JP2019526537A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2019526537A5 JP2019526537A5 JP2019503703A JP2019503703A JP2019526537A5 JP 2019526537 A5 JP2019526537 A5 JP 2019526537A5 JP 2019503703 A JP2019503703 A JP 2019503703A JP 2019503703 A JP2019503703 A JP 2019503703A JP 2019526537 A5 JP2019526537 A5 JP 2019526537A5
- Authority
- JP
- Japan
- Prior art keywords
- human insulin
- zinc complex
- acylated derivative
- group
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2022066071A JP2022095872A (ja) | 2016-08-02 | 2022-04-13 | ヒトインスリンまたはそのアナログのアシル化誘導体 |
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN201610625257 | 2016-08-02 | ||
| CN201610625257.5 | 2016-08-02 | ||
| CN201610779132.8 | 2016-08-31 | ||
| CN201610779132 | 2016-08-31 | ||
| PCT/CN2017/095377 WO2018024186A1 (zh) | 2016-08-02 | 2017-08-01 | 一种人胰岛素或其类似物的酰化衍生物 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022066071A Division JP2022095872A (ja) | 2016-08-02 | 2022-04-13 | ヒトインスリンまたはそのアナログのアシル化誘導体 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2019526537A JP2019526537A (ja) | 2019-09-19 |
| JP2019526537A5 true JP2019526537A5 (enExample) | 2020-07-02 |
| JP7432361B2 JP7432361B2 (ja) | 2024-02-16 |
Family
ID=61074099
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019503703A Active JP7432361B2 (ja) | 2016-08-02 | 2017-08-01 | ヒトインスリンまたはそのアナログのアシル化誘導体 |
| JP2022066071A Pending JP2022095872A (ja) | 2016-08-02 | 2022-04-13 | ヒトインスリンまたはそのアナログのアシル化誘導体 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022066071A Pending JP2022095872A (ja) | 2016-08-02 | 2022-04-13 | ヒトインスリンまたはそのアナログのアシル化誘導体 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US10815287B2 (enExample) |
| EP (1) | EP3495384A4 (enExample) |
| JP (2) | JP7432361B2 (enExample) |
| CN (2) | CN114478747B (enExample) |
| TW (1) | TWI747929B (enExample) |
| WO (1) | WO2018024186A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2019149245A1 (zh) * | 2018-02-01 | 2019-08-08 | 江苏恒瑞医药股份有限公司 | 含人胰岛素类似物的酰化衍生物的药物组合物及其制备方法 |
| MX2020007929A (es) | 2018-02-09 | 2020-10-01 | Jiangsu Hengrui Medicine Co | Gen percursor del codón optimizado y gen de péptido señal de analógo de la insulina humana. |
| EP3805257A4 (en) | 2018-05-24 | 2022-03-16 | Jiangsu Hengrui Medicine Co., Ltd. | METHOD OF PRODUCTION OF A PRECURSOR OF RECOMBINANT HUMAN INSULIN OR ANALOGUE THEREOF |
| SG11202106168VA (en) | 2018-12-11 | 2021-07-29 | Sanofi Sa | Insulin analogs having reduced insulin receptor binding affinity |
| CN118772259A (zh) * | 2019-12-30 | 2024-10-15 | 甘李药业股份有限公司 | 胰岛素衍生物 |
| CN116583531A (zh) * | 2020-11-27 | 2023-08-11 | 江苏恒瑞医药股份有限公司 | 一种制备胰岛素或其类似物的酰化衍生物的方法 |
| CN112939771A (zh) * | 2021-01-28 | 2021-06-11 | 宁夏蓝博思化学技术有限公司 | 长链烷基二酸单叔丁酯的制备方法 |
| KR20240013778A (ko) | 2021-05-24 | 2024-01-30 | 선샤인 레이크 파르마 컴퍼니 리미티드 | 신규한 아실화된 인슐린 유사체 |
| US20250262282A1 (en) | 2021-06-25 | 2025-08-21 | Gan & Lee Pharmaceuticals Co., Ltd. | Acylated Insulin-Containing Pharmaceutical Composition |
| EP4471053A1 (en) | 2022-01-28 | 2024-12-04 | Gan & Lee Pharmaceuticals Co., Ltd. | Acylated insulin |
| CN117756914B (zh) * | 2023-12-15 | 2024-09-03 | 瀚晖制药有限公司 | 依柯胰岛素的制备方法 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PH25772A (en) * | 1985-08-30 | 1991-10-18 | Novo Industri As | Insulin analogues, process for their preparation |
| SI0792290T1 (en) * | 1993-09-17 | 2001-12-31 | Novo Nordisk As | Acylated insulin |
