JP2018501287A5 - - Google Patents

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Publication number
JP2018501287A5
JP2018501287A5 JP2017536301A JP2017536301A JP2018501287A5 JP 2018501287 A5 JP2018501287 A5 JP 2018501287A5 JP 2017536301 A JP2017536301 A JP 2017536301A JP 2017536301 A JP2017536301 A JP 2017536301A JP 2018501287 A5 JP2018501287 A5 JP 2018501287A5
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JP
Japan
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JP2017536301A
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English (en)
Japanese (ja)
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JP6659703B2 (ja
JP2018501287A (ja
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Priority claimed from PCT/US2016/012659 external-priority patent/WO2016112298A1/en
Publication of JP2018501287A publication Critical patent/JP2018501287A/ja
Publication of JP2018501287A5 publication Critical patent/JP2018501287A5/ja
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Publication of JP6659703B2 publication Critical patent/JP6659703B2/ja
Expired - Fee Related legal-status Critical Current
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JP2017536301A 2015-01-09 2016-01-08 ピリダジノン誘導体および癌の処置におけるそれらの使用 Expired - Fee Related JP6659703B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562101953P 2015-01-09 2015-01-09
US62/101,953 2015-01-09
PCT/US2016/012659 WO2016112298A1 (en) 2015-01-09 2016-01-08 Pyridazinone derivatives and their use in the treatment of cancer

Publications (3)

Publication Number Publication Date
JP2018501287A JP2018501287A (ja) 2018-01-18
JP2018501287A5 true JP2018501287A5 (https=) 2019-01-31
JP6659703B2 JP6659703B2 (ja) 2020-03-04

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ID=55299747

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2017536301A Expired - Fee Related JP6659703B2 (ja) 2015-01-09 2016-01-08 ピリダジノン誘導体および癌の処置におけるそれらの使用

Country Status (5)

Country Link
US (1) US10239861B2 (https=)
EP (1) EP3242874B1 (https=)
JP (1) JP6659703B2 (https=)
CN (1) CN107406429B (https=)
WO (1) WO2016112298A1 (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3189046B1 (en) 2014-09-05 2020-08-26 Genentech, Inc. Therapeutic compounds and uses thereof
EP3189049B1 (en) 2014-09-05 2024-03-20 Genentech, Inc. Phthalazine derivatives of formula (i) as pcaf and gcn5 inhibitors for use in the treatment of cancer
KR102194536B1 (ko) * 2019-06-10 2020-12-23 연세대학교 산학협력단 타목시펜의 반응성 예측용 조성물
CN112824381B (zh) * 2019-11-21 2024-04-26 广东东阳光药业股份有限公司 一种哌啶胺的制备方法
IL298760A (en) 2020-06-05 2023-02-01 Kinnate Biopharma Inc Fibroblast growth factor receptor kinase inhibitors
US20230391730A1 (en) * 2020-10-09 2023-12-07 Regents Of The University Of Minnesota Inhibitors of the bromodomain phd finger transcription factor (bptf) as anti-cancer agents
KR102766287B1 (ko) * 2021-10-15 2025-02-12 고려대학교 산학협력단 피리다벤을 포함하는 자궁내막 세포, 영양막 세포 또는 고환 세포의 비정상적 증식 관련 질환의 예방 또는 치료용 약학적 조성물
WO2024050078A1 (en) 2022-09-02 2024-03-07 Auron Therapeutics, Inc. Pyridazinon derivatives as kat2 degraders for the treatment of proliferative disorders

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EP3189049B1 (en) 2014-09-05 2024-03-20 Genentech, Inc. Phthalazine derivatives of formula (i) as pcaf and gcn5 inhibitors for use in the treatment of cancer

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