JP2011527677A - Ｎｈｅ−１阻害剤として有用なピロリジニル及びピペリジニル化合物 - Google Patents

Ｎｈｅ−１阻害剤として有用なピロリジニル及びピペリジニル化合物 Download PDF

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JP2011527677A
JP2011527677A JP2011517461A JP2011517461A JP2011527677A JP 2011527677 A JP2011527677 A JP 2011527677A JP 2011517461 A JP2011517461 A JP 2011517461A JP 2011517461 A JP2011517461 A JP 2011517461A JP 2011527677 A JP2011527677 A JP 2011527677A
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JP2011527677A5 (enExample
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ベントツィーン，イェルク・マルティン
ボイヤー，スティーヴン・ジェームズ
バーク，ジェニファー
エルドラプ，アンネ・ベッティーナ
グオ，シン
ヒューバー，ジョン・デヴィッド
カーレーン，トーマス・マーティン
ソリマンザデー，ファリバ
スウィナマー，アラン・デヴィッド
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ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
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    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/34—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • C07D471/04—Ortho-condensed systems

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JP2011517461A 2008-07-08 2009-06-24 Ｎｈｅ−１阻害剤として有用なピロリジニル及びピペリジニル化合物 Pending JP2011527677A (ja)

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