JP2013513596A - 造血細胞キナーゼ(p59−HCK)の阻害剤およびインフルエンザ感染の処置におけるそれらの使用 - Google Patents

造血細胞キナーゼ(p59−HCK)の阻害剤およびインフルエンザ感染の処置におけるそれらの使用 Download PDF

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JP2013513596A
JP2013513596A JP2012542622A JP2012542622A JP2013513596A JP 2013513596 A JP2013513596 A JP 2013513596A JP 2012542622 A JP2012542622 A JP 2012542622A JP 2012542622 A JP2012542622 A JP 2012542622A JP 2013513596 A JP2013513596 A JP 2013513596A
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シヤロン,キヤサリン・エリザベス
フエントン,ロバート
クロウ,スコツト
一洋 伊藤
ストロング,ピーター
ラペポート,ウイリアム・ガース
キース レイ,
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レスピバート・リミテツド
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    • AHUMAN NECESSITIES
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • A61K31/41551,2-Diazoles non condensed and containing further heterocyclic rings
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    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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JP2012542622A 2009-12-11 2010-12-10 造血細胞キナーゼ(p59−HCK)の阻害剤およびインフルエンザ感染の処置におけるそれらの使用 Pending JP2013513596A (ja)

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GB0921730.8 2009-12-11
GBGB0921730.8A GB0921730D0 (en) 2009-12-11 2009-12-11 Method of treatment
PCT/GB2010/052067 WO2011070369A1 (en) 2009-12-11 2010-12-10 Inhibitors of hemopoietic cell kinase (p59-hck) and their use in the treatment of influenza infection

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JP2016017330A Division JP6247709B2 (ja) 2009-12-11 2016-02-01 造血細胞キナーゼ(p59−HCK)の阻害剤およびインフルエンザ感染の処置におけるそれらの使用

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JP2016017330A Active JP6247709B2 (ja) 2009-12-11 2016-02-01 造血細胞キナーゼ(p59−HCK)の阻害剤およびインフルエンザ感染の処置におけるそれらの使用

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EP (1) EP2509595B1 (enExample)
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AU (1) AU2010329645B2 (enExample)
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GB0905955D0 (en) 2009-04-06 2009-05-20 Respivert Ltd Novel compounds
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JP5787977B2 (ja) 2010-04-08 2015-09-30 レスピバート・リミテツド P38mapキナーゼ阻害剤
US9260410B2 (en) 2010-04-08 2016-02-16 Respivert Ltd. P38 MAP kinase inhibitors
EP2582700B1 (en) 2010-06-17 2016-11-02 Respivert Limited Respiratory formulations containing p38 mapk inhibitors
GB201010193D0 (en) 2010-06-17 2010-07-21 Respivert Ltd Medicinal use
PT2763984T (pt) 2011-10-03 2016-07-25 Respivert Ltd 1-pirazolil-3-(4-((2-anilinopirimidin-4-il)oxi)naftalen-1-il) ureias como inibidores da map cinase p38
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GB201215357D0 (en) 2012-08-29 2012-10-10 Respivert Ltd Compounds
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JP2016128489A (ja) 2016-07-14
GB0921730D0 (en) 2010-01-27
WO2011070369A1 (en) 2011-06-16
US20180000830A1 (en) 2018-01-04
AU2010329645B2 (en) 2015-05-28
CN102762204B (zh) 2014-11-19
US20160045512A1 (en) 2016-02-18
US20120244120A1 (en) 2012-09-27
JP6247709B2 (ja) 2017-12-13
CN102762204A (zh) 2012-10-31
EP2509595A1 (en) 2012-10-17
EP2509595B1 (en) 2018-04-11

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