JP2019534301A - Ｒｏｒガンマ調節剤 - Google Patents

Ｒｏｒガンマ調節剤 Download PDF

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JP2019534301A
JP2019534301A JP2019524149A JP2019524149A JP2019534301A JP 2019534301 A JP2019534301 A JP 2019534301A JP 2019524149 A JP2019524149 A JP 2019524149A JP 2019524149 A JP2019524149 A JP 2019524149A JP 2019534301 A JP2019534301 A JP 2019534301A
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substituted
alkyl
phenyl
hydrogen
independently
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JP2019534301A5 (enExample
Inventor
ジンウー・ドワン
ビン・ジアン
ティ・ジー・ムラリ・ダール
ジョンホイ・ルー
アルン・クマール・グプタ
アナンタ・カルマカル
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Bristol Myers Squibb Co
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Bristol Myers Squibb Co
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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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    • A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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    • A61K31/415—1,2-Diazoles
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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