JP2017534675A5 - - Google Patents

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Publication number
JP2017534675A5
JP2017534675A5 JP2017536216A JP2017536216A JP2017534675A5 JP 2017534675 A5 JP2017534675 A5 JP 2017534675A5 JP 2017536216 A JP2017536216 A JP 2017536216A JP 2017536216 A JP2017536216 A JP 2017536216A JP 2017534675 A5 JP2017534675 A5 JP 2017534675A5
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JP
Japan
Prior art keywords
alkyl
group
glycine
acid
prodrug according
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Application number
JP2017536216A
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English (en)
Japanese (ja)
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JP2017534675A (ja
JP6701208B2 (ja
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Priority claimed from PCT/US2015/051705 external-priority patent/WO2016049174A1/en
Publication of JP2017534675A publication Critical patent/JP2017534675A/ja
Publication of JP2017534675A5 publication Critical patent/JP2017534675A5/ja
Application granted granted Critical
Publication of JP6701208B2 publication Critical patent/JP6701208B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2017536216A 2014-09-24 2015-09-23 脂質化アミド系インスリンプロドラッグ Expired - Fee Related JP6701208B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201462054670P 2014-09-24 2014-09-24
US62/054,670 2014-09-24
PCT/US2015/051705 WO2016049174A1 (en) 2014-09-24 2015-09-23 Lipidated amide-based insulin prodrugs

Publications (3)

Publication Number Publication Date
JP2017534675A JP2017534675A (ja) 2017-11-24
JP2017534675A5 true JP2017534675A5 (enExample) 2018-10-25
JP6701208B2 JP6701208B2 (ja) 2020-05-27

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ID=55581947

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2017536216A Expired - Fee Related JP6701208B2 (ja) 2014-09-24 2015-09-23 脂質化アミド系インスリンプロドラッグ

Country Status (6)

Country Link
US (1) US10385107B2 (enExample)
EP (1) EP3197912B1 (enExample)
JP (1) JP6701208B2 (enExample)
CN (1) CN107001441A (enExample)
ES (1) ES2947409T3 (enExample)
WO (1) WO2016049174A1 (enExample)

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AU2021312323A1 (en) 2020-07-22 2023-02-02 Novo Nordisk A/S Co-agonists at GLP-1 and GIP receptors suitable for oral delivery
CA3199254A1 (en) * 2020-10-22 2022-04-28 The Trustees Of Indiana University Molecular designs of glucose-responsive and glucose-cleavable insulin analogues
JP7484018B2 (ja) 2020-11-06 2024-05-15 ノヴォ ノルディスク アー/エス Glp-1プロドラッグおよびその使用
WO2023012263A1 (en) 2021-08-04 2023-02-09 Novo Nordisk A/S Solid oral peptide formulations
TW202330584A (zh) 2022-01-20 2023-08-01 丹麥商諾佛 儂迪克股份有限公司 前藥及其用途
US20250304645A1 (en) 2022-05-10 2025-10-02 Novo Nordisk A/S Prodrugs of GLP-1 Polypeptide and Uses Thereof
TW202421645A (zh) 2022-11-25 2024-06-01 丹麥商諾佛 儂迪克股份有限公司 如glp—1之肽治療劑的口服投與
WO2026139053A1 (zh) * 2024-12-27 2026-07-02 深圳信立泰药业股份有限公司 一种包含glp-1化合物的药物组合物及其制备方法与应用

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