JP2017538692A5 - - Google Patents

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Publication number
JP2017538692A5
JP2017538692A5 JP2017528156A JP2017528156A JP2017538692A5 JP 2017538692 A5 JP2017538692 A5 JP 2017538692A5 JP 2017528156 A JP2017528156 A JP 2017528156A JP 2017528156 A JP2017528156 A JP 2017528156A JP 2017538692 A5 JP2017538692 A5 JP 2017538692A5
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JP
Japan
Prior art keywords
group
nitrogen
alkyl
carbon
optionally substituted
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JP2017528156A
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English (en)
Japanese (ja)
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JP7349773B2 (ja
JP2017538692A (ja
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Priority claimed from GBGB1421020.7A external-priority patent/GB201421020D0/en
Priority claimed from GBGB1516059.1A external-priority patent/GB201516059D0/en
Application filed filed Critical
Priority claimed from PCT/EP2015/077821 external-priority patent/WO2016083531A1/en
Publication of JP2017538692A publication Critical patent/JP2017538692A/ja
Publication of JP2017538692A5 publication Critical patent/JP2017538692A5/ja
Application granted granted Critical
Publication of JP7349773B2 publication Critical patent/JP7349773B2/ja
Active legal-status Critical Current
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JP2017528156A 2014-11-26 2015-11-26 化合物 Active JP7349773B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB1421020.7 2014-11-26
GBGB1421020.7A GB201421020D0 (en) 2014-11-26 2014-11-26 Compounds
GB1516059.1 2015-09-10
GBGB1516059.1A GB201516059D0 (en) 2015-09-10 2015-09-10 Compounds
PCT/EP2015/077821 WO2016083531A1 (en) 2014-11-26 2015-11-26 Compounds

Publications (3)

Publication Number Publication Date
JP2017538692A JP2017538692A (ja) 2017-12-28
JP2017538692A5 true JP2017538692A5 (enExample) 2019-01-17
JP7349773B2 JP7349773B2 (ja) 2023-09-25

Family

ID=54705181

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2017528156A Active JP7349773B2 (ja) 2014-11-26 2015-11-26 化合物

Country Status (8)

Country Link
US (2) US12146004B2 (enExample)
EP (1) EP3224273A1 (enExample)
JP (1) JP7349773B2 (enExample)
CN (1) CN107108699A (enExample)
AU (1) AU2015352440B2 (enExample)
CA (1) CA2968902C (enExample)
TW (1) TWI757229B (enExample)
WO (1) WO2016083531A1 (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3224273A1 (en) * 2014-11-26 2017-10-04 New Pharma Licence Holdings Limited Compounds
WO2018006063A1 (en) * 2016-07-01 2018-01-04 Cidara Therapeutics, Inc. Compositions and methods for the treatment of bacterial infections
AU2017376711B2 (en) * 2016-12-16 2020-07-16 Institute Of Medicinal Biotechnology, Chinese Academy Of Medical Sciences Polymyxin derivative, preparation method and application thereof
US11279733B2 (en) 2017-11-02 2022-03-22 The University Of Queensland Peptide antibiotics
PL3810633T3 (pl) * 2018-06-25 2024-04-08 Spero Therapeutics, Inc. Związki
CN111690040A (zh) * 2019-03-12 2020-09-22 上海来益生物药物研究开发中心有限责任公司 多粘菌素衍生物、其制备方法和应用
WO2021150792A1 (en) 2020-01-21 2021-07-29 Micurx Pharmaceuticals, Inc. Novel compounds and composition for targeted therapy of kidney-associated cancers
CN111559992B (zh) * 2020-05-29 2022-04-08 华中科技大学 一种2-芳基-γ-氨基丁酸衍生物的制备方法
TW202233649A (zh) 2020-11-06 2022-09-01 美商斯佩羅治療學股份有限公司 化合物
WO2022206826A1 (zh) * 2021-03-31 2022-10-06 江苏奥赛康药业有限公司 一种多粘菌素衍生物的硫酸盐及其药物组合物

Family Cites Families (27)

