JP2014518199A5 - - Google Patents

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JP2014518199A5
JP2014518199A5 JP2014513214A JP2014513214A JP2014518199A5 JP 2014518199 A5 JP2014518199 A5 JP 2014518199A5 JP 2014513214 A JP2014513214 A JP 2014513214A JP 2014513214 A JP2014513214 A JP 2014513214A JP 2014518199 A5 JP2014518199 A5 JP 2014518199A5
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formula
compound
group
alkyl
reacting
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JP2014513214A
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JP6425540B2 (ja
JP2014518199A (ja
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Priority claimed from PCT/EP2012/060447 external-priority patent/WO2012164096A1/en
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JP2014513214A 2011-06-01 2012-06-01 エステトロール中間体を製造するための方法 Active JP6425540B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201161492300P 2011-06-01 2011-06-01
EP11168561.6 2011-06-01
US61/492,300 2011-06-01
EP11168561 2011-06-01
PCT/EP2012/060447 WO2012164096A1 (en) 2011-06-01 2012-06-01 Process for the production of estetrol intermediates

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2017155801A Division JP6479912B2 (ja) 2011-06-01 2017-08-10 エステトロール中間体を製造するための方法

Publications (3)

Publication Number Publication Date
JP2014518199A JP2014518199A (ja) 2014-07-28
JP2014518199A5 true JP2014518199A5 (US07714131-20100511-C00001.png) 2016-02-12
JP6425540B2 JP6425540B2 (ja) 2018-11-21

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JP2014513214A Active JP6425540B2 (ja) 2011-06-01 2012-06-01 エステトロール中間体を製造するための方法
JP2017155801A Active JP6479912B2 (ja) 2011-06-01 2017-08-10 エステトロール中間体を製造するための方法

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JP2017155801A Active JP6479912B2 (ja) 2011-06-01 2017-08-10 エステトロール中間体を製造するための方法

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US (1) US11053274B2 (US07714131-20100511-C00001.png)
EP (1) EP2714710B1 (US07714131-20100511-C00001.png)
JP (2) JP6425540B2 (US07714131-20100511-C00001.png)
KR (1) KR101994805B1 (US07714131-20100511-C00001.png)
CN (2) CN107266514A (US07714131-20100511-C00001.png)
AU (1) AU2012264602B2 (US07714131-20100511-C00001.png)
BR (1) BR112013030830B1 (US07714131-20100511-C00001.png)
CA (1) CA2835981C (US07714131-20100511-C00001.png)
CY (1) CY1118150T1 (US07714131-20100511-C00001.png)
DK (1) DK2714710T3 (US07714131-20100511-C00001.png)
EA (1) EA023991B1 (US07714131-20100511-C00001.png)
ES (1) ES2579175T3 (US07714131-20100511-C00001.png)
HR (1) HRP20160692T2 (US07714131-20100511-C00001.png)
HU (1) HUE029252T2 (US07714131-20100511-C00001.png)
ME (1) ME02454B (US07714131-20100511-C00001.png)
MX (1) MX341561B (US07714131-20100511-C00001.png)
PL (1) PL2714710T3 (US07714131-20100511-C00001.png)
PT (1) PT2714710T (US07714131-20100511-C00001.png)
RS (1) RS54880B1 (US07714131-20100511-C00001.png)
SG (1) SG195118A1 (US07714131-20100511-C00001.png)
SI (1) SI2714710T1 (US07714131-20100511-C00001.png)
SM (1) SMT201600206B (US07714131-20100511-C00001.png)
WO (1) WO2012164096A1 (US07714131-20100511-C00001.png)
ZA (1) ZA201308446B (US07714131-20100511-C00001.png)

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CN107266514A (zh) 2011-06-01 2017-10-20 埃斯特拉私人有限责任公司 用于产生雌四醇中间体的方法
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EP2383279A1 (en) 2011-07-19 2011-11-02 Pantarhei Bioscience B.V. Process for the preparation of estetrol
US8987484B2 (en) 2011-10-07 2015-03-24 Estetra S.P.R.L. Process for the production of estetrol
EA035687B1 (ru) 2015-06-18 2020-07-27 Эстетра Спрл Диспергируемая в полости рта единица дозирования, содержащая эстетрольный компонент
DK3310345T3 (da) 2015-06-18 2021-05-25 Estetra Sprl Orodispersibel tablet indeholdende estetrol
EP3310346B1 (en) 2015-06-18 2021-03-24 Estetra SPRL Orodispersible tablet containing estetrol
UA123098C2 (uk) 2015-06-18 2021-02-17 Естетра Спрл Диспергована у порожнині рота одиниця дозування, що містить естетрольний компонент
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JOP20200260A1 (ar) 2018-04-19 2019-10-19 Estetra Sprl مركبات واستخداماتها للتخفيف من الأعراض المصاحبة لانقطاع الطمث
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IT201900017414A1 (it) 2019-09-27 2021-03-27 Ind Chimica Srl Processo per la preparazione di (15α,16α,17β)-estra-1,3,5(10)-triene-3,15,16,17-tetrolo (Estetrolo) ed intermedi di detto processo
FR3101348B1 (fr) 2019-09-27 2024-01-19 Ind Chimica Srl PROCÉDÉ DE PRÉPARATION DE (15α,16α,17β)-OESTRA-1,3,5(10)-TRIÈNE-3,15,16,17-TÉTROL (OESTÉTROL) ET INTERMÉDIAIRES DUDIT PROCÉDÉ
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GB2626482A (en) 2021-10-01 2024-07-24 Ind Chimica Srl Process for preparing (15alpha,16alpha,17eta)-estra-1,3,5-(10)-triene-3,15,16,17-tetrol(estetrol) monohydrate
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EP3310346B1 (en) 2015-06-18 2021-03-24 Estetra SPRL Orodispersible tablet containing estetrol
EA035687B1 (ru) 2015-06-18 2020-07-27 Эстетра Спрл Диспергируемая в полости рта единица дозирования, содержащая эстетрольный компонент
DK3310345T3 (da) 2015-06-18 2021-05-25 Estetra Sprl Orodispersibel tablet indeholdende estetrol

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