JP2014506230A5 - - Google Patents

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Publication number
JP2014506230A5
JP2014506230A5 JP2013528778A JP2013528778A JP2014506230A5 JP 2014506230 A5 JP2014506230 A5 JP 2014506230A5 JP 2013528778 A JP2013528778 A JP 2013528778A JP 2013528778 A JP2013528778 A JP 2013528778A JP 2014506230 A5 JP2014506230 A5 JP 2014506230A5
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JP
Japan
Prior art keywords
compound
general formula
formula
range
gastric
Prior art date
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Application number
JP2013528778A
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English (en)
Japanese (ja)
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JP5868980B2 (ja
JP2014506230A (ja
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Application filed filed Critical
Priority claimed from PCT/IB2011/002129 external-priority patent/WO2012035406A1/en
Publication of JP2014506230A publication Critical patent/JP2014506230A/ja
Publication of JP2014506230A5 publication Critical patent/JP2014506230A5/ja
Application granted granted Critical
Publication of JP5868980B2 publication Critical patent/JP5868980B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2013528778A 2010-09-14 2011-09-14 トリプタミン誘導体、その製造方法および胃疾患についての使用 Expired - Fee Related JP5868980B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN2173/DEL/2010 2010-09-14
IN2173DE2010 2010-09-14
PCT/IB2011/002129 WO2012035406A1 (en) 2010-09-14 2011-09-14 Tryptamine derivatives, their preparation and their use in gastropathy

Publications (3)

Publication Number Publication Date
JP2014506230A JP2014506230A (ja) 2014-03-13
JP2014506230A5 true JP2014506230A5 (enExample) 2014-05-22
JP5868980B2 JP5868980B2 (ja) 2016-02-24

Family

ID=44898070

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013528778A Expired - Fee Related JP5868980B2 (ja) 2010-09-14 2011-09-14 トリプタミン誘導体、その製造方法および胃疾患についての使用

Country Status (4)

Country Link
US (1) US8901317B2 (enExample)
EP (1) EP2616439B1 (enExample)
JP (1) JP5868980B2 (enExample)
WO (1) WO2012035406A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102439852B1 (ko) * 2015-04-17 2022-09-05 가천대학교 산학협력단 2-아미노퀴놀린-8-올 유도체, 및 이의 용도
US20190083462A1 (en) * 2016-03-18 2019-03-21 The Texas A&M University System Prevention of nsaid enteropathy with microbiota-derived tryptophan-metabolite
CA3176091C (en) 2020-12-31 2023-07-25 1280225 B.C. Ltd. Method of synthesizing indole compounds
CN113880749B (zh) * 2021-10-11 2023-06-30 江南大学 化合物JNc-463的制备方法及其应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3202669A (en) * 1963-11-06 1965-08-24 Upjohn Co 6-methoxy-1-(3, 4, 5-trimethoxy phenyl)-9h-pyrido [3, 4-b] indole and its acid addition salts
ES2083390T3 (es) * 1988-02-25 1996-04-16 I F L O S A S Di Giorgio E Ald Procedimiento de sintesis total para preparar una clase de producto derivado de estructura indol, del tipo triptamina, en particular la melatonia o la n-acetil-5-metoxitriptamina, con un elevado grado de pureza y facilmente soluble, para uso terapeutico contra los sindromes de la
AU1928892A (en) * 1991-06-21 1993-01-25 Smithkline Beecham Plc Tryptamine analogues, their synthesis and their use as 5-ht1-like or 5-ht2 receptor agonists
US6403808B1 (en) * 1999-12-10 2002-06-11 Virginia Commonwealth University Selective 5-HT6 receptor ligands
JP4156825B2 (ja) * 2001-11-01 2008-09-24 株式会社ロッテ 抗鬱・抗ストレス剤及びそれを含有する組成物
WO2004056769A2 (en) * 2002-12-20 2004-07-08 Ciba Specialty Chemicals Holding Inc. Synthesis of amines and intermediates for the synthesis thereof
JP3964417B2 (ja) * 2004-09-27 2007-08-22 国立大学法人金沢大学 インドール誘導体を有効成分とするα２受容体遮断剤及び血管拡張剤
JP5370957B2 (ja) * 2008-08-20 2013-12-18 学校法人日本大学 アポトーシス抑制剤

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