JP2018504379A5 - - Google Patents
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- JP2018504379A5 JP2018504379A5 JP2017532682A JP2017532682A JP2018504379A5 JP 2018504379 A5 JP2018504379 A5 JP 2018504379A5 JP 2017532682 A JP2017532682 A JP 2017532682A JP 2017532682 A JP2017532682 A JP 2017532682A JP 2018504379 A5 JP2018504379 A5 JP 2018504379A5
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- alkyl
- hydrogen
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- methyl
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- 0 CCCC[C@@](C(N[C@@](CC(C)C)C(N[C@@](CSCC(N[C@@](Cc(cc1)ccc1O)C(N(C)[C@@](C)C(N[C@@](CC(N)=O)C(N(CCC1)[C@@]1C(N[C@](C1)C(N[C@@](CCC(O)=O)C(N(C[C@@](C2)O)[C@@]2C(N[C@@](Cc2c[n]c3c2cccc3)C(N[C@@](CCN)C(N[C@@](Cc2c[n]c3c2cccc3)C(N(CCN)[C@]2C)=O)=O)=O)=O)=O)=*3C1=CN=C3)=O)=O)=O)=O)=O)C(NCC(N)=O)=O)=O)=O)N(C)C2=O Chemical compound CCCC[C@@](C(N[C@@](CC(C)C)C(N[C@@](CSCC(N[C@@](Cc(cc1)ccc1O)C(N(C)[C@@](C)C(N[C@@](CC(N)=O)C(N(CCC1)[C@@]1C(N[C@](C1)C(N[C@@](CCC(O)=O)C(N(C[C@@](C2)O)[C@@]2C(N[C@@](Cc2c[n]c3c2cccc3)C(N[C@@](CCN)C(N[C@@](Cc2c[n]c3c2cccc3)C(N(CCN)[C@]2C)=O)=O)=O)=O)=O)=*3C1=CN=C3)=O)=O)=O)=O)=O)C(NCC(N)=O)=O)=O)=O)N(C)C2=O 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201462094008P | 2014-12-18 | 2014-12-18 | |
| US62/094,008 | 2014-12-18 | ||
| PCT/US2015/065723 WO2016100285A1 (en) | 2014-12-18 | 2015-12-15 | Immunomodulators |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2018504379A JP2018504379A (ja) | 2018-02-15 |
| JP2018504379A5 true JP2018504379A5 (https=) | 2018-04-26 |
| JP6625129B2 JP6625129B2 (ja) | 2019-12-25 |
Family
ID=55071200
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017532682A Active JP6625129B2 (ja) | 2014-12-18 | 2015-12-15 | 免疫修飾因子 |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US9861680B2 (https=) |
| EP (1) | EP3233888B1 (https=) |
| JP (1) | JP6625129B2 (https=) |
| KR (1) | KR102602643B1 (https=) |
| CN (1) | CN107108697B (https=) |
| AR (1) | AR103093A1 (https=) |
| AU (1) | AU2015362703A1 (https=) |
| BR (1) | BR112017012679A2 (https=) |
| CA (1) | CA2971189A1 (https=) |
| EA (1) | EA033894B1 (https=) |
| ES (1) | ES2940632T3 (https=) |
| IL (1) | IL252853A0 (https=) |
| MX (1) | MX2017007677A (https=) |
| SG (1) | SG11201704823TA (https=) |
| TW (1) | TW201629086A (https=) |
| WO (1) | WO2016100285A1 (https=) |
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| JP5818237B2 (ja) | 2010-09-09 | 2015-11-18 | 国立大学法人 東京大学 | Ｎ−メチルアミノ酸およびその他の特殊アミノ酸を含む特殊ペプチド化合物ライブラリーの翻訳構築と活性種探索法 |
| EP2647720B1 (en) | 2010-12-03 | 2019-06-19 | The University of Tokyo | Peptide library production method, peptide library, and screening method |
| WO2012168944A1 (en) | 2011-06-08 | 2012-12-13 | Aurigene Discovery Technologies Limited | Therapeutic compounds for immunomodulation |
| WO2013132317A1 (en) * | 2012-03-07 | 2013-09-12 | Aurigene Discovery Technologies Limited | Peptidomimetic compounds as immunomodulators |
| CA2868408A1 (en) | 2012-03-29 | 2013-10-03 | Aurigene Discovery Technologies Limited | Immunomodulating cyclic compounds from the bc loop of human pd1 |
| AU2013273481B2 (en) * | 2012-06-06 | 2018-04-05 | Bionor Immuno As | HIV vaccine |
