|
HRP20161774T1
(hr)
|
2012-06-13 |
2017-02-24 |
F. Hoffmann - La Roche Ag |
Novi diazaspirocikloalkan i azaspirocikloalkan
|
|
BR112015004111A2
(pt)
|
2012-09-25 |
2017-07-04 |
Hoffmann La Roche |
novos derivados bicíclicos
|
|
AR095079A1
(es)
|
2013-03-12 |
2015-09-16 |
Hoffmann La Roche |
Derivados de octahidro-pirrolo[3,4-c]-pirrol y piridina-fenilo
|
|
KR20160087900A
(ko)
|
2013-11-26 |
2016-07-22 |
에프. 호프만-라 로슈 아게 |
신규한 옥타하이드로-사이클로부타[1,2-c;3,4-c'']다이피롤-2-일
|
|
SI3122750T1
(sl)
|
2014-03-26 |
2019-12-31 |
F. Hoffmann-La Roche Ag |
Biciklične spojine kot zaviralci proizvodnje avtotaksina (ATX) in lizofosfatidne kisline (LPA)
|
|
KR20160128428A
(ko)
|
2014-03-26 |
2016-11-07 |
에프. 호프만-라 로슈 아게 |
오토탁신(atx) 및 리소포스파티드산(lpa) 생성 억제제로서의 축합형 [1,4]다이아제핀 화합물
|
|
TWI676626B
(zh)
*
|
2014-04-23 |
2019-11-11 |
美商美國禮來大藥廠 |
抑制瞬時受體電位a1離子通道
|
|
EP3798214B1
(en)
|
2014-10-06 |
2022-09-14 |
Vertex Pharmaceuticals Incorporated |
Modulators of cystic fibrosis transmembrane conductance regulator
|
|
BR112017019150B1
(pt)
|
2015-03-06 |
2023-05-09 |
Pharmakea, Inc |
Compostos inibidores de lisil oxidase-like 2 fluorados, composição farmacêutica e uso desses compostos
|
|
EP3265445B1
(en)
|
2015-03-06 |
2021-05-05 |
Pharmakea, Inc. |
Lysyl oxidase-like 2 inhibitors and uses thereof
|
|
MA41898A
(fr)
|
2015-04-10 |
2018-02-13 |
Hoffmann La Roche |
Dérivés de quinazolinone bicyclique
|
|
WO2017003862A1
(en)
*
|
2015-07-01 |
2017-01-05 |
Pharmakea, Inc. |
Lysyl oxidase-like 2 inhibitors and uses thereof
|
|
JP6886967B2
(ja)
|
2015-09-04 |
2021-06-16 |
エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft |
フェノキシメチル誘導体
|
|
AU2016328365B2
(en)
|
2015-09-24 |
2020-04-23 |
F. Hoffmann-La Roche Ag |
New bicyclic compounds as dual ATX/CA inhibitors
|
|
RU2018112230A
(ru)
|
2015-09-24 |
2019-10-30 |
Ф. Хоффманн-Ля Рош Аг |
Бициклические соединения в качестве ингибиторов atx
|
|
CN107635995B
(zh)
|
2015-09-24 |
2022-08-19 |
豪夫迈·罗氏有限公司 |
作为atx抑制剂的二环化合物
|
|
JP6877413B2
(ja)
|
2015-09-24 |
2021-05-26 |
エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft |
二重atx/ca阻害剤としての新規な二環式化合物
|
|
PL3412664T3
(pl)
*
|
2016-02-05 |
2022-06-06 |
Ea Pharma Co., Ltd. |
Heterocykliczna pochodna sulfonamidowa i lek zawierający tę pochodną
|
|
JP7043483B2
(ja)
*
|
2016-07-20 |
2022-03-29 |
エフ.ホフマン-ラ ロシュ アーゲー |
二環式プロリン化合物
|
|
JP6975515B2
(ja)
|
2016-07-20 |
2021-12-01 |
エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft |
Trpa1モデュレーターとしてのスルホニルシクロアルキルカルボキサミド化合物
|
|
EP3497093B1
(en)
*
|
2016-08-12 |
2021-09-15 |
F. Hoffmann-La Roche AG |
Sulfonyl pyridyl trp inhibitors
|
|
JP7079772B2
(ja)
|
2016-09-07 |
2022-06-02 |
ファーマケア,インク. |
リシルオキシダーゼ様2阻害剤の結晶形態および製造方法
|
|
KR102615565B1
(ko)
|
2016-09-07 |
2023-12-18 |
파마케아, 인크. |
리실 옥시다제 유사 2 억제제의 용도
|
|
MA49235B1
(fr)
|
2016-12-09 |
2021-02-26 |
Vertex Pharma |
Modulateur de régulateur de conductance transmembranaire de fibrose kystique, compositions pharmaceutiques, procédés de traitement et procédé de fabrication du modulateur
|
|
WO2018109155A1
(en)
|
2016-12-16 |
2018-06-21 |
Galderma Research & Development |
Trpa1 antagonists for use in the treatment of atopic dermatitis
|
|
AU2018207776B2
(en)
|
2017-01-10 |
2021-06-17 |
Bayer Aktiengesellschaft |
