JP2013535424A5 - - Google Patents

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Publication number
JP2013535424A5
JP2013535424A5 JP2013518748A JP2013518748A JP2013535424A5 JP 2013535424 A5 JP2013535424 A5 JP 2013535424A5 JP 2013518748 A JP2013518748 A JP 2013518748A JP 2013518748 A JP2013518748 A JP 2013518748A JP 2013535424 A5 JP2013535424 A5 JP 2013535424A5
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JP
Japan
Prior art keywords
group
alkyl
compound according
aryl
alkoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2013518748A
Other languages
English (en)
Japanese (ja)
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JP2013535424A (ja
JP5922116B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2011/042729 external-priority patent/WO2012003414A1/en
Publication of JP2013535424A publication Critical patent/JP2013535424A/ja
Publication of JP2013535424A5 publication Critical patent/JP2013535424A5/ja
Application granted granted Critical
Publication of JP5922116B2 publication Critical patent/JP5922116B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2013518748A 2010-07-01 2011-07-01 複数のプロスタグランジン受容体で作用する全般的な抗炎症反応をもたらす化合物 Expired - Fee Related JP5922116B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US36075510P 2010-07-01 2010-07-01
US61/360,755 2010-07-01
PCT/US2011/042729 WO2012003414A1 (en) 2010-07-01 2011-07-01 Compounds act at multiple prostaglandin receptors giving a general anti-inflammatory response

Publications (3)

Publication Number Publication Date
JP2013535424A JP2013535424A (ja) 2013-09-12
JP2013535424A5 true JP2013535424A5 (https=) 2014-08-21
JP5922116B2 JP5922116B2 (ja) 2016-05-24

Family

ID=44514984

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013518748A Expired - Fee Related JP5922116B2 (ja) 2010-07-01 2011-07-01 複数のプロスタグランジン受容体で作用する全般的な抗炎症反応をもたらす化合物

Country Status (18)

Country Link
US (3) US8492424B2 (https=)
EP (1) EP2588459B1 (https=)
JP (1) JP5922116B2 (https=)
KR (1) KR20130141434A (https=)
CN (1) CN103038219B (https=)
AR (1) AR082073A1 (https=)
AU (1) AU2011272716B2 (https=)
BR (1) BR112013000065A2 (https=)
CA (1) CA2804194C (https=)
CL (1) CL2013000002A1 (https=)
CO (1) CO6680625A2 (https=)
ES (1) ES2625355T3 (https=)
MX (1) MX2013000170A (https=)
PH (1) PH12013500121A1 (https=)
RU (1) RU2013102967A (https=)
SG (1) SG186886A1 (https=)
TW (1) TW201206891A (https=)
WO (1) WO2012003414A1 (https=)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10206813B2 (en) 2009-05-18 2019-02-19 Dose Medical Corporation Implants with controlled drug delivery features and methods of using same
US12478503B2 (en) 2009-05-18 2025-11-25 Glaukos Corporation Implants with controlled drug delivery features and methods of using same
US8859606B2 (en) * 2010-07-01 2014-10-14 Allergan, Inc. Compounds act at multiple prostaglandin receptors giving a general anti-inflammatory response
US9006450B2 (en) 2010-07-01 2015-04-14 Boehringer Ingelheim International Gmbh Compounds, pharmaceutical compositions and uses thereof
AU2012358983B2 (en) * 2011-12-21 2017-09-14 Allergan, Inc. Compounds acting at multiple prostaglandin receptors giving a general anti-inflammatory response
US9035071B2 (en) * 2011-12-27 2015-05-19 Allergan, Inc. Compounds acting at multiple prostaglandin receptors giving a general anti-inflammatory response
CA2862266C (en) 2011-12-27 2016-10-04 Allergan, Inc. Compounds acting at multiple prostaglandin receptors giving a general anti-inflammatory response
WO2014028762A1 (en) 2012-08-15 2014-02-20 University Of Virginia Patent Foundation Compositions and methods for treating peripheral arterial disease
CA2898720A1 (en) * 2013-01-21 2014-07-24 Allergan, Inc. Compounds act at multiple prostaglandin receptors giving a general anti-inflammatory response
US9387196B2 (en) 2013-10-31 2016-07-12 Allergan, Inc. 3-{1-[5-chloro-2-(2-ethylbutoxy)benzyl]-5-methyl-1H-pyrazol-3-yl}propanoic acid in crystalline form and methods for use thereof
CN106146400A (zh) * 2015-03-20 2016-11-23 四川大学 苄基-1h-吡唑、苄基-1h-吡咯衍生物及其制备方法和用途
US10462745B2 (en) 2016-01-15 2019-10-29 Google Llc Systems and methods for extending battery life by monitoring device activity
CN107723304A (zh) * 2016-08-10 2018-02-23 中国科学院上海生命科学研究院 Prkar2a在炎症消退中的应用
WO2020113094A1 (en) 2018-11-30 2020-06-04 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4166452A (en) 1976-05-03 1979-09-04 Generales Constantine D J Jr Apparatus for testing human responses to stimuli
US4256108A (en) 1977-04-07 1981-03-17 Alza Corporation Microporous-semipermeable laminated osmotic system
US4265874A (en) 1980-04-25 1981-05-05 Alza Corporation Method of delivering drug with aid of effervescent activity generated in environment of use
US4826868A (en) * 1986-05-29 1989-05-02 Ortho Pharmaceutical Corporation 1,5-Diaryl-3-substituted pyrazoles pharmaceutical compositions and use
US7273883B2 (en) 2000-09-14 2007-09-25 Allergan, Inc. Prostaglandin EP4 antagonist
US7217725B2 (en) 2000-09-14 2007-05-15 Allergan, Inc. Prostaglandin D2 antagonist
US6511999B2 (en) 2000-09-14 2003-01-28 Allergan, Inc. Interheteroaryl 7-oxabicyclic [2.2.1]heptane oxazoles as prostaglandin F2α antagonists
AU2004240705A1 (en) * 2003-05-20 2004-12-02 Merck Frosst Canada & Co. Fluoro-methanesulfonyl-substituted cycloalkanoindoles and their use as prostaglandin D2 antagonists
ES2298832T3 (es) * 2003-10-24 2008-05-16 Glaxo Group Limited Compuestos heterociclicos.
GB0508472D0 (en) 2005-04-26 2005-06-01 Glaxo Group Ltd Compounds

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