JP2019534301A5 - - Google Patents
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- Publication number
- JP2019534301A5 JP2019534301A5 JP2019524149A JP2019524149A JP2019534301A5 JP 2019534301 A5 JP2019534301 A5 JP 2019534301A5 JP 2019524149 A JP2019524149 A JP 2019524149A JP 2019524149 A JP2019524149 A JP 2019524149A JP 2019534301 A5 JP2019534301 A5 JP 2019534301A5
- Authority
- JP
- Japan
- Prior art keywords
- substituted
- alkyl
- hydrogen
- present
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662420182P | 2016-11-10 | 2016-11-10 | |
| US62/420,182 | 2016-11-10 | ||
| US201662433425P | 2016-12-13 | 2016-12-13 | |
| US62/433,425 | 2016-12-13 | ||
| PCT/US2017/060507 WO2018089406A1 (en) | 2016-11-10 | 2017-11-08 | Ror gamma modulators |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2019534301A JP2019534301A (ja) | 2019-11-28 |
| JP2019534301A5 true JP2019534301A5 (enExample) | 2020-11-12 |
Family
ID=60570205
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019524149A Withdrawn JP2019534301A (ja) | 2016-11-10 | 2017-11-08 | Rorガンマ調節剤 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US11078186B2 (enExample) |
| EP (1) | EP3538522A1 (enExample) |
| JP (1) | JP2019534301A (enExample) |
| KR (1) | KR20190076041A (enExample) |
| CN (1) | CN110167930A (enExample) |
| MA (1) | MA46760A (enExample) |
| WO (1) | WO2018089406A1 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP7014795B2 (ja) * | 2016-12-13 | 2022-02-01 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Rorガンマのモデュレーターとしての化合物 |
| US11034669B2 (en) | 2018-11-30 | 2021-06-15 | Nuvation Bio Inc. | Pyrrole and pyrazole compounds and methods of use thereof |
| CN109761863B (zh) * | 2019-01-19 | 2020-10-02 | 湘潭大学 | (e)-(2-(苯基磺酰基)乙烯基)苯及其衍生物及合成方法 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2852526A (en) * | 1955-05-03 | 1958-09-16 | Schering Corp | Substituted pyrrolidines |
| JPS5821622B2 (ja) * | 1973-02-28 | 1983-05-02 | ウェルファイド株式会社 | ピロリジンメタノ−ル ノ セイゾウホウ |
| JP3637974B2 (ja) * | 1993-03-25 | 2005-04-13 | エーザイ株式会社 | ピロリジン誘導体 |
| US5665754A (en) * | 1993-09-20 | 1997-09-09 | Glaxo Wellcome Inc. | Substituted pyrrolidines |
| CN105209457A (zh) * | 2013-03-15 | 2015-12-30 | 艾伯维德国有限责任两合公司 | 吡咯烷衍生物,含有其的药物组合物及其在治疗中的用途 |
| ES2669208T3 (es) * | 2014-01-06 | 2018-05-24 | Bristol-Myers Squibb Company | Derivados de pirrolidinilsulfona y su uso como moduladores de ROR gamma |
-
2017
- 2017-11-08 CN CN201780082798.0A patent/CN110167930A/zh active Pending
- 2017-11-08 MA MA046760A patent/MA46760A/fr unknown
- 2017-11-08 WO PCT/US2017/060507 patent/WO2018089406A1/en not_active Ceased
- 2017-11-08 KR KR1020197016350A patent/KR20190076041A/ko not_active Withdrawn
- 2017-11-08 US US16/348,195 patent/US11078186B2/en active Active
- 2017-11-08 JP JP2019524149A patent/JP2019534301A/ja not_active Withdrawn
- 2017-11-08 EP EP17808660.9A patent/EP3538522A1/en not_active Withdrawn
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