JP2012513982A5 - - Google Patents
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- Publication number
- JP2012513982A5 JP2012513982A5 JP2011543072A JP2011543072A JP2012513982A5 JP 2012513982 A5 JP2012513982 A5 JP 2012513982A5 JP 2011543072 A JP2011543072 A JP 2011543072A JP 2011543072 A JP2011543072 A JP 2011543072A JP 2012513982 A5 JP2012513982 A5 JP 2012513982A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- optionally substituted
- alkyl group
- aromatic
- atom
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US20388708P | 2008-12-29 | 2008-12-29 | |
| US61/203,887 | 2008-12-29 | ||
| PCT/JP2009/071919 WO2010076896A1 (en) | 2008-12-29 | 2009-12-28 | Prophylactic/therapeutic agent for cancer |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2012513982A JP2012513982A (ja) | 2012-06-21 |
| JP2012513982A5 true JP2012513982A5 (enExample) | 2013-01-31 |
Family
ID=42025816
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011543072A Pending JP2012513982A (ja) | 2008-12-29 | 2009-12-28 | 癌の予防・治療剤 |
Country Status (26)
| Country | Link |
|---|---|
| US (1) | US20110312898A1 (enExample) |
| EP (1) | EP2379053A1 (enExample) |
| JP (1) | JP2012513982A (enExample) |
| KR (1) | KR20110111420A (enExample) |
| CN (1) | CN102333520B (enExample) |
| AR (1) | AR074918A1 (enExample) |
| AU (1) | AU2009334235A1 (enExample) |
| BR (1) | BRPI0923663A2 (enExample) |
| CA (1) | CA2748517A1 (enExample) |
| CL (1) | CL2011001519A1 (enExample) |
| CO (1) | CO6382105A2 (enExample) |
| CR (1) | CR20110374A (enExample) |
| DO (1) | DOP2011000163A (enExample) |
| EA (1) | EA019738B1 (enExample) |
| EC (1) | ECSP11011166A (enExample) |
| GE (1) | GEP20146001B (enExample) |
| IL (1) | IL212913A0 (enExample) |
| MA (1) | MA32935B1 (enExample) |
| MX (1) | MX2011006170A (enExample) |
| NZ (1) | NZ593381A (enExample) |
| PE (1) | PE20110939A1 (enExample) |
| TN (1) | TN2011000250A1 (enExample) |
| TW (1) | TW201029660A (enExample) |
| UY (1) | UY32367A (enExample) |
| WO (1) | WO2010076896A1 (enExample) |
| ZA (1) | ZA201103627B (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8592379B2 (en) * | 2008-04-30 | 2013-11-26 | Kyoto University | Metastin derivative and use thereof |
| CN107412725A (zh) * | 2009-12-22 | 2017-12-01 | 武田药品工业株式会社 | 缓释制剂 |
| US20130210742A1 (en) * | 2010-06-25 | 2013-08-15 | Takeda Pharmaceutical Company Limited | Sustained-release formulation |
| JP6253146B2 (ja) * | 2014-02-04 | 2017-12-27 | 国立大学法人山口大学 | 新規なペプチド誘導体及びこれを含有する医薬 |
| WO2016099232A2 (ru) * | 2014-10-20 | 2016-06-23 | Товарищество С Ограниченной Ответственностью "Фармацевтическая Компания "Ромат" | Фармацевтический состав лечебно-профилактического действия и способ его приготовления |
| TWI855377B (zh) | 2016-09-30 | 2024-09-11 | 瑞士商麥歐文科學有限公司 | 治療女性不孕症之方法 |
| WO2024206577A1 (en) * | 2023-03-28 | 2024-10-03 | Radionetics Oncology, Inc. | Kisspeptin receptor (kiss1r) targeted therapeutics and uses thereof |
| WO2025217074A1 (en) | 2024-04-08 | 2025-10-16 | Radionetics Oncology, Inc. | Kisspeptin receptor (kiss1r) targeted therapeutics and uses thereof |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2003292696A1 (en) * | 2002-12-26 | 2004-08-10 | Takeda Pharmaceutical Company Limited | Metastin derivative and use thereof |