Heterocyclene derivatives as pest control agents
|
|
EP3596059B1
(en)
|
2017-03-16 |
2024-04-24 |
F. Hoffmann-La Roche AG |
Heterocyclic compounds useful as dual atx/ca inhibitors
|
|
WO2018167113A1
(en)
|
2017-03-16 |
2018-09-20 |
F. Hoffmann-La Roche Ag |
New bicyclic compounds as atx inhibitors
|
|
EP3634402B1
(en)
|
2017-06-08 |
2026-01-21 |
Vertex Pharmaceuticals Incorporated |
Methods of treatment for cystic fibrosis
|
|
BR112020000941A2
(pt)
|
2017-07-17 |
2020-07-21 |
Vertex Pharmaceuticals Incorporated |
métodos de tratamento para fibrose cística
|
|
TWI799435B
(zh)
|
2017-08-02 |
2023-04-21 |
美商維泰克斯製藥公司 |
製備化合物之製程
|
|
IL273831B2
(en)
|
2017-10-19 |
2024-10-01 |
Vertex Pharma |
Crystalline forms and compositions of cftr modulators
|
|
CN111757874B
(zh)
*
|
2017-12-08 |
2024-03-08 |
弗特克斯药品有限公司 |
用于制备囊性纤维化跨膜传导调节因子的调节剂的方法
|
|
TWI810243B
(zh)
|
2018-02-05 |
2023-08-01 |
美商維泰克斯製藥公司 |
用於治療囊腫纖化症之醫藥組合物
|
|
TW202000201A
(zh)
|
2018-02-20 |
2020-01-01 |
瑞士商赫孚孟拉羅股份公司 |
製備1-芳基磺醯基-吡咯啶-2-甲醯胺瞬時受體電位通道拮抗劑化合物及其結晶型式之方法
|
|
US10710994B2
(en)
|
2018-03-19 |
2020-07-14 |
Genentech, Inc. |
Oxadiazole transient receptor potential channel inhibitors
|
|
US11414439B2
(en)
|
2018-04-13 |
2022-08-16 |
Vertex Pharmaceuticals Incorporated |
Modulators of cystic fibrosis transmembrane conductance regulator, pharmaceutical compositions, methods of treatment, and process for making the modulator
|
|
CN112739689B
(zh)
|
2018-12-07 |
2022-06-03 |
优迈特株式会社 |
含氟嘧啶化合物及其制造方法
|
|
CN110156834A
(zh)
*
|
2019-06-05 |
2019-08-23 |
镇江市高等专科学校 |
一种黄色荧光铜(i)配合物及其制备方法和应用
|
|
EP4155299A4
(en)
|
2020-05-19 |
2024-07-10 |
Unimatec Co., Ltd. |
Fluoropyrimidine compound and fluoropyrimidinone compound
|
|
FR3114235A1
(fr)
|
2020-09-18 |
2022-03-25 |
Université Grenoble Alpes |
Inhibition du canal trpa1 astrocytaire comme nouvelle cible therapeutique neuroprotectrice dans les phases prodromales de la maladie d’alzheimer
|
|
KR20230107307A
(ko)
*
|
2020-11-19 |
2023-07-14 |
아코우지아 테라포이틱스 게엠베하 |
비수성 겔 조성물
|
|
IT202100015098A1
(it)
|
2021-06-09 |
2022-12-09 |
Flonext S R L |
Composto antagonista del canale trpa1 per uso in patologie degenerative della retina
|
|
WO2023133502A1
(en)
*
|
2022-01-07 |
2023-07-13 |
The Johns Hopkins University |
Treatment and prevention of trigeminal neuralgia
|
|
AR131541A1
(es)
|
2023-01-07 |
2025-04-09 |
Syngenta Crop Protection Ag |
Compuestos de carboxamida novedosos
|
|
WO2025109114A1
(en)
|
2023-11-24 |
2025-05-30 |
Syngenta Crop Protection Ag |
Novel carboxamide compounds
|
|
WO2025124698A1
(en)
|
2023-12-12 |
2025-06-19 |
Idorsia Pharmaceuticals Ltd |
Aryl sulfone and sulfanone derivatives as orexin receptor modulators
|
|
WO2025132542A1
(en)
|
2023-12-19 |
2025-06-26 |
Idorsia Pharmaceuticals Ltd |
Macrocyclic orexin agonists
|
|
WO2025149629A1
(en)
|
2024-01-12 |
2025-07-17 |
Syngenta Crop Protection Ag |
Novel carboxamide compounds
|
|
WO2025149637A1
(en)
|
2024-01-12 |
2025-07-17 |
Syngenta Crop Protection Ag |
Novel carboxamide compounds
|
|
WO2025155669A1
(en)
*
|
2024-01-17 |
2025-07-24 |
The Jackson Laboratory |
Trpc3 inhibitors and uses thereof
|
|
WO2026008750A1
(en)
|
2024-07-05 |
2026-01-08 |
Syngenta Crop Protection Ag |
Novel carboxamide compounds
|