JP2013544811A5 - - Google Patents

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Publication number
JP2013544811A5
JP2013544811A5 JP2013537774A JP2013537774A JP2013544811A5 JP 2013544811 A5 JP2013544811 A5 JP 2013544811A5 JP 2013537774 A JP2013537774 A JP 2013537774A JP 2013537774 A JP2013537774 A JP 2013537774A JP 2013544811 A5 JP2013544811 A5 JP 2013544811A5
Authority
JP
Japan
Prior art keywords
phenyl
isoxazol
trifluoromethyl
chroman
oxadiazol
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP2013537774A
Other languages
English (en)
Japanese (ja)
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JP2013544811A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2011/058891 external-priority patent/WO2012061459A1/en
Publication of JP2013544811A publication Critical patent/JP2013544811A/ja
Publication of JP2013544811A5 publication Critical patent/JP2013544811A5/ja
Ceased legal-status Critical Current

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JP2013537774A 2010-11-03 2011-11-02 自己免疫疾患および血管疾患の治療用のs1p1アゴニストとしての複素環式化合物 Ceased JP2013544811A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US40968210P 2010-11-03 2010-11-03
US61/409,682 2010-11-03
PCT/US2011/058891 WO2012061459A1 (en) 2010-11-03 2011-11-02 Heterocyclic compounds as s1p1 agonists for the treatment of autoimmune and vascular diseases

Publications (2)

Publication Number Publication Date
JP2013544811A JP2013544811A (ja) 2013-12-19
JP2013544811A5 true JP2013544811A5 (https=) 2014-11-06

Family

ID=44983720

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013537774A Ceased JP2013544811A (ja) 2010-11-03 2011-11-02 自己免疫疾患および血管疾患の治療用のs1p1アゴニストとしての複素環式化合物

Country Status (6)

Country Link
US (1) US8629282B2 (https=)
EP (1) EP2635573B1 (https=)
JP (1) JP2013544811A (https=)
CN (1) CN103298807A (https=)
ES (1) ES2525298T3 (https=)
WO (1) WO2012061459A1 (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5788507B2 (ja) 2010-07-20 2015-09-30 ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company 置換3−フェニル−1,2,4−オキサジアゾール化合物
EP2619190B1 (en) 2010-09-24 2015-08-12 Bristol-Myers Squibb Company Substituted oxadiazole compounds and their use as s1p1 agonists
TWI613182B (zh) 2013-02-21 2018-02-01 必治妥美雅史谷比公司 雙環化合物
TWI689487B (zh) 2014-08-20 2020-04-01 美商必治妥美雅史谷比公司 經取代雙環化合物
ES2877686T3 (es) 2016-07-22 2021-11-17 Shijiazhuang Sagacity New Drug Dev Co Ltd Agonista S1P1 y aplicación del mismo
IL271149B2 (en) 2017-06-14 2024-05-01 Trevena Inc Compounds for modulating s1p1 activity and methods of using the same
KR20200128386A (ko) * 2018-01-18 2020-11-12 스자좡 서개시티 뉴 드러그 디벨롭먼트 컴퍼니, 엘티디. 트리사이클릭 화합물의 결정형 및 염 형태, 및 이의 제조방법
EP4061352A4 (en) * 2019-11-19 2024-02-28 Trevena, Inc. COMPOUNDS AND METHODS FOR PRODUCING S1P1-MODULATING COMPOUNDS
JP2023502355A (ja) * 2019-11-20 2023-01-24 アリーナ ファーマシューティカルズ, インコーポレイテッド S1p1受容体に関連する状態を処置する方法

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JP5788507B2 (ja) 2010-07-20 2015-09-30 ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company 置換3−フェニル−1,2,4−オキサジアゾール化合物
EP2619190B1 (en) 2010-09-24 2015-08-12 Bristol-Myers Squibb Company Substituted oxadiazole compounds and their use as s1p1 agonists

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