| CN1163574A (zh) * | 1994-11-17 | 1997-10-29 | 伊莱利利公司 | 酰化的胰岛素类似物 |
| US6310038B1 (en) * | 1997-03-20 | 2001-10-30 | Novo Nordisk A/S | Pulmonary insulin crystals |
| AU2003208316A1 (en) * | 2002-03-13 | 2003-09-22 | Novo Nordisk A/S | Minimising body weight gain in insulin treatment |
| KR101159559B1 (ko) * | 2003-08-05 | 2012-06-26 | 노보 노르디스크 에이/에스 | 신규의 인슐린 유도체 |
| KR101186851B1 (ko) * | 2003-08-05 | 2012-10-02 | 노보 노르디스크 에이/에스 | 신규의 인슐린 유도체 |
| US20090074882A1 (en) * | 2005-12-28 | 2009-03-19 | Novo Nordisk A/S | Insulin compositions and method of making a composition |
| CN101784563B (zh) | 2007-08-15 | 2015-02-04 | 诺沃-诺迪斯克有限公司 | 具有包括含亚烷基二醇的氨基酸的重复单位的酰基部分的胰岛素 |
| MX2010009850A (es) * | 2008-03-18 | 2010-09-30 | Novo Nordisk As | Analogos de insulina acilados y etabilizados contra proteasas. |
| US8935928B2 (en) * | 2011-10-10 | 2015-01-20 | Lockheed Martin Corporation | Integrated air-cycle refrigeration and power generation system |
| EP2784085A4 (en) * | 2011-12-15 | 2015-07-08 | Shanghai Hengrui Pharm Co Ltd | HUMAN INSULIN ANALOG AND ACYLATED DERIVATIVITY THEREOF |
| CN106496322A (zh) | 2015-09-07 | 2017-03-15 | 江苏恒瑞医药股份有限公司 | 人胰岛素或其类似物的酰化衍生物的制备方法 |
| KR20180105236A (ko) * | 2016-02-05 | 2018-09-27 | 메모리얼 슬로안-케터링 캔서 센터 | 줄기 세포-유래 외배엽 계통 전구체의 분화 방법 |
-
2017
- 2017-08-01 TW TW106125882A patent/TWI747929B/zh active
- 2017-08-01 US US16/320,997 patent/US10815287B2/en active Active
- 2017-08-01 WO PCT/CN2017/095377 patent/WO2018024186A1/zh not_active Ceased
- 2017-08-01 CN CN202210131921.6A patent/CN114478747B/zh active Active
- 2017-08-01 JP JP2019503703A patent/JP7432361B2/ja active Active
- 2017-08-01 CN CN201780005001.7A patent/CN108463468B/zh active Active
- 2017-08-01 EP EP17836368.5A patent/EP3495384A4/en not_active Withdrawn
-
2022
- 2022-04-13 JP JP2022066071A patent/JP2022095872A/ja active Pending
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2019526537A5 (enExample) | ||
| JP2022095872A5 (enExample) | ||
| JP2012512901A5 (enExample) | ||
| JP2011006428A5 (enExample) | ||
| RU99106518A (ru) | Glp-1 производные | |
| RU2008143668A (ru) | Производное инсулина | |
| WO2019117274A1 (ja) | ペプチドの製造方法、及び塩基の処理方法 | |
| JP2016523241A5 (enExample) | ||
| WO2011080102A3 (en) | Glp-1 analogues and derivatives | |
| CA3084688A1 (fr) | Solution injectable a ph 7 comprenant au moins une insuline basale dont le pi est compris entre 5,8 et 8,5 et un co-polyaminoacide porteur de charges carboxylates et de radicaux hydrophobes | |
| JP2013526501A5 (enExample) | ||
| JP2015110654A5 (enExample) | ||
| RU2009122582A (ru) | Пэг-модифицированный эксендин или аналог эксендина и его композиции и применение | |
| JP2007523881A5 (enExample) | ||
| KR970042553A (ko) | 캠프토테신 유도체 | |
| EP3495384A1 (en) | Acylated derivative of human insulin or analogue thereof | |
| RU2008141280A (ru) | Агонисты рецептора нейромедина u и их применение | |
| JP2008545793A5 (enExample) | ||
| NZ599791A (en) | Therapeutic peptides | |
| RU2019109719A (ru) | Конъюгаты полимиксин-альгинатных олигомеров | |
| JP5982562B2 (ja) | ペプチドの塩酸塩及び他のペプチドとの併用によるその免疫治療用途 | |
| JP2017508741A5 (enExample) | ||
| JP2009532384A5 (enExample) | ||
| EP3740227A1 (fr) | Compositions sous forme d'une solution aqueuse injectable comprenant de l'amyline, un agoniste au recepteur de l'amyline ou un analogue d'amyline et un co-polyaminoacide | |
| RU2020108281A (ru) | Новые ацилированные аналоги инсулина и варианты их применения |