JP2019507130A5 - - Google Patents
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- Publication number
- JP2019507130A5 JP2019507130A5 JP2018539873A JP2018539873A JP2019507130A5 JP 2019507130 A5 JP2019507130 A5 JP 2019507130A5 JP 2018539873 A JP2018539873 A JP 2018539873A JP 2018539873 A JP2018539873 A JP 2018539873A JP 2019507130 A5 JP2019507130 A5 JP 2019507130A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- cycloalkyl
- heterocycloalkyl
- compound according
- aryl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 CCCCC*(C(C(C)C(N1C)=O)C1=O)=C Chemical compound CCCCC*(C(C(C)C(N1C)=O)C1=O)=C 0.000 description 6
- XDTMQSROBMDMFD-UHFFFAOYSA-N C1CCCCC1 Chemical compound C1CCCCC1 XDTMQSROBMDMFD-UHFFFAOYSA-N 0.000 description 3
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2021126415A JP7257462B2 (ja) | 2016-02-01 | 2021-08-02 | ベンゾピラゾール化合物及びその類似体 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662289653P | 2016-02-01 | 2016-02-01 | |
| US62/289,653 | 2016-02-01 | ||
| PCT/US2017/015953 WO2017136395A1 (en) | 2016-02-01 | 2017-02-01 | Benzopyrazole compounds and analogues thereof |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021126415A Division JP7257462B2 (ja) | 2016-02-01 | 2021-08-02 | ベンゾピラゾール化合物及びその類似体 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2019507130A JP2019507130A (ja) | 2019-03-14 |
| JP2019507130A5 true JP2019507130A5 (enExample) | 2020-02-27 |
| JP6924766B2 JP6924766B2 (ja) | 2021-08-25 |
Family
ID=59500923
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018539873A Active JP6924766B2 (ja) | 2016-02-01 | 2017-02-01 | ベンゾピラゾール化合物及びその類似体 |
| JP2021126415A Active JP7257462B2 (ja) | 2016-02-01 | 2021-08-02 | ベンゾピラゾール化合物及びその類似体 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021126415A Active JP7257462B2 (ja) | 2016-02-01 | 2021-08-02 | ベンゾピラゾール化合物及びその類似体 |
Country Status (30)
| Country | Link |
|---|---|
| US (3) | US10849883B2 (enExample) |
| EP (2) | EP3925956B1 (enExample) |
| JP (2) | JP6924766B2 (enExample) |
| KR (1) | KR102828456B1 (enExample) |
| CN (2) | CN115490751B (enExample) |
| AR (1) | AR107488A1 (enExample) |
| AU (1) | AU2017213768B2 (enExample) |
| CA (1) | CA3011549A1 (enExample) |
| CO (1) | CO2018008916A2 (enExample) |
| CY (1) | CY1124652T1 (enExample) |
| DK (1) | DK3411411T6 (enExample) |
| EA (1) | EA039719B1 (enExample) |
| ES (2) | ES2982426T3 (enExample) |
| HR (1) | HRP20210926T4 (enExample) |
| HU (1) | HUE055258T2 (enExample) |
| IL (2) | IL290154B2 (enExample) |
| LT (1) | LT3411411T (enExample) |
| MA (1) | MA43979B1 (enExample) |
| MD (1) | MD3411411T2 (enExample) |
| MX (2) | MX2018008869A (enExample) |
| MY (1) | MY201629A (enExample) |
| PH (1) | PH12018501537B1 (enExample) |
| PL (1) | PL3411411T6 (enExample) |
| PT (1) | PT3411411T (enExample) |
| RS (1) | RS62187B2 (enExample) |
| SG (2) | SG11201805940QA (enExample) |
| SI (1) | SI3411411T1 (enExample) |
| SM (1) | SMT202100494T1 (enExample) |
| TW (2) | TWI747873B (enExample) |
| WO (1) | WO2017136395A1 (enExample) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2017035361A1 (en) | 2015-08-26 | 2017-03-02 | Achillion Pharmaceuticals, Inc. | Disubstituted compounds for the treatment of medical disorders |
| AR106018A1 (es) | 2015-08-26 | 2017-12-06 | Achillion Pharmaceuticals Inc | Compuestos de arilo, heteroarilo y heterocíclicos para el tratamiento de trastornos médicos |
| AR105809A1 (es) | 2015-08-26 | 2017-11-08 | Achillion Pharmaceuticals Inc | Compuestos para el tratamiento de trastornos médicos |
