JP2015532289A5 - - Google Patents

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Publication number
JP2015532289A5
JP2015532289A5 JP2015534772A JP2015534772A JP2015532289A5 JP 2015532289 A5 JP2015532289 A5 JP 2015532289A5 JP 2015534772 A JP2015534772 A JP 2015534772A JP 2015534772 A JP2015534772 A JP 2015534772A JP 2015532289 A5 JP2015532289 A5 JP 2015532289A5
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JP
Japan
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aliphatic
independently
cor
independently selected
optionally
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JP2015534772A
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English (en)
Japanese (ja)
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JP2015532289A (ja
JP6523958B2 (ja
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Priority claimed from PCT/US2013/062413 external-priority patent/WO2014052896A1/en
Publication of JP2015532289A publication Critical patent/JP2015532289A/ja
Publication of JP2015532289A5 publication Critical patent/JP2015532289A5/ja
Priority to JP2019004203A priority Critical patent/JP6913698B2/ja
Application granted granted Critical
Publication of JP6523958B2 publication Critical patent/JP6523958B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2015534772A 2012-09-28 2013-09-27 ウリジン二リン酸誘導体、プロドラッグ、組成物およびそれらの使用 Expired - Fee Related JP6523958B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2019004203A JP6913698B2 (ja) 2012-09-28 2019-01-15 ウリジン二リン酸誘導体、プロドラッグ、組成物およびそれらの使用

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201261707568P 2012-09-28 2012-09-28
US61/707,568 2012-09-28
US201361780171P 2013-03-13 2013-03-13
US61/780,171 2013-03-13
PCT/US2013/062413 WO2014052896A1 (en) 2012-09-28 2013-09-27 Uridine diphosphate derivatives, prodrugs, compositions and uses thereof

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2019004203A Division JP6913698B2 (ja) 2012-09-28 2019-01-15 ウリジン二リン酸誘導体、プロドラッグ、組成物およびそれらの使用

Publications (3)

Publication Number Publication Date
JP2015532289A JP2015532289A (ja) 2015-11-09
JP2015532289A5 true JP2015532289A5 (enExample) 2016-10-20
JP6523958B2 JP6523958B2 (ja) 2019-06-05

Family

ID=50389029

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2015534772A Expired - Fee Related JP6523958B2 (ja) 2012-09-28 2013-09-27 ウリジン二リン酸誘導体、プロドラッグ、組成物およびそれらの使用
JP2019004203A Expired - Fee Related JP6913698B2 (ja) 2012-09-28 2019-01-15 ウリジン二リン酸誘導体、プロドラッグ、組成物およびそれらの使用

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2019004203A Expired - Fee Related JP6913698B2 (ja) 2012-09-28 2019-01-15 ウリジン二リン酸誘導体、プロドラッグ、組成物およびそれらの使用

Country Status (6)

Country Link
US (6) US9163055B2 (enExample)
EP (1) EP2900680A4 (enExample)
JP (2) JP6523958B2 (enExample)
AU (2) AU2013323188B2 (enExample)
CA (1) CA2885369A1 (enExample)
WO (1) WO2014052896A1 (enExample)

Families Citing this family (13)

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Publication number Priority date Publication date Assignee Title
CN103906745B (zh) * 2011-09-30 2017-08-25 塔夫斯大学 用于治疗神经变性疾病的尿苷二磷酸衍生物、组合物和方法
JP6523958B2 (ja) 2012-09-28 2019-06-05 タフツ・ユニバーシティ ウリジン二リン酸誘導体、プロドラッグ、組成物およびそれらの使用
HUE039871T2 (hu) 2013-03-13 2019-02-28 Univ Tufts Uridin nukleozid származékok, kompozíciók és alkalmazási eljárások
US10138265B2 (en) 2013-03-13 2018-11-27 Tufts University Uridine nucleoside derivatives, compositions and methods of use
EP3623364A1 (en) * 2014-02-13 2020-03-18 Ligand Pharmaceuticals, Inc. Prodrug compounds and their uses
EP3286172B1 (en) 2015-04-23 2019-06-12 Constellation Pharmaceuticals, Inc. Lsd1 inhibitors and uses thereof
WO2018058148A1 (en) 2016-09-26 2018-03-29 Tufts University Uridine nucleoside derivatives, compositions and methods of use
HUE063848T2 (hu) 2016-10-26 2024-02-28 Constellation Pharmaceuticals Inc LSD1 gátlók és gyógyászati alkalmazásaik
WO2018236221A2 (en) * 2017-06-03 2018-12-27 Can Holding B.V. Neurodegenerative peptide deposit dissolution
KR102010558B1 (ko) * 2017-12-08 2019-08-13 윤주석 금속 미네랄 디아미네이트 및 이의 제조방법
WO2019112383A1 (ko) * 2017-12-08 2019-06-13 윤주석 금속 미네랄 디아미네이트 및 이의 제조방법
US20210169911A1 (en) * 2018-08-17 2021-06-10 The United States Of America,As Represented By The Secretary,Department Of Health And Human Services Purine and pyrimidine nucleotides as ecto-5'-nucleotidase inhibitors
CN117700468B (zh) * 2024-02-05 2024-05-03 深圳赛陆医疗科技有限公司 一种核苷酸类似物的制备方法

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Publication number Priority date Publication date Assignee Title
JPH0621073B2 (ja) 1986-03-06 1994-03-23 日水製薬株式会社 中枢抑制剤
JP3032053B2 (ja) 1991-09-06 2000-04-10 日水製薬株式会社 ウリジン誘導体及びこれを含有する医薬
ATE185070T1 (de) * 1992-05-22 1999-10-15 Senju Pharma Co Arzneimittel gegen glaukom
US5962459A (en) 1996-05-28 1999-10-05 Polifarma S.P.A. Therapeutic active agent for treatment of neuron degenerative diseases
WO1999009998A1 (en) 1997-08-29 1999-03-04 The University Of North Carolina At Chapel Hill Use of uridine 5'-diphosphate and analogs thereof for the treatment of lung diseases
US8314064B2 (en) 1998-07-31 2012-11-20 Massachusetts Institute Of Technology Uridine administration stimulates membrane production
ATE446097T1 (de) 1998-07-31 2009-11-15 Massachusetts Inst Technology Verwendung von uridin in kombination mit cholin zur behandlung von gedächtnisstörungen
US20070004670A1 (en) 1998-07-31 2007-01-04 Richard Wurtman Compositions containing citicoline, and methods of use thereof
US20050203053A1 (en) 1999-07-30 2005-09-15 Wurtman Richard J. Uridine administration improves phosphatide synthesis, synaptic transmission and cogntive function
US8518882B2 (en) 1998-07-31 2013-08-27 Massachusetts Institute Of Technology Methods and compositions for ameliorating or inhibiting decline in memory or intelligence or improving same
US8143234B2 (en) 1998-07-31 2012-03-27 Massachusetts Institute Of Technology Uridine administration improves phosphatide synthesis, synaptic transmission and cognitive function
US20060069061A1 (en) 1998-07-31 2006-03-30 Dick Wurtman Compositions containing uridine and choline, and methods utilizing same
GB0004297D0 (en) 2000-02-23 2000-04-12 Ucb Sa 2-oxo-1 pyrrolidine derivatives process for preparing them and their uses
US6875751B2 (en) 2000-06-15 2005-04-05 Idenix Pharmaceuticals, Inc. 3′-prodrugs of 2′-deoxy-β-L-nucleosides
CA2444161A1 (en) 2003-10-01 2005-04-01 Japan Health Sciences Foundation A screening method of drug for treatment of neuropathic pain
EP1765075A4 (en) 2004-06-10 2010-11-10 Mclean Hospital Corp PYRIMIDINES, AS FORM. uridine; IN THE TREATMENT OF PATIENTS WITH MANIC-DEPRESSIVE PSYCHOSIS
US7851456B2 (en) 2005-06-29 2010-12-14 Inspire Pharmaceuticals, Inc. P2Y6 receptor agonists for treating lung diseases
US8618074B2 (en) * 2007-03-15 2013-12-31 Board Of Regents Of The University Of Texas System GPCR enhanced neuroprotection to treat brain injury
WO2008115499A1 (en) 2007-03-19 2008-09-25 State Of Oregon Acting By And Through The Oregon State Board Of Higher Education On Behalf Of The University Of Oregon Mannich base n-oxide drugs
US7964580B2 (en) 2007-03-30 2011-06-21 Pharmasset, Inc. Nucleoside phosphoramidate prodrugs
US8962580B2 (en) * 2008-09-23 2015-02-24 Alnylam Pharmaceuticals, Inc. Chemical modifications of monomers and oligonucleotides with cycloaddition
IT1398378B1 (it) * 2010-02-22 2013-02-22 Omikron Italia S R L Citicolina per il trattamento del glaucoma e dell'ipertensione oculare.
CN103339136A (zh) 2010-12-01 2013-10-02 巴伊兰大学 尿苷二-或三-磷酸衍生物以及其用途
CN103906745B (zh) * 2011-09-30 2017-08-25 塔夫斯大学 用于治疗神经变性疾病的尿苷二磷酸衍生物、组合物和方法
JP6523958B2 (ja) 2012-09-28 2019-06-05 タフツ・ユニバーシティ ウリジン二リン酸誘導体、プロドラッグ、組成物およびそれらの使用
US10138265B2 (en) 2013-03-13 2018-11-27 Tufts University Uridine nucleoside derivatives, compositions and methods of use
HUE039871T2 (hu) 2013-03-13 2019-02-28 Univ Tufts Uridin nukleozid származékok, kompozíciók és alkalmazási eljárások

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