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Publication number Priority date Publication date Assignee Title
GB2128617A (en) 1982-10-06 1984-05-02 Martti Vaara Polypeptides for use in antibacterial therapy
AU7753787A (en) 1986-08-06 1988-02-24 Jean-Luc Fauchere Production of covalent-linked conjugates from an antibiotic and a non-toxic derivative of polymyxine b
US20010021697A1 (en) 1987-09-14 2001-09-13 Henning Lowenstein Methods and compositions for the treatment of mammalian infections employing medicaments comprising hymenoptera venom, proteinageous or polypeptide components thereof, or analogues of such proteinaceous or polypeptide components
TW274552B (enExample) 1992-05-26 1996-04-21 Hoechst Ag
US5767068A (en) 1997-02-13 1998-06-16 Pathogenesis Corporation Pure biologically active colistin, its components and a colistin formulation for treatment of pulmonary infections
CA2540742A1 (en) 2003-09-30 2005-04-14 Terry Hicks Compositions and methods for treating burns
US20060004185A1 (en) 2004-07-01 2006-01-05 Leese Richard A Peptide antibiotics and peptide intermediates for their prepartion
CN103059106B (zh) 2006-08-11 2015-01-14 北方抗生素有限公司 多粘菌素衍生物及其用途
US7807637B2 (en) * 2006-08-11 2010-10-05 Northern Antibiotics Oy Polymyxin derivatives and uses thereof
US8329645B2 (en) 2008-02-08 2012-12-11 Northern Antibiotics Ltd. Polymyxin derivatives and uses thereof
FI20085469A0 (fi) 2008-02-08 2008-05-16 Northern Antibiotics Oy Polymyksiinijohdannaiset, joissa on lyhyt rasvahappohäntä, ja niiden käyttöjä
US8193148B2 (en) 2008-02-08 2012-06-05 Northern Antibiotics Ltd. Short fatty acid tail polymyxin derivatives and uses thereof
ES2334547B1 (es) 2008-09-10 2010-12-03 Universidad De Barcelona Compuestos peptidicos antibacterianos.
US8343912B2 (en) 2008-12-23 2013-01-01 Biosource Pharm, Inc. Antibiotic compositions for the treatment of gram negative infections
CN101851270A (zh) 2009-04-03 2010-10-06 梁浩 一种多粘菌素衍生物及其制备方法
WO2010130007A1 (en) * 2009-05-14 2010-11-18 Monash University Antimicrobial compounds
US8415307B1 (en) 2010-06-23 2013-04-09 Biosource Pharm, Inc. Antibiotic compositions for the treatment of gram negative infections
WO2012051663A1 (en) * 2010-10-21 2012-04-26 Monash University Antimicrobial compounds
WO2012168820A1 (en) * 2011-06-08 2012-12-13 Pfizer Inc. Polymyxin derivatives useful as antibacterial agents
WO2013072695A1 (en) * 2011-11-18 2013-05-23 Novacta Biosystems Limited Polymyxin derivatives
PL2999711T3 (pl) 2013-05-22 2022-09-26 Spero Therapeutics, Inc. Pochodne polimyksyny i ich zastosowanie w terapii skojarzonej razem z różnymi antybiotykami
LT3116897T (lt) 2014-03-11 2022-05-10 Spero Therapeutics, Inc. Polimiksino dariniai ir jų panaudojimas kompleksinėje terapijoje kartu su skirtingais antibiotikais
US10047126B2 (en) 2014-04-01 2018-08-14 Monash University Polymyxin derivatives as antimicrobial compounds
EP3224273A1 (en) * 2014-11-26 2017-10-04 New Pharma Licence Holdings Limited Compounds
WO2016166103A1 (en) 2015-04-13 2016-10-20 Xellia Pharmaceuticals Aps Polymyxin derivatives
AU2016331658B2 (en) 2015-09-29 2021-04-01 Monash University Antimicrobial polymyxin derivative compounds
PL3810633T3 (pl) 2018-06-25 2024-04-08 Spero Therapeutics, Inc. Związki

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