| WO2017035401A1 (en) | 2015-08-26 | 2017-03-02 | Achillion Pharmaceuticals, Inc. | Amide compounds for treatment of immune and inflammatory disorders |
| EP3340983B1 (en) | 2015-08-26 | 2023-10-04 | Achillion Pharmaceuticals, Inc. | Aryl, heteroaryl, and heterocyclic compounds for treatment of immune and inflammatory disorders |
| WO2017035357A1 (en) | 2015-08-26 | 2017-03-02 | Achillion Pharmaceuticals, Inc. | Phosphonate compounds for treatment of medical disorders |
| EP3340982B1 (en) | 2015-08-26 | 2021-12-15 | Achillion Pharmaceuticals, Inc. | Compounds for treatment of immune and inflammatory disorders |
| WO2017035405A1 (en) | 2015-08-26 | 2017-03-02 | Achillion Pharmaceuticals, Inc. | Amino compounds for treatment of immune and inflammatory disorders |
| TWI747873B (zh) | 2016-02-01 | 2021-12-01 | 美商百歐克斯製藥公司 | 苯并吡唑化合物及其類似物 |
| WO2018160892A1 (en) | 2017-03-01 | 2018-09-07 | Achillion Pharmaceuticals, Inc. | Macrocyclic compounds for treatment of medical disorders |
| KR102632860B1 (ko) | 2017-03-01 | 2024-02-02 | 아칠리온 파르마세우티칼스 인코포레이티드 | 의학적 장애의 치료를 위한 아릴, 헤테로아릴, 및 헤테로사이클릭 약학적 화합물 |
| WO2018160891A1 (en) | 2017-03-01 | 2018-09-07 | Achillion Pharmaceutical, Inc. | Pharmaceutical compounds for treatment of medical disorders |
| TWI873092B (zh) | 2018-04-06 | 2025-02-21 | 美商百歐克斯製藥公司 | 取代的苯并呋喃、苯并吡咯、苯并噻吩及結構相關的補體抑制劑 |
| US12448374B2 (en) | 2018-06-07 | 2025-10-21 | Disarm Therapeutics, Inc. | Inhibitors of SARM1 |
| US20230022157A1 (en) | 2018-08-20 | 2023-01-26 | Achillion Pharmaceuticals, Inc. | Pharmaceutical compounds for the treatment of complement factor d medical disorders |
| US11814363B2 (en) | 2018-09-06 | 2023-11-14 | Achillion Pharmaceuticals, Inc. | Morphic forms of danicopan |
| EP3846803A4 (en) | 2018-09-06 | 2022-08-10 | Achillion Pharmaceuticals, Inc. | Macrocyclic compounds for the treatment of medical disorders |
| EP3856164B1 (en) | 2018-09-25 | 2024-08-07 | Achillion Pharmaceuticals, Inc. | Morphic forms of complement factor d inhibitors |
| BR112021011727A2 (pt) | 2018-12-17 | 2021-08-31 | Achillion Pharmaceuticals, Inc | Dosagem direcionada para o tratamento de distúrbios mediados do complemento |
| CN113164508B (zh) | 2018-12-19 | 2025-07-08 | 达萨玛治疗公司 | 与神经保护剂组合的sarm1抑制剂 |
| WO2020198062A1 (en) | 2019-03-22 | 2020-10-01 | Achillion Pharmaceuticals, Inc. | Pharmaceutical compounds for the treatment of complement mediated disorders |
| UY38912A (es) | 2019-10-09 | 2021-05-31 | Biocryst Pharm Inc | Inhibidores del factor d del complemento para administración oral |
| TWI890699B (zh) * | 2019-10-09 | 2025-07-21 | 美商百歐克斯製藥公司 | 口服補體因子d抑制劑 |
| CN115362162A (zh) | 2020-02-20 | 2022-11-18 | 艾其林医药公司 | 用于治疗补体因子d介导的障碍的杂芳基化合物 |
| AR121715A1 (es) | 2020-04-03 | 2022-06-29 | Biocryst Pharm Inc | Pirrolopirimidinaminas como inhibidores del sistema del complemento |
| CN113512025B (zh) * | 2020-07-31 | 2023-01-06 | 四川大学 | 一种吲唑酯类化合物及其制药用途 |
| WO2025080823A1 (en) | 2023-10-11 | 2025-04-17 | Regeneron Pharmaceuticals, Inc. | Treatment of macular degeneration with complement factor d (cfd) inhibitors |
| CN119638611B (zh) * | 2024-12-08 | 2025-10-31 | 胥江生物科技(苏州)有限公司 | N-乙酰-5-羟色胺衍生物、免疫原、抗体及检测试剂制备与应用 |
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| EP3340983B1 (en) | 2015-08-26 | 2023-10-04 | Achillion Pharmaceuticals, Inc. | Aryl, heteroaryl, and heterocyclic compounds for treatment of immune and inflammatory disorders |
| WO2017035415A1 (en) | 2015-08-26 | 2017-03-02 | Achillion Pharmaceuticals, Inc. | Alkyne compounds for treatment of immune and inflammatory disorders |
| WO2017035401A1 (en) | 2015-08-26 | 2017-03-02 | Achillion Pharmaceuticals, Inc. | Amide compounds for treatment of immune and inflammatory disorders |
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| WO2017035405A1 (en) | 2015-08-26 | 2017-03-02 | Achillion Pharmaceuticals, Inc. | Amino compounds for treatment of immune and inflammatory disorders |
| WO2017035418A1 (en) | 2015-08-26 | 2017-03-02 | Achillion Pharmaceuticals, Inc. | Disubstituted compounds for treatment of immune and inflammatory disorders |
| EP3340982B1 (en) | 2015-08-26 | 2021-12-15 | Achillion Pharmaceuticals, Inc. | Compounds for treatment of immune and inflammatory disorders |
| TWI747873B (zh) | 2016-02-01 | 2021-12-01 | 美商百歐克斯製藥公司 | 苯并吡唑化合物及其類似物 |
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2017
- 2017-01-26 TW TW106103180A patent/TWI747873B/zh active
- 2017-01-26 TW TW110141309A patent/TWI854164B/zh active
- 2017-01-30 AR ARP170100240A patent/AR107488A1/es unknown
- 2017-02-01 ES ES21173901T patent/ES2982426T3/es active Active
- 2017-02-01 PH PH1/2018/501537A patent/PH12018501537B1/en unknown
- 2017-02-01 MY MYPI2018001324A patent/MY201629A/en unknown
- 2017-02-01 AU AU2017213768A patent/AU2017213768B2/en active Active
- 2017-02-01 LT LTEP17748044.9T patent/LT3411411T/lt unknown
- 2017-02-01 PL PL17748044T patent/PL3411411T6/pl unknown
- 2017-02-01 JP JP2018539873A patent/JP6924766B2/ja active Active
- 2017-02-01 KR KR1020187024635A patent/KR102828456B1/ko active Active
- 2017-02-01 EP EP21173901.6A patent/EP3925956B1/en active Active
- 2017-02-01 MA MA43979A patent/MA43979B1/fr unknown
- 2017-02-01 MX MX2018008869A patent/MX2018008869A/es unknown
- 2017-02-01 MD MDE20181197T patent/MD3411411T2/ro unknown
- 2017-02-01 IL IL290154A patent/IL290154B2/en unknown
- 2017-02-01 CN CN202210705604.0A patent/CN115490751B/zh active Active
- 2017-02-01 SG SG11201805940QA patent/SG11201805940QA/en unknown
- 2017-02-01 EP EP17748044.9A patent/EP3411411B3/en active Active
- 2017-02-01 SM SM20210494T patent/SMT202100494T1/it unknown
- 2017-02-01 SI SI201730796T patent/SI3411411T1/sl unknown
- 2017-02-01 HU HUE17748044A patent/HUE055258T2/hu unknown
- 2017-02-01 RS RS20210979A patent/RS62187B2/sr unknown
- 2017-02-01 SG SG10202108797UA patent/SG10202108797UA/en unknown
- 2017-02-01 CA CA3011549A patent/CA3011549A1/en active Pending
- 2017-02-01 ES ES17748044T patent/ES2882495T7/es active Active
- 2017-02-01 CN CN201780021413.XA patent/CN109121414B/zh active Active
- 2017-02-01 EA EA201891703A patent/EA039719B1/ru unknown
- 2017-02-01 HR HRP20210926TT patent/HRP20210926T4/hr unknown
- 2017-02-01 PT PT177480449T patent/PT3411411T/pt unknown
- 2017-02-01 DK DK17748044.9T patent/DK3411411T6/da active
- 2017-02-01 US US16/073,934 patent/US10849883B2/en active Active
- 2017-02-01 WO PCT/US2017/015953 patent/WO2017136395A1/en not_active Ceased
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2018
- 2018-07-11 IL IL260545A patent/IL260545B/en unknown
- 2018-07-19 MX MX2022007915A patent/MX2022007915A/es unknown
- 2018-08-27 CO CONC2018/0008916A patent/CO2018008916A2/es unknown
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2020
- 2020-08-26 US US17/003,552 patent/US11559515B2/en active Active
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2021
- 2021-08-02 JP JP2021126415A patent/JP7257462B2/ja active Active
- 2021-08-03 CY CY20211100696T patent/CY1124652T1/el unknown
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2023
- 2023-01-23 US US18/158,029 patent/US12485109B2/en active Active