O)C(F)(F)F DTQVDTLACAAQTR-UHFFFAOYSA-N 0.000 claims 3
- JAEJSNFTJMYIEF-UHFFFAOYSA-N 2-benzylpropanedioic acid Chemical class OC(=O)C(C(O)=O)CC1=CC=CC=C1 JAEJSNFTJMYIEF-UHFFFAOYSA-N 0.000 claims 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2016228897 | 2016-11-25 | ||
| JP2016228897 | 2016-11-25 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018552978A Division JP6600103B2 (ja) | 2016-11-25 | 2017-11-24 | トリアゾロピリジン化合物の製造方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2020073474A JP2020073474A (ja) | 2020-05-14 |
| JP2020073474A5 true JP2020073474A5 (enExample) | 2021-01-07 |
Family
ID=62195187
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018552978A Active JP6600103B2 (ja) | 2016-11-25 | 2017-11-24 | トリアゾロピリジン化合物の製造方法 |
| JP2019183028A Ceased JP2020073474A (ja) | 2016-11-25 | 2019-10-03 | トリアゾロピリジン化合物の製造方法 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018552978A Active JP6600103B2 (ja) | 2016-11-25 | 2017-11-24 | トリアゾロピリジン化合物の製造方法 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US11434238B2 (enExample) |
| EP (1) | EP3546459A4 (enExample) |
| JP (2) | JP6600103B2 (enExample) |
| KR (1) | KR102523786B1 (enExample) |
| CN (1) | CN110214139B (enExample) |
| AU (1) | AU2017364725B2 (enExample) |
| CA (1) | CA3044654A1 (enExample) |
| IL (1) | IL266858B (enExample) |
| MX (1) | MX2019006083A (enExample) |
| RU (1) | RU2752384C2 (enExample) |
| WO (1) | WO2018097254A1 (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2018097254A1 (ja) * | 2016-11-25 | 2018-05-31 | 日本たばこ産業株式会社 | トリアゾロピリジン化合物の製造方法 |
| CN113387948B (zh) * | 2021-02-06 | 2022-06-10 | 成都诺和晟泰生物科技有限公司 | 一种稠环杂芳基衍生物及其药物组合物和治疗方法及用途 |
| CN114773333A (zh) * | 2021-12-25 | 2022-07-22 | 上海泰坦科技股份有限公司 | 一种卤代三唑并吡啶的合成方法 |
| CN117486878A (zh) * | 2023-10-27 | 2024-02-02 | 扬州市普林斯医药科技有限公司 | 一种恩那司他的制备方法 |
| CN119039291A (zh) * | 2024-09-09 | 2024-11-29 | 南京药坦生物科技有限公司 | 一种恩那度司他中间体及其制备方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK2455381T5 (en) * | 2009-07-17 | 2015-02-09 | Japan Tobacco Inc | Triazolopyridinforbindelse and its effect as an inhibitor of prolyl hydroxylase and induce erythropoietin production by |
| JP6814134B2 (ja) | 2015-05-28 | 2021-01-13 | 日本たばこ産業株式会社 | 糖尿病性腎症を治療又は予防する方法 |
| EP3374350B1 (en) * | 2015-11-09 | 2022-01-05 | Forge Therapeutics, Inc. | Hydroxypyridinone and hydroxypyrimidinone based compounds for treating bacterial infections |
| WO2018097254A1 (ja) * | 2016-11-25 | 2018-05-31 | 日本たばこ産業株式会社 | トリアゾロピリジン化合物の製造方法 |
-
2017
- 2017-11-24 WO PCT/JP2017/042239 patent/WO2018097254A1/ja not_active Ceased
- 2017-11-24 MX MX2019006083A patent/MX2019006083A/es unknown
- 2017-11-24 JP JP2018552978A patent/JP6600103B2/ja active Active
- 2017-11-24 US US16/463,216 patent/US11434238B2/en active Active
- 2017-11-24 EP EP17874271.4A patent/EP3546459A4/en active Pending
- 2017-11-24 CN CN201780072928.2A patent/CN110214139B/zh active Active
- 2017-11-24 RU RU2019119584A patent/RU2752384C2/ru active
- 2017-11-24 CA CA3044654A patent/CA3044654A1/en active Pending
- 2017-11-24 AU AU2017364725A patent/AU2017364725B2/en active Active
- 2017-11-24 KR KR1020197015696A patent/KR102523786B1/ko active Active
-
2019
- 2019-05-23 IL IL266858A patent/IL266858B/en unknown
- 2019-10-03 JP JP2019183028A patent/JP2020073474A/ja not_active Ceased
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