JP2017526662A5 - - Google Patents

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Publication number
JP2017526662A5
JP2017526662A5 JP2017506390A JP2017506390A JP2017526662A5 JP 2017526662 A5 JP2017526662 A5 JP 2017526662A5 JP 2017506390 A JP2017506390 A JP 2017506390A JP 2017506390 A JP2017506390 A JP 2017506390A JP 2017526662 A5 JP2017526662 A5 JP 2017526662A5
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JP
Japan
Prior art keywords
cancer
composition
compound
pharmaceutically acceptable
combination
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JP2017506390A
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English (en)
Japanese (ja)
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JP6892381B2 (ja
JP2017526662A (ja
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Priority claimed from PCT/US2015/043825 external-priority patent/WO2016022697A1/en
Publication of JP2017526662A publication Critical patent/JP2017526662A/ja
Publication of JP2017526662A5 publication Critical patent/JP2017526662A5/ja
Application granted granted Critical
Publication of JP6892381B2 publication Critical patent/JP6892381B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2017506390A 2014-08-05 2015-08-05 多発性骨髄腫を治療するための薬物の組み合わせ Expired - Fee Related JP6892381B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201462033386P 2014-08-05 2014-08-05
US62/033,386 2014-08-05
PCT/US2015/043825 WO2016022697A1 (en) 2014-08-05 2015-08-05 Drug combinations to treat multiple myeloma

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2019186703A Division JP2020002179A (ja) 2014-08-05 2019-10-10 多発性骨髄腫を治療するための薬物の組み合わせ

Publications (3)

Publication Number Publication Date
JP2017526662A JP2017526662A (ja) 2017-09-14
JP2017526662A5 true JP2017526662A5 (enExample) 2018-09-06
JP6892381B2 JP6892381B2 (ja) 2021-06-23

Family

ID=53836256

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2017506390A Expired - Fee Related JP6892381B2 (ja) 2014-08-05 2015-08-05 多発性骨髄腫を治療するための薬物の組み合わせ
JP2019186703A Pending JP2020002179A (ja) 2014-08-05 2019-10-10 多発性骨髄腫を治療するための薬物の組み合わせ

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2019186703A Pending JP2020002179A (ja) 2014-08-05 2019-10-10 多発性骨髄腫を治療するための薬物の組み合わせ

Country Status (13)

Country Link
US (1) US11065240B2 (enExample)
EP (1) EP3177311B1 (enExample)
JP (2) JP6892381B2 (enExample)
KR (1) KR102634247B1 (enExample)
CN (1) CN106573042A (enExample)
AU (1) AU2015301097B2 (enExample)
BR (1) BR112017002318A2 (enExample)
CA (1) CA2957466C (enExample)
EA (1) EA034992B1 (enExample)
MA (1) MA40457A (enExample)
MX (1) MX382904B (enExample)
UA (1) UA121482C2 (enExample)
WO (1) WO2016022697A1 (enExample)

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WO2015142928A1 (en) 2014-03-17 2015-09-24 Exelixis, Inc. Dosing of cabozantinib formulations
MA40386A (fr) 2014-07-31 2016-02-04 Exelixis Inc Procédé de préparation de cabozantinib marqué au fluor-18 et d'analogues de celui-ci
EA034992B1 (ru) 2014-08-05 2020-04-15 Экселиксис, Инк. Комбинации лекарственных средств для лечения множественной миеломы
EP3442531A1 (en) 2016-04-15 2019-02-20 Exelixis, Inc. Method of treating renal cell carcinoma using n-(4-(6,7-dimethoxyquinolin-4-yloxy) phenyl)-n'-(4-fluoropheny)cyclopropane-1,1-dicarboxamide, (2s)-hydroxybutanedioate
CN111108125A (zh) * 2017-09-14 2020-05-05 葛兰素史密斯克莱知识产权发展有限公司 用于癌症的组合治疗
MY210421A (en) 2018-01-26 2025-09-22 Exelixis Inc Compounds for the treatment of kinase-dependent disorders
AU2019285066B2 (en) 2018-06-15 2024-06-13 Handa Pharmaceuticals, Inc. Kinase inhibitor salts and compositions thereof
WO2023222946A1 (en) 2022-05-18 2023-11-23 Fermion Oy Process for the preparation of cabozantinib
EP4658271A1 (en) 2023-01-31 2025-12-10 Handa Oncology, LLC Improved cabozantinib compositions and methods of use

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CA2603748A1 (en) 2005-04-06 2006-10-12 Exelixis, Inc. C-met modulators and methods of use
JP5311673B2 (ja) 2006-12-14 2013-10-09 エグゼリクシス, インコーポレイテッド Mek阻害剤の使用方法
UY31800A (es) 2008-05-05 2009-11-10 Smithkline Beckman Corp Metodo de tratamiento de cancer usando un inhibidor de cmet y axl y un inhibidor de erbb
AR075084A1 (es) 2008-09-26 2011-03-09 Smithkline Beecham Corp Metodo de preparacion de quinolinil -oxidifenil - ciclopropanodicarboxamidas e intermediarios correspondientes
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UA108618C2 (uk) 2009-08-07 2015-05-25 Застосування c-met-модуляторів в комбінації з темозоломідом та/або променевою терапією для лікування раку
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EA034992B1 (ru) 2014-08-05 2020-04-15 Экселиксис, Инк. Комбинации лекарственных средств для лечения множественной миеломы
US20170224670A1 (en) 2014-10-14 2017-08-10 Exelixis, Inc. Drug Combination to Treat Melanoma

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