| JP2013253842A (ja) | 2012-06-06 | 2013-12-19 | Univ Of Tokyo | ｐＨ依存的に標的分子に結合するペプチドのスクリーニング方法 |
| JP6047231B2 (ja) | 2012-06-06 | 2016-12-21 | ポリフォー・アクチェンゲゼルシャフトＰｏｌｙｐｈｏｒ Ａｇ | β−ヘアピンペプチド模倣薬 |
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| BR112015023120A2 (pt) | 2013-03-15 | 2017-11-21 | Genentech Inc | método para identificar um indivíduo com uma doença ou disfunção, método para prever a responsividade de um indivíduo com uma doença ou disfunção, método para determinar a probabilidade de que um indivíduo com uma doença ou disfunção exibirá benefício do tratamento, método para selecionar uma terapia, usos de um antagonista de ligação do eixo pd-l1, ensaio para identificar um indivíduo com uma doença, kit de diagnóstico, método para avaliar uma resposta ao tratamento e método para monitorar a resposta de um indivíduo tratado |
| HRP20181271T1 (hr) | 2013-09-06 | 2018-10-05 | Aurigene Discovery Technologies Limited | Ciklički peptidomimetički spojevi kao imunomodulatori |
| WO2015044900A1 (en) | 2013-09-27 | 2015-04-02 | Aurigene Discovery Technologies Limited | Therapeutic immunomodulating compounds |
| WO2016039749A1 (en) | 2014-09-11 | 2016-03-17 | Bristol-Myers Squibb Company | Macrocyclic inhibitors of the pd-1/pd-l1 and cd80 (b7-1)/pd-li protein/protein interactions |
| US9732119B2 (en) | 2014-10-10 | 2017-08-15 | Bristol-Myers Squibb Company | Immunomodulators |
| US9856292B2 (en) | 2014-11-14 | 2018-01-02 | Bristol-Myers Squibb Company | Immunomodulators |
| US9944678B2 (en) | 2014-12-19 | 2018-04-17 | Bristol-Myers Squibb Company | Immunomodulators |
| US20160222060A1 (en) | 2015-02-04 | 2016-08-04 | Bristol-Myers Squibb Company | Immunomodulators |
| US9809625B2 (en) | 2015-03-18 | 2017-11-07 | Bristol-Myers Squibb Company | Immunomodulators |
| US10358463B2 (en) * | 2016-04-05 | 2019-07-23 | Bristol-Myers Squibb Company | Immunomodulators |
-
2015
- 2015-12-14 US US14/967,960 patent/US9861680B2/en active Active
- 2015-12-15 EP EP15820747.2A patent/EP3233888B1/en active Active
- 2015-12-15 WO PCT/US2015/065723 patent/WO2016100285A1/en not_active Ceased
- 2015-12-15 EA EA201791231A patent/EA033894B1/ru not_active IP Right Cessation
- 2015-12-15 ES ES15820747T patent/ES2940632T3/es active Active
- 2015-12-15 JP JP2017532682A patent/JP6625129B2/ja active Active
- 2015-12-15 KR KR1020177019417A patent/KR102602643B1/ko active Active
- 2015-12-15 AU AU2015362703A patent/AU2015362703A1/en not_active Abandoned
- 2015-12-15 MX MX2017007677A patent/MX2017007677A/es unknown
- 2015-12-15 CN CN201580069483.3A patent/CN107108697B/zh active Active
- 2015-12-15 CA CA2971189A patent/CA2971189A1/en not_active Abandoned
- 2015-12-15 SG SG11201704823TA patent/SG11201704823TA/en unknown
- 2015-12-15 BR BR112017012679A patent/BR112017012679A2/pt not_active Application Discontinuation
- 2015-12-17 TW TW104142534A patent/TW201629086A/zh unknown
- 2015-12-17 AR ARP150104168A patent/AR103093A1/es unknown
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2017
- 2017-06-12 IL IL252853A patent/IL252853A0/en unknown
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