JP2018522929A5 - - Google Patents

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Publication number
JP2018522929A5
JP2018522929A5 JP2018507023A JP2018507023A JP2018522929A5 JP 2018522929 A5 JP2018522929 A5 JP 2018522929A5 JP 2018507023 A JP2018507023 A JP 2018507023A JP 2018507023 A JP2018507023 A JP 2018507023A JP 2018522929 A5 JP2018522929 A5 JP 2018522929A5
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JP
Japan
Prior art keywords
methyl
oxaspiro
methoxy
carboxylate
octane
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2018507023A
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English (en)
Japanese (ja)
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JP2018522929A (ja
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Publication date
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Priority claimed from PCT/US2016/046511 external-priority patent/WO2017027684A1/en
Publication of JP2018522929A publication Critical patent/JP2018522929A/ja
Publication of JP2018522929A5 publication Critical patent/JP2018522929A5/ja
Withdrawn legal-status Critical Current

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JP2018507023A 2015-08-11 2016-08-11 フマギロール複素環化合物ならびにその作製および使用方法 Withdrawn JP2018522929A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562203742P 2015-08-11 2015-08-11
US62/203,742 2015-08-11
PCT/US2016/046511 WO2017027684A1 (en) 2015-08-11 2016-08-11 Fumagillol heterocyclic compounds and methods of making and using same

Publications (2)

Publication Number Publication Date
JP2018522929A JP2018522929A (ja) 2018-08-16
JP2018522929A5 true JP2018522929A5 (enExample) 2019-08-29

Family

ID=56799580

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2018507023A Withdrawn JP2018522929A (ja) 2015-08-11 2016-08-11 フマギロール複素環化合物ならびにその作製および使用方法

Country Status (15)

Country Link
US (5) US20180230137A1 (enExample)
EP (1) EP3334728A1 (enExample)
JP (1) JP2018522929A (enExample)
KR (1) KR20180035907A (enExample)
CN (1) CN108026085A (enExample)
AR (1) AR105671A1 (enExample)
AU (1) AU2016306558A1 (enExample)
CA (1) CA2995366A1 (enExample)
EA (1) EA201890449A1 (enExample)
IL (1) IL257443A (enExample)
MA (1) MA42612A (enExample)
MX (1) MX2018001733A (enExample)
PH (1) PH12018500315A1 (enExample)
TW (1) TW201718550A (enExample)
WO (1) WO2017027684A1 (enExample)

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CN106432255A (zh) 2015-08-11 2017-02-22 扎夫根公司 烟曲霉素醇螺环化合物和制备和使用其的方法
US20200030278A1 (en) * 2017-02-10 2020-01-30 Zafgen, Inc. Pharmaceutical compositions of metap-2 inhibitors
WO2019118612A1 (en) * 2017-12-12 2019-06-20 Zafgen, Inc. Targeting compounds
WO2019173505A1 (en) * 2018-03-06 2019-09-12 Zafgen, Inc. Methods of treating disorders related to glycemic control
CN109180551A (zh) * 2018-07-17 2019-01-11 宜春学院 一种四元氮杂环中间体的制备方法
US11612577B2 (en) 2018-10-26 2023-03-28 Syndevrx, Inc. Biomarkers of METAP2 inhibitors and applications thereof
CN111606836B (zh) * 2020-06-12 2021-01-15 上海馨远医药科技有限公司 一种R-N-Boc-3-吡咯烷乙酸的制备方法
GB202011996D0 (en) 2020-07-31 2020-09-16 Adorx Therapeutics Ltd Antagonist compounds

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