JP2011521896A - 免疫関連障害に対する局部治療に使用するための局所lfa−1アンタゴニスト - Google Patents

免疫関連障害に対する局部治療に使用するための局所lfa−1アンタゴニスト Download PDF

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JP2011521896A
JP2011521896A JP2011505028A JP2011505028A JP2011521896A JP 2011521896 A JP2011521896 A JP 2011521896A JP 2011505028 A JP2011505028 A JP 2011505028A JP 2011505028 A JP2011505028 A JP 2011505028A JP 2011521896 A JP2011521896 A JP 2011521896A
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lfa
antagonist
formulation
aryl
heteroaryl
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ジョン バーニアー,
トーマス ガデック,
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サーコード コーポレイション
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    • C07D405/06Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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JP2011505028A 2008-04-15 2009-04-15 免疫関連障害に対する局部治療に使用するための局所lfa−1アンタゴニスト Withdrawn JP2011521896A (ja)

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US4524008P 2008-04-15 2008-04-15
US61/045,240 2008-04-15
PCT/US2009/002389 WO2009128934A1 (en) 2008-04-15 2009-04-15 Topical lfa-1 antagonists for use in localized treatment of immune related disorders

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JP2014080832A Division JP2014132032A (ja) 2008-04-15 2014-04-10 免疫関連障害に対する局部治療に使用するための局所lfa−1アンタゴニスト

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JP2011521896A true JP2011521896A (ja) 2011-07-28
JP2011521896A5 JP2011521896A5 (https=) 2012-06-07

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JP2011505028A Withdrawn JP2011521896A (ja) 2008-04-15 2009-04-15 免疫関連障害に対する局部治療に使用するための局所lfa−1アンタゴニスト
JP2014080832A Pending JP2014132032A (ja) 2008-04-15 2014-04-10 免疫関連障害に対する局部治療に使用するための局所lfa−1アンタゴニスト

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US (2) US20090258070A1 (https=)
EP (2) EP3632444A3 (https=)
JP (2) JP2011521896A (https=)
CN (1) CN102056485A (https=)
ES (1) ES2763703T3 (https=)
WO (1) WO2009128934A1 (https=)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2011516607A (ja) * 2008-04-15 2011-05-26 サーコード コーポレイション 胃腸系へのlfa−1アンタゴニストの送達
JP2011518155A (ja) * 2008-04-15 2011-06-23 サーコード コーポレイション 免疫関連障害の局所治療に使用するためのエアゾール化lfa−1アンタゴニスト
JP2022546120A (ja) * 2019-09-03 2022-11-02 スクエア パワー リミテッド セリアック病の予防および治療に使用するためのレバミピド
WO2024058212A1 (ja) * 2022-09-15 2024-03-21 日油株式会社 コンタクトレンズ用溶液

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US8193232B2 (en) * 2009-02-13 2012-06-05 Topica Pharmaceuticals, Inc. Anti-fungal formulation
JP2013516459A (ja) * 2010-01-20 2013-05-13 カディラ・ヘルスケア・リミテッド ピタバスタチン及び医薬として許容可能なそれらの塩の製造方法
EP2582391B1 (en) * 2010-06-18 2018-10-03 XBiotech, Inc Arthritis treatment
KR101910760B1 (ko) 2010-08-23 2018-10-22 엑스바이오테크, 인크. 종양성 질병들에 대한 치료
US9724409B2 (en) 2011-04-01 2017-08-08 Xbiotech, Inc. Treatment of inflammatory skin disease
CN108404127B (zh) 2011-09-23 2025-12-12 埃克斯生物科技公司 恶病质治疗
WO2013108644A1 (ja) * 2012-01-20 2013-07-25 京都府公立大学法人 レバミピドのアレルギー性結膜炎治療剤
US9545441B2 (en) 2012-09-18 2017-01-17 Xbiotech, Inc. Treatment of diabetes
BR112015014367B1 (pt) 2012-12-19 2022-11-22 Novartis Ag Composição inibidora de lfa-1, método para estabilizar a dita composição e uso da mesma para tratar uma doença ocular
US9688943B2 (en) 2015-05-29 2017-06-27 beauty Avenues LLC Candle containing non-ionic emulsifer
AU2017376961A1 (en) * 2016-12-16 2019-06-27 Novartis Ag Ocular distribution and pharmacokinetics of lifitegrast formulations
EP3582813A4 (en) 2017-02-16 2020-12-30 XBiotech, Inc TREATMENT OF SUPPURATIVE HIDRADENITIS
CN106920239B (zh) * 2017-03-08 2019-10-18 福建师范大学 一种基于改进sift算法的图像关键点检测方法
WO2019065936A1 (ja) * 2017-09-29 2019-04-04 参天製薬株式会社 涙液中のmuc5ac量の測定方法
WO2019108814A1 (en) * 2017-11-29 2019-06-06 The Rockefeller University Combination of local and systemic therapies for enhanced treatment of dermatologic conditions
JP7700045B2 (ja) * 2019-04-18 2025-06-30 アズーラ オフサルミックス エルティーディー. 眼障害を処置するための化合物および方法
AU2020315758B2 (en) 2019-07-16 2024-08-01 Donaghys Limited Transdermal solvent system and methods of use
CN112494488B (zh) * 2020-06-17 2022-01-18 中国药科大学 瑞巴派特的防脱发和生发用途
CA3095679A1 (en) 2020-10-07 2022-04-07 Xbiotech Inc. True human antibody specific for interleuken 1 alpha (il-1a)
CA3095676A1 (en) 2020-10-07 2022-04-07 Xbiotech Inc. True human antibody specific for interleukin 1 alpha (il-1a)
CA3095740A1 (en) 2020-10-07 2022-04-07 Xbiotech Inc. True human antibody specific for interleukin alpha (il-1a)
CA3095675A1 (en) 2020-10-07 2022-04-07 Xbiotech Inc. True human antibody specific for interleukin 1 alpha (il-1a)
US12393057B2 (en) 2020-12-15 2025-08-19 Coopervision International Limited Oleic acid-releasing contact lens
EP4271370A4 (en) * 2020-12-29 2024-12-04 Next Science IP Holdings Pty Ltd COMPOSITION AND METHOD FOR CANCER TREATMENT
US20240189245A1 (en) * 2021-06-14 2024-06-13 Protransit Nanotherapy Llc Cyclosporine compositions and methods of use thereof
CN115707698A (zh) * 2021-08-18 2023-02-21 辽宁何氏医学院 5,7-二氯-1,2,3,4-四氢异喹啉-6-甲酰胺类化合物及其制备方法和应用
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WO2025223511A1 (zh) * 2024-04-25 2025-10-30 上海翊石医药科技有限公司 一类苯甲酰基甘氨酸衍生物及其制备方法和应用

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005044817A1 (en) * 2003-11-05 2005-05-19 Sunesis Pharmaceuticals, Inc. Modulators of cellular adhesion
WO2006125119A1 (en) * 2005-05-17 2006-11-23 Sarcode Corporation Compositions and methods for treatment of eye disorders
JP2011516607A (ja) * 2008-04-15 2011-05-26 サーコード コーポレイション 胃腸系へのlfa−1アンタゴニストの送達
JP2011518155A (ja) * 2008-04-15 2011-06-23 サーコード コーポレイション 免疫関連障害の局所治療に使用するためのエアゾール化lfa−1アンタゴニスト

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