| US6800611B2 (en) * | 2003-01-06 | 2004-10-05 | Takeda Chemical Industries, Ltd. | Metastin derivatives and their use |
| BRPI0512397A (pt) * | 2004-06-25 | 2008-03-04 | Takeda Pharmaceutical | composto,produto farmacêutico, métodos para suprimir a metástase de cáncer ou o crescimento do cáncer, para prevenir ou tratar uma doença ou condição, para controlar a função placentária, para melhorar a função gonadal, para induzir ou estimular a ovulação, para promover a secreção do hormÈnio gonadotrópico ou promover a secreção do hormÈnio sexual, para suprimir a secreção do hormÈnio gonadotrópico ou suprimir a secreção do hormÈnio sexual, para infra regular hormÈnio gonadrotópico ou hormÈnio sexual, e a proteìna ot7t175 humana, e para realçar a estabilidade no sangue, uso do composto, e, agente para suprimir a secreção do hormÈnio gonadotrópico ou um agente para suprimir a secreção do hormÈnio sexual |
| CN1972959A (zh) * | 2004-06-25 | 2007-05-30 | 武田药品工业株式会社 | 转移素衍生物及其用途 |
| AR058584A1 (es) * | 2005-12-22 | 2008-02-13 | Takeda Pharmaceutical | Derivados de metastina y uso de los mismos |
-
2009
- 2009-12-28 KR KR1020117017317A patent/KR20110111420A/ko not_active Withdrawn
- 2009-12-28 TW TW098145251A patent/TW201029660A/zh unknown
- 2009-12-28 MA MA33959A patent/MA32935B1/fr unknown
- 2009-12-28 AU AU2009334235A patent/AU2009334235A1/en not_active Abandoned
- 2009-12-28 BR BRPI0923663A patent/BRPI0923663A2/pt not_active IP Right Cessation
- 2009-12-28 PE PE2011001293A patent/PE20110939A1/es not_active Application Discontinuation
- 2009-12-28 WO PCT/JP2009/071919 patent/WO2010076896A1/en not_active Ceased
- 2009-12-28 AR ARP090105129A patent/AR074918A1/es not_active Application Discontinuation
- 2009-12-28 CA CA2748517A patent/CA2748517A1/en not_active Abandoned
- 2009-12-28 EP EP09801574A patent/EP2379053A1/en not_active Withdrawn
- 2009-12-28 NZ NZ593381A patent/NZ593381A/xx not_active IP Right Cessation
- 2009-12-28 CN CN2009801575361A patent/CN102333520B/zh not_active Expired - Fee Related
- 2009-12-28 EA EA201100882A patent/EA019738B1/ru not_active IP Right Cessation
- 2009-12-28 JP JP2011543072A patent/JP2012513982A/ja active Pending
- 2009-12-28 UY UY0001032367A patent/UY32367A/es not_active Application Discontinuation
- 2009-12-28 US US13/142,414 patent/US20110312898A1/en not_active Abandoned
- 2009-12-28 MX MX2011006170A patent/MX2011006170A/es not_active Application Discontinuation
- 2009-12-28 GE GEAP200912275A patent/GEP20146001B/en unknown
-
2011
- 2011-05-16 IL IL212913A patent/IL212913A0/en unknown
- 2011-05-17 TN TN2011000250A patent/TN2011000250A1/fr unknown
- 2011-05-17 ZA ZA2011/03627A patent/ZA201103627B/en unknown
- 2011-05-31 DO DO2011000163A patent/DOP2011000163A/es unknown
- 2011-06-20 CL CL2011001519A patent/CL2011001519A1/es unknown
- 2011-06-23 CO CO11078830A patent/CO6382105A2/es not_active Application Discontinuation
- 2011-06-29 EC EC2011011166A patent/ECSP11011166A/es unknown
- 2011-06-29 CR CR20110374A patent/CR20110374A/es not_active Application Discontinuation
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