AU2013323188B2 - Uridine diphosphate derivatives, prodrugs, compositions and uses thereof - Google Patents

Uridine diphosphate derivatives, prodrugs, compositions and uses thereof Download PDF

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AU2013323188B2
AU2013323188B2 AU2013323188A AU2013323188A AU2013323188B2 AU 2013323188 B2 AU2013323188 B2 AU 2013323188B2 AU 2013323188 A AU2013323188 A AU 2013323188A AU 2013323188 A AU2013323188 A AU 2013323188A AU 2013323188 B2 AU2013323188 B2 AU 2013323188B2
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compound
independently selected
aliphatic
condition
inflammatory
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AU2013323188A1 (en
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Philip G. Haydon
Jinbo Lee
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Tufts University
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Tufts University
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    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7068—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
    • A61K31/7072—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid having two oxo groups directly attached to the pyrimidine ring, e.g. uridine, uridylic acid, thymidine, zidovudine
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    • C07F9/02—Phosphorus compounds
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    • C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
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AU2013323188A 2012-09-28 2013-09-27 Uridine diphosphate derivatives, prodrugs, compositions and uses thereof Ceased AU2013323188B2 (en)

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US201261707568P 2012-09-28 2012-09-28
US61/707,568 2012-09-28
US201361780171P 2013-03-13 2013-03-13
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PCT/US2013/062413 WO2014052896A1 (en) 2012-09-28 2013-09-27 Uridine diphosphate derivatives, prodrugs, compositions and uses